ATE207929T1 - Diastereomerenreine 3-oxo und 3-thioxo-4-aza- androstanderivate und ihre verwendung als antiandrogene - Google Patents

Diastereomerenreine 3-oxo und 3-thioxo-4-aza- androstanderivate und ihre verwendung als antiandrogene

Info

Publication number
ATE207929T1
ATE207929T1 AT95942689T AT95942689T ATE207929T1 AT E207929 T1 ATE207929 T1 AT E207929T1 AT 95942689 T AT95942689 T AT 95942689T AT 95942689 T AT95942689 T AT 95942689T AT E207929 T1 ATE207929 T1 AT E207929T1
Authority
AT
Austria
Prior art keywords
androan
antiandrogens
thioxo
aza
oxo
Prior art date
Application number
AT95942689T
Other languages
English (en)
Inventor
Stefano Poli
Roberto Girardello
Paride Grisenti
Ambrogio Magni
Vincenzo Olgiati
Original Assignee
Polichem Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Polichem Sa filed Critical Polichem Sa
Application granted granted Critical
Publication of ATE207929T1 publication Critical patent/ATE207929T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • C07J73/001—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
    • C07J73/005—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by nitrogen as hetero atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
AT95942689T 1994-12-23 1995-12-18 Diastereomerenreine 3-oxo und 3-thioxo-4-aza- androstanderivate und ihre verwendung als antiandrogene ATE207929T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ITMI942626A IT1271325B (it) 1994-12-23 1994-12-23 Composti diastereomericamente puri derivati da 3-oxo e 3-tioxo-4-azaandrostani e loro uso come antiandrogeni
PCT/EP1995/005008 WO1996020210A2 (en) 1994-12-23 1995-12-18 Diastereomerically pure 3-oxo and 3-thioxo-4-aza-androstan derivatives and the use thereof as antiandrogens

Publications (1)

Publication Number Publication Date
ATE207929T1 true ATE207929T1 (de) 2001-11-15

Family

ID=11370067

Family Applications (1)

Application Number Title Priority Date Filing Date
AT95942689T ATE207929T1 (de) 1994-12-23 1995-12-18 Diastereomerenreine 3-oxo und 3-thioxo-4-aza- androstanderivate und ihre verwendung als antiandrogene

Country Status (10)

Country Link
US (1) US6147213A (de)
EP (1) EP0799239B1 (de)
AT (1) ATE207929T1 (de)
AU (1) AU4387296A (de)
DE (1) DE69523622T2 (de)
DK (1) DK0799239T3 (de)
ES (1) ES2163538T3 (de)
IT (1) IT1271325B (de)
PT (1) PT799239E (de)
WO (1) WO1996020210A2 (de)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6645974B2 (en) 2001-07-31 2003-11-11 Merck & Co., Inc. Androgen receptor modulators and methods for use thereof
BRPI0718811B1 (pt) 2006-11-15 2020-05-19 Basf Se dispositivo elétrico de capacitância de camada dupla
JP5456669B2 (ja) * 2007-05-03 2014-04-02 エール ユニヴァーシティ 局所活性「ソフト」抗アンドロゲン剤
US8404384B2 (en) 2009-07-01 2013-03-26 Energ2 Technologies, Inc. Ultrapure synthetic carbon materials
EP2510569B1 (de) * 2009-12-11 2020-07-22 Basf Se Kohlenstoffmaterialien mit einem elektrochemischen modifikator
WO2011112992A1 (en) 2010-03-12 2011-09-15 Energ2, Inc. Mesoporous carbon materials comprising bifunctional catalysts
CN103261090A (zh) 2010-09-30 2013-08-21 艾纳G2技术公司 储能颗粒的增强式装填
JP6324726B2 (ja) 2010-12-28 2018-05-16 ビーエーエスエフ ソシエタス・ヨーロピアＢａｓｆ Ｓｅ 電気化学特性が向上した炭素材料
US20120262127A1 (en) 2011-04-15 2012-10-18 Energ2 Technologies, Inc. Flow ultracapacitor
EP2715840B1 (de) 2011-06-03 2015-05-27 Basf Se Kohlenstoff-blei-mischungen zur verwendung in hybriden energiespeichereinrichtungen
US9409777B2 (en) 2012-02-09 2016-08-09 Basf Se Preparation of polymeric resins and carbon materials
WO2014143213A1 (en) 2013-03-14 2014-09-18 Energ2 Technologies, Inc. Composite carbon materials comprising lithium alloying electrochemical modifiers
US10195583B2 (en) 2013-11-05 2019-02-05 Group 14 Technologies, Inc. Carbon-based compositions with highly efficient volumetric gas sorption
EP4496080A3 (de) 2014-03-14 2025-05-07 Group14 Technologies, Inc. Neuartige verfahren zur sol-gel-polymerisation ohne lösungsmittel und erzeugung einer abstimmbaren kohlenstoffstruktur daraus
US10763501B2 (en) 2015-08-14 2020-09-01 Group14 Technologies, Inc. Nano-featured porous silicon materials
JP7115976B2 (ja) 2015-08-28 2022-08-09 グループ１４・テクノロジーズ・インコーポレイテッド リチウムの非常に耐久性のある挿入を有する新規な材料およびその製造方法
KR20250061765A (ko) 2017-03-09 2025-05-08 그룹14 테크놀로지스, 인코포레이티드 다공성 스캐폴드 재료 상의 실리콘 함유 전구체의 분해
US11335903B2 (en) 2020-08-18 2022-05-17 Group14 Technologies, Inc. Highly efficient manufacturing of silicon-carbon composites materials comprising ultra low z
US11639292B2 (en) 2020-08-18 2023-05-02 Group14 Technologies, Inc. Particulate composite materials
US11174167B1 (en) 2020-08-18 2021-11-16 Group14 Technologies, Inc. Silicon carbon composites comprising ultra low Z
CN116457309B (zh) 2020-09-30 2025-02-14 14集团技术公司 控制硅-碳复合材料的氧含量和反应性的钝化方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4845104A (en) * 1986-11-20 1989-07-04 Merck & Co., Inc. Oxidized analogs of 17β-N-monosubstituted-carbamoyl-4-aza-5-α-androstan-3-ones
IE76452B1 (en) * 1990-10-29 1997-10-22 Sankyo Co Azasteroid compounds for the treatment of prostatic hypertrophy their preparation and use
GB9216329D0 (en) * 1992-07-31 1992-09-16 Erba Carlo Spa 17beta-substituted 4-aza-5alpha-androstan-3-one derivatives

