ATE23860T1 - Imidazo(1,2-a)pyridine, ihre herstellung und therapeutische verwendung. - Google Patents

Imidazo(1,2-a)pyridine, ihre herstellung und therapeutische verwendung.

Info

Publication number
ATE23860T1
ATE23860T1 AT83400706T AT83400706T ATE23860T1 AT E23860 T1 ATE23860 T1 AT E23860T1 AT 83400706 T AT83400706 T AT 83400706T AT 83400706 T AT83400706 T AT 83400706T AT E23860 T1 ATE23860 T1 AT E23860T1
Authority
AT
Austria
Prior art keywords
radical
alkyl
hydrogen atom
optionally carrying
halogen atom
Prior art date
Application number
AT83400706T
Other languages
English (en)
Inventor
Jean-Pierre Kaplan
Pascal George
Jean-Michel Bernardon
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Application granted granted Critical
Publication of ATE23860T1 publication Critical patent/ATE23860T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Biomedical Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Neurosurgery (AREA)
  • Medicinal Chemistry (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
AT83400706T 1982-04-21 1983-04-07 Imidazo(1,2-a)pyridine, ihre herstellung und therapeutische verwendung. ATE23860T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8206841A FR2525602A1 (fr) 1982-04-21 1982-04-21 Imidazo(1,2-a)pyridines, leur preparation et leur application en therapeutique
EP83400706A EP0092459B1 (de) 1982-04-21 1983-04-07 Imidazo(1,2-a)Pyridine, ihre Herstellung und therapeutische Verwendung

Publications (1)

Publication Number Publication Date
ATE23860T1 true ATE23860T1 (de) 1986-12-15

Family

ID=9273216

Family Applications (1)

Application Number Title Priority Date Filing Date
AT83400706T ATE23860T1 (de) 1982-04-21 1983-04-07 Imidazo(1,2-a)pyridine, ihre herstellung und therapeutische verwendung.

Country Status (19)

Country Link
US (1) US4492695A (de)
EP (1) EP0092459B1 (de)
JP (1) JPS58189180A (de)
AT (1) ATE23860T1 (de)
AU (1) AU553112B2 (de)
CA (1) CA1254207A (de)
DE (1) DE3367918D1 (de)
DK (1) DK173783A (de)
ES (1) ES8402298A1 (de)
FI (1) FI73998C (de)
FR (1) FR2525602A1 (de)
GR (1) GR78577B (de)
HU (1) HU189648B (de)
IE (1) IE54923B1 (de)
IL (1) IL68443A0 (de)
NO (1) NO156048C (de)
NZ (1) NZ203955A (de)
PT (1) PT76574B (de)
ZA (1) ZA832787B (de)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3406329A1 (de) * 1984-02-22 1985-08-22 Merck Patent Gmbh, 6100 Darmstadt Pyridone
FR2606410B1 (fr) * 1986-11-07 1989-02-24 Synthelabo Imidazopyridines, leur preparation et leur application en therapeutique
US5364849A (en) * 1989-04-22 1994-11-15 John Wyeth & Brother, Limited 1-[3 or 4-[1-[4-piperazinyl]]-2 arylpropionyl or butryl]-heterocyclic derivatives
AU5409998A (en) * 1996-12-11 1998-07-03 Takeda Chemical Industries Ltd. Imidazopyridine derivatives and their production
AUPP278498A0 (en) 1998-04-03 1998-04-30 Australian Nuclear Science & Technology Organisation Peripheral benzodiazepine receptor binding agents
CA2387719C (en) 1999-07-30 2010-04-27 Zenyaku Kogyo Kabushiki Kaisha Azaindolizinone derivatives and cognitive enhancers comprising the same as effective components
IT1318624B1 (it) * 2000-07-14 2003-08-27 Dinamite Dipharma S P A In For Processo per la preparazione di 2-fenil-imidazo (1,2-a)piridin-3-acetammidi.
SE0003186D0 (sv) * 2000-09-07 2000-09-07 Astrazeneca Ab New process
US6596731B2 (en) 2001-03-27 2003-07-22 Hoffmann-La Roche Inc. Substituted imidazo[1,2-A] pyridine derivatives
WO2010074753A1 (en) 2008-12-23 2010-07-01 Map Pharmaceuticals, Inc. Inhalation devices and related methods for administration of sedative hypnotic compounds
WO2010117787A2 (en) * 2009-03-30 2010-10-14 The Brigham And Women's Hospital, Inc. Inhibiting eph b-3 kinase
CN106866667B (zh) 2009-11-05 2019-11-15 圣母大学 咪唑并[1,2-a]吡啶类化合物及其合成及使用方法
CN103360387B (zh) * 2012-03-28 2016-12-14 江苏豪森药业集团有限公司 一种制备化合物唑吡坦的方法
KR20180053386A (ko) 2015-09-17 2018-05-21 마빈 제이. 밀러 마이코박테리아 감염에 대해 유용한 벤질 아민-함유 헤테로사이클릭 화합물 및 조성물
EP3468545A4 (de) 2016-06-08 2020-07-22 President and Fellows of Harvard College Verfahren und zusammensetzungen zur verringerung von taktiler dysfunktion und angst im zusammenhang mit autismus-spektrum-störungen, rett-syndrom und fragilem x-syndrom
CN107163039A (zh) * 2017-05-11 2017-09-15 浙江工业大学 一种6‑甲基‑2‑对甲苯基咪唑并[1,2‑a]吡啶‑3‑甲醛的制备方法
CA3099791A1 (en) * 2018-05-29 2019-12-05 President And Fellows Of Harvard College Compositions and methods for reducing tactile dysfunction, anxiety, and social impairment
US12077512B2 (en) 2019-03-25 2024-09-03 President And Fellows Of Harvard College Compositions and methods for reducing tactile dysfunction, anxiety, and social impairment

