ATE293970T1 - Lipasehemmer enthaltende pharmazeutische zusammensetzungen - Google Patents

Lipasehemmer enthaltende pharmazeutische zusammensetzungen

Info

Publication number
ATE293970T1
ATE293970T1 AT99940127T AT99940127T ATE293970T1 AT E293970 T1 ATE293970 T1 AT E293970T1 AT 99940127 T AT99940127 T AT 99940127T AT 99940127 T AT99940127 T AT 99940127T AT E293970 T1 ATE293970 T1 AT E293970T1
Authority
AT
Austria
Prior art keywords
pharmaceutical compositions
compositions containing
lipase inhibitors
containing lipase
inhibitors
Prior art date
Application number
AT99940127T
Other languages
English (en)
Inventor
Manuela Hug
Hans-Peter Maerki
Marcel Meier
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Application granted granted Critical
Publication of ATE293970T1 publication Critical patent/ATE293970T1/de

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/365Lactones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0087Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Zoology (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Child & Adolescent Psychology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Jellies, Jams, And Syrups (AREA)
  • General Preparation And Processing Of Foods (AREA)
AT99940127T 1998-08-14 1999-08-02 Lipasehemmer enthaltende pharmazeutische zusammensetzungen ATE293970T1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP98115311 1998-08-14
EP99109516 1999-05-12
PCT/EP1999/005607 WO2000009122A1 (en) 1998-08-14 1999-08-02 Pharmaceutical compositions containing lipase inhibitors

Publications (1)

Publication Number Publication Date
ATE293970T1 true ATE293970T1 (de) 2005-05-15

Family

ID=26149537

Family Applications (1)

Application Number Title Priority Date Filing Date
AT99940127T ATE293970T1 (de) 1998-08-14 1999-08-02 Lipasehemmer enthaltende pharmazeutische zusammensetzungen

Country Status (19)

Country Link
US (1) US6358522B1 (de)
EP (1) EP1105122B1 (de)
JP (1) JP3774118B2 (de)
KR (1) KR20010079635A (de)
CN (1) CN1170534C (de)
AR (1) AR035001A1 (de)
AT (1) ATE293970T1 (de)
AU (1) AU761351B2 (de)
BR (1) BR9912980B1 (de)
CA (1) CA2340056C (de)
CO (1) CO5130009A1 (de)
DE (1) DE69924999T2 (de)
DK (1) DK1105122T3 (de)
ES (1) ES2242413T3 (de)
MA (1) MA26671A1 (de)
PE (1) PE20000953A1 (de)
PT (1) PT1105122E (de)
TR (1) TR200100471T2 (de)
WO (1) WO2000009122A1 (de)