Also Published As

Publication number Publication date
EP0799239A2 (de) 1997-10-08
ITMI942626A0 (it) 1994-12-23
IT1271325B (it) 1997-05-27
WO1996020210A2 (en) 1996-07-04
DE69523622T2 (de) 2002-05-29
ITMI942626A1 (it) 1996-06-23
EP0799239B1 (de) 2001-10-31
US6147213A (en) 2000-11-14
PT799239E (pt) 2002-02-28
AU4387296A (en) 1996-07-19
DE69523622D1 (de) 2001-12-06
DK0799239T3 (da) 2001-12-10
ES2163538T3 (es) 2002-02-01
WO1996020210A3 (en) 1996-09-06

Similar Documents

Publication Publication Date Title
ATE207929T1 (de) Diastereomerenreine 3-oxo und 3-thioxo-4-aza- androstanderivate und ihre verwendung als antiandrogene
NO970092D0 (no) Dihydrobenzofuraner
TR199901653T2 (xx) Fitalazinonlar.
TR199901305T2 (xx) Calpain-�nleyicileri olarak ketonbenzamidler
ATE172968T1 (de) Substituierte azadioxacycloalkene und ihre verwendung als fungizide
DE69910831D1 (de) Epothilonderivate und ihre verwendung als antitumormittel
MY138525A (en) Substituted acid derivatives useful as antidiabetic and antiobesity agents and method
AR010062A1 (es) Nuevos benzamidaldehidos y su utilizacion
TR199800011T1 (xx) Benzo$g] kuinolin t�revleri
AR006390A1 (es) Derivados de lactama
TR200800474T2 (tr) Florfenikole aracı maddelerin hazırlanmasına ilişkin işlem.
BR9408246A (pt) Composto derivado de 3-azabicicloalcano N-substituído
DK0831837T3 (da) Anvendelse af squalamin i fremstilling af et medikament til inhibering af NHE
TR199901282T2 (xx) Heterosiklik olarak ikame edilmi� yeni benzamitler.
ES2184077T3 (es) Nuevas fenantridinas sustituidas en la posicion 6.
BG103310A (en) Benzonaphthyridins as bronchial therapeutical means
NO943100L (no) Forbindelser for anvendelse i kontrastmidler for radiografi
EP1042352A4 (de) Androgene steroidderivate und ein verfahren zur herstellung und verwendung derselben
DK0730581T3 (da) 3-acylaminobezazepiner
BR9509970A (pt) Composto
ATE178886T1 (de) 1-aryl-2-acylamino-ethan-verbindungen und ihre verwendung als neurokinin- insbesondere als neurokinin-1-antagonisten
TR200201128T2 (tr) PDE4 inhibitörleri olarak tetrahidrotiyopiranfitalazinon türevleri.
TR200302288T2 (tr) Terapi için yeni bileşikler ve metotlar.
DE59510713D1 (de) N-substituierte 3-azabicyclo(3.2.0)heptan-derivate als neuroleptika
TR200101979T2 (tr) Antidepresyon tedavisi için 5HT1 antagonistleri.

Legal Events

Date Code Title Description
UEP Publication of translation of european patent specification