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1076089A (en) * 1965-11-09 1967-07-19 Selvi & C Lab Bioterapico New derivatives of imidazo [1,2-a]-pyridine and a process for the manufacture thereof
FR2492382A1 (fr) * 1980-10-22 1982-04-23 Synthelabo Derives d'imidazo (1,2-a) pyridine, leur preparation et leur application en therapeutique

Also Published As

Publication number Publication date
IL68443A0 (en) 1983-07-31
FR2525602B1 (de) 1984-06-22
AU1370083A (en) 1983-10-27
DK173783A (da) 1983-10-22
HU189648B (en) 1986-07-28
FR2525602A1 (fr) 1983-10-28
CA1254207A (en) 1989-05-16
NO831390L (no) 1983-10-24
NZ203955A (en) 1985-11-08
JPS58189180A (ja) 1983-11-04
JPH0412270B2 (de) 1992-03-04
FI73998C (fi) 1987-12-10
EP0092459A3 (en) 1984-02-01
NO156048B (no) 1987-04-06
AU553112B2 (en) 1986-07-03
FI831349A0 (fi) 1983-04-20
FI73998B (fi) 1987-08-31
GR78577B (de) 1984-09-27
PT76574A (fr) 1983-05-01
PT76574B (fr) 1986-02-27
IE830896L (en) 1983-10-21
FI831349L (fi) 1983-10-22
NO156048C (no) 1987-07-15
US4492695A (en) 1985-01-08
ZA832787B (en) 1983-12-28
IE54923B1 (en) 1990-03-28
DE3367918D1 (en) 1987-01-15
ES521651A0 (es) 1984-01-16
ES8402298A1 (es) 1984-01-16
EP0092459A2 (de) 1983-10-26
EP0092459B1 (de) 1986-11-26
DK173783D0 (da) 1983-04-20

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ATE23860T1 (de) Imidazo(1,2-a)pyridine, ihre herstellung und therapeutische verwendung.
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Legal Events

Date Code Title Description
UEP Publication of translation of european patent specification
REN Ceased due to non-payment of the annual fee