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AR025609A1 (es) 1999-09-13 2002-12-04 Hoffmann La Roche Formulaciones lipidas solidas
AR025587A1 (es) 1999-09-13 2002-12-04 Hoffmann La Roche Formulaciones en dispersion que contienen inhibidores de lipasa
EP1132389A1 (de) 2000-03-06 2001-09-12 Vernalis Research Limited Neue Azaindolyl-Derivate für die Behandlung von Fettleibigheit
PT1296656E (pt) 2000-06-27 2006-12-29 Hoffmann La Roche Processo para a preparação de uma composição
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EP1307263B1 (de) 2000-07-28 2005-04-20 F. Hoffmann-La Roche Ag Neue verwendung von lipase-inhibitoren
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GB0106177D0 (en) 2001-03-13 2001-05-02 Hoffmann La Roche Piperazine derivatives
AU2002338896B2 (en) 2001-05-21 2006-04-27 F.Hoffman-La Roche Ag Quinoline derivatives as ligands for the neuropeptide Y receptor
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US7041280B2 (en) * 2001-06-29 2006-05-09 Genzyme Corporation Aryl boronate functionalized polymers for treating obesity
US7049345B2 (en) * 2001-06-29 2006-05-23 Genzyme Corporation Fat-binding polymers
US6787558B2 (en) 2001-09-28 2004-09-07 Hoffmann-La Roche Inc. Quinoline derivatives
GB0202015D0 (en) 2002-01-29 2002-03-13 Hoffmann La Roche Piperazine Derivatives
KR100659428B1 (ko) 2002-02-04 2006-12-19 에프. 호프만-라 로슈 아게 Npy 길항제로서의 퀴놀린 유도체
KR100611854B1 (ko) 2002-02-28 2006-08-11 에프. 호프만-라 로슈 아게 신경 펩타이드 y(npy) 수용체 길항제로서의 티아졸유도체
WO2003090742A1 (en) * 2002-04-26 2003-11-06 F. Hoffmann-La Roche Ag Pharmaceutical composition comprising a lipase inhibitor and glucomannan
EP1560816A1 (de) 2002-07-05 2005-08-10 F. Hoffmann-La Roche Ag Chinazoline derivate
EP1539722A1 (de) 2002-08-07 2005-06-15 F. Hoffmann-La Roche Ag Thiazolderivate
EP1539746B1 (de) 2002-09-12 2006-11-15 F. Hoffmann-La Roche Ag N-substituierte-1h-indol-5-propansäure verbindungen als ppar-agonisten zur behandlung von diabetis
MXPA05005445A (es) 2002-11-25 2005-08-26 Hoffmann La Roche Derivados de indolilo.
US8372430B2 (en) * 2002-12-17 2013-02-12 The Procter & Gamble Company Compositions, methods, and kits useful for the alleviation of gastrointestinal effects
GB0314967D0 (en) 2003-06-26 2003-07-30 Hoffmann La Roche Piperazine derivatives
WO2005014592A1 (en) 2003-08-12 2005-02-17 F. Hoffmann-La Roche Ag 2-amino-5-benzoylthiazole npy antagonists
WO2005014593A1 (en) 2003-08-12 2005-02-17 F. Hoffmann-La Roche Ag Thiazole derivatives as npy antagonists
KR100895758B1 (ko) 2005-05-03 2009-04-30 에프. 호프만-라 로슈 아게 5-ht2 리간드로서 테트라사이클릭 아자피라지노인돌린
PL1897558T3 (pl) * 2005-06-09 2014-01-31 Norgine Bv Stały preparat 2-heksadecyloksy-6-metylo-4H-3,1-benzoksazyn-4-onu
JP2009504707A (ja) 2005-08-18 2009-02-05 エフ.ホフマン−ラ ロシュ アーゲー H3受容体調節剤として有用なチアゾリルピペリジン誘導体
BRPI0619268A2 (pt) 2005-11-30 2011-09-20 Hoffmann La Roche compostos, processo para a sua manufatura, composições farmacêuticas, método para o tratamento e/ou prevenção de enfermidades que estão associadas com a modulação de receptores de h3, uso dos compostos e método para o tratamento ou prevenção de obesidade e de diabetes do tipo ii em um ser humano ou animal
EP1968967B1 (de) 2005-11-30 2011-04-27 F. Hoffmann-La Roche AG 1,1-dioxo-thiomorpholinyl-indolyl-methanon-derivate zur verwendung als h3-modulatoren
ATE466007T1 (de) 2005-11-30 2010-05-15 Hoffmann La Roche 5-substituierte indol-2-carbonsäureamidderivate
US7579351B2 (en) 2005-12-09 2009-08-25 Hoffmann-La Roche Inc. Tricyclic amide derivatives
ES2334580T3 (es) 2005-12-15 2010-03-12 F. Hoffmann-La Roche Ag Derivados de pirrolo(2,3-c)piridina.
AU2006326067A1 (en) 2005-12-16 2007-06-21 F. Hoffmann-La Roche Ag Pyrrolo [2 , 3-b] pyridine derivatives as H3 receptor modulators
US7432255B2 (en) 2006-05-16 2008-10-07 Hoffmann-La Roche Inc. 1H-indol-5-yl-piperazin-1-yl-methanone derivatives
AU2007267184A1 (en) 2006-05-30 2007-12-06 F. Hoffmann-La Roche Ag Piperidinyl pyrimidine derivatives
US7514433B2 (en) 2006-08-03 2009-04-07 Hoffmann-La Roche Inc. 1H-indole-6-yl-piperazin-1-yl-methanone derivatives
US20080146559A1 (en) 2006-12-08 2008-06-19 Li Chen 4,5,6,7-Tetrahydro-Thieno [2,3-C] Pyridine Derivatives
ES2623411T3 (es) * 2007-05-16 2017-07-11 Buckman Laboratories International, Inc. Métodos para controlar los contaminantes orgánicos en fibras
US7534788B2 (en) 2007-07-25 2009-05-19 Hoffmann-La Roche Inc. Benzofuran and benzothiophene-2-carboxylic acid amide derivatives
WO2009044380A2 (en) 2007-10-05 2009-04-09 Ranbaxy Laboratories Limited Formulations containing orlistat particles having controlled particle size
EP2219614A1 (de) * 2007-10-15 2010-08-25 Inventis DDS Pvt Limited Pharmazeutische zusammensetzung von orlistat
PL216542B1 (pl) 2008-03-20 2014-04-30 Zakłady Farmaceutyczne POLPHARMA Spółka Akcyjna Sposób wytwarzania stabilnej kompozycji orlistatu w postaci kapsułkowanego proszku
US8309107B2 (en) 2008-10-06 2012-11-13 Banner Pharmacaps, Inc. Stable solutions of orlistat for pharmaceutical dosage forms
GB201122213D0 (en) * 2011-12-23 2012-02-01 Norgine Bv Compositions
CN104546768B (zh) * 2014-12-30 2017-06-16 重庆植恩药业有限公司 含有脂肪酶抑制剂的咀嚼片组合物及其制备方法
MX386290B (es) * 2016-06-17 2025-03-18 Procter & Gamble Composicion masticable blanda que comprende psyllium
CN112220831A (zh) * 2020-08-07 2021-01-15 天津盛实百草中药科技有限公司 圆苞车前子壳粉在缓解奥利司他副作用中的应用

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US4005195A (en) * 1976-02-12 1977-01-25 The Procter & Gamble Company Compositions for treating hypercholesterolemia
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TW381025B (en) * 1993-08-05 2000-02-01 Hoffmann La Roche Pharmaceutical composition containing a glucosidase inhibitor and a lipase inhibitor
JPH09252746A (ja) * 1996-03-22 1997-09-30 Nippon Kankyo Yakuhin Kk 栄養補助食品
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Also Published As

Publication number Publication date
US6358522B1 (en) 2002-03-19
JP3774118B2 (ja) 2006-05-10
PE20000953A1 (es) 2000-09-26
WO2000009122A1 (en) 2000-02-24
BR9912980B1 (pt) 2013-10-22
AU5418599A (en) 2000-03-06
CA2340056A1 (en) 2000-02-24
AU761351B2 (en) 2003-06-05
MA26671A1 (fr) 2004-12-20
CN1170534C (zh) 2004-10-13
EP1105122B1 (de) 2005-04-27
AR035001A1 (es) 2004-04-14
CN1312713A (zh) 2001-09-12
DE69924999D1 (de) 2005-06-02
JP2002522491A (ja) 2002-07-23
ES2242413T3 (es) 2005-11-01
CA2340056C (en) 2007-01-09
KR20010079635A (ko) 2001-08-22
BR9912980A (pt) 2001-05-08
DK1105122T3 (da) 2005-08-08
PT1105122E (pt) 2005-08-31
CO5130009A1 (es) 2002-02-27
EP1105122A1 (de) 2001-06-13
DE69924999T2 (de) 2006-05-04
TR200100471T2 (tr) 2001-07-23

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