ATE268771T1 - Verfahren zur herstellung von pyrazolopyridinderivaten - Google Patents

Verfahren zur herstellung von pyrazolopyridinderivaten

Info

Publication number
ATE268771T1
ATE268771T1 AT01932738T AT01932738T ATE268771T1 AT E268771 T1 ATE268771 T1 AT E268771T1 AT 01932738 T AT01932738 T AT 01932738T AT 01932738 T AT01932738 T AT 01932738T AT E268771 T1 ATE268771 T1 AT E268771T1
Authority
AT
Austria
Prior art keywords
6alkyl
6alkoxy
substituted
fluorine atoms
halogen
Prior art date
Application number
AT01932738T
Other languages
English (en)
Inventor
Russ N Fitzgerald
David Kendall Jung
John F Eaddy
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Application granted granted Critical
Publication of ATE268771T1 publication Critical patent/ATE268771T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Rheumatology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
AT01932738T 2000-04-28 2001-04-27 Verfahren zur herstellung von pyrazolopyridinderivaten ATE268771T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US20040000P 2000-04-28 2000-04-28
PCT/US2001/013801 WO2001083479A2 (en) 2000-04-28 2001-04-27 Process for the preparation of pyrazolopyridine derivatives

Publications (1)

Publication Number Publication Date
ATE268771T1 true ATE268771T1 (de) 2004-06-15

Family

ID=22741567

Family Applications (1)

Application Number Title Priority Date Filing Date
AT01932738T ATE268771T1 (de) 2000-04-28 2001-04-27 Verfahren zur herstellung von pyrazolopyridinderivaten

Country Status (7)

Country Link
EP (1) EP1276742B1 (de)
JP (1) JP2003531906A (de)
AT (1) ATE268771T1 (de)
AU (1) AU2001259242A1 (de)
DE (1) DE60103752T2 (de)
ES (1) ES2222372T3 (de)
WO (1) WO2001083479A2 (de)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE325115T1 (de) 2002-08-19 2006-06-15 Glaxo Group Ltd Pyrimidinderivate als selektive cox-2-inhibitoren
GB0221443D0 (en) 2002-09-16 2002-10-23 Glaxo Group Ltd Pyridine derivates
UA103319C2 (en) 2008-05-06 2013-10-10 Глаксосмитклайн Ллк Thiazole- and oxazole-benzene sulfonamide compounds
FR2950345B1 (fr) * 2009-09-18 2011-09-23 Sanofi Aventis Derives acetyleniques de 5-phenyl-pyrazolopyridine, leur preparation et leur application en therapeutique
TWI600654B (zh) 2012-11-19 2017-10-01 艾姆公司 用於治療寄生蟲疾病之化合物及組合物
US8871754B2 (en) 2012-11-19 2014-10-28 Irm Llc Compounds and compositions for the treatment of parasitic diseases

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS4821117B1 (de) * 1970-09-25 1973-06-26
JPS5753486A (en) * 1980-09-17 1982-03-30 Mitsubishi Paper Mills Ltd Preparation of 3-formyl-pyrazolo 1,5-a pyridine derivative
JPS57126489A (en) * 1981-01-28 1982-08-06 Mitsubishi Paper Mills Ltd Preparation of pyrazolo(1, 5-a)pyridine derivative
JPS60248689A (ja) * 1984-05-24 1985-12-09 Mitsubishi Paper Mills Ltd ３−（３′−ピラゾロ〔１，５−ａ〕ピリジル）アクロレイン誘導体

Also Published As

Publication number Publication date
DE60103752D1 (de) 2004-07-15
EP1276742B1 (de) 2004-06-09
JP2003531906A (ja) 2003-10-28
DE60103752T2 (de) 2005-07-14
AU2001259242A1 (en) 2001-11-12
WO2001083479A3 (en) 2002-05-23
EP1276742A2 (de) 2003-01-22
ES2222372T3 (es) 2005-02-01
WO2001083479A2 (en) 2001-11-08

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Legal Events

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