IT1271325B - Composti diastereomericamente puri derivati da 3-oxo e 3-tioxo-4-azaandrostani e loro uso come antiandrogeni - Google Patents

Composti diastereomericamente puri derivati da 3-oxo e 3-tioxo-4-azaandrostani e loro uso come antiandrogeni

Info

Publication number
IT1271325B
IT1271325B ITMI942626A ITMI942626A IT1271325B IT 1271325 B IT1271325 B IT 1271325B IT MI942626 A ITMI942626 A IT MI942626A IT MI942626 A ITMI942626 A IT MI942626A IT 1271325 B IT1271325 B IT 1271325B
Authority
IT
Italy
Prior art keywords
azaandrostani
thioxo
androgen
oxo
compounds derived
Prior art date
Application number
ITMI942626A
Other languages
English (en)
Inventor
Stefano Poli
Roberto Girardello
Paride Grisenti
Ambrogio Magni
Vincenzo Olgiati
Original Assignee
Poli Ind Chimica Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Poli Ind Chimica Spa filed Critical Poli Ind Chimica Spa
Publication of ITMI942626A0 publication Critical patent/ITMI942626A0/it
Priority to ITMI942626A priority Critical patent/IT1271325B/it
Priority to DK95942689T priority patent/DK0799239T3/da
Priority to ES95942689T priority patent/ES2163538T3/es
Priority to PCT/EP1995/005008 priority patent/WO1996020210A2/en
Priority to AT95942689T priority patent/ATE207929T1/de
Priority to EP95942689A priority patent/EP0799239B1/en
Priority to AU43872/96A priority patent/AU4387296A/en
Priority to DE69523622T priority patent/DE69523622T2/de
Priority to US08/879,442 priority patent/US6147213A/en
Priority to PT95942689T priority patent/PT799239E/pt
Publication of ITMI942626A1 publication Critical patent/ITMI942626A1/it
Application granted granted Critical
Publication of IT1271325B publication Critical patent/IT1271325B/it

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • C07J73/001—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
    • C07J73/005—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by nitrogen as hetero atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
ITMI942626A 1994-12-23 1994-12-23 Composti diastereomericamente puri derivati da 3-oxo e 3-tioxo-4-azaandrostani e loro uso come antiandrogeni IT1271325B (it)

Priority Applications (10)

Application Number Priority Date Filing Date Title
ITMI942626A IT1271325B (it) 1994-12-23 1994-12-23 Composti diastereomericamente puri derivati da 3-oxo e 3-tioxo-4-azaandrostani e loro uso come antiandrogeni
AT95942689T ATE207929T1 (de) 1994-12-23 1995-12-18 Diastereomerenreine 3-oxo und 3-thioxo-4-aza- androstanderivate und ihre verwendung als antiandrogene
ES95942689T ES2163538T3 (es) 1994-12-23 1995-12-18 Derivados de 3-oxo y 3-tioxo-4-aza-androstano diastereomericamente puros y su uso como antiandrogenos.
PCT/EP1995/005008 WO1996020210A2 (en) 1994-12-23 1995-12-18 Diastereomerically pure 3-oxo and 3-thioxo-4-aza-androstan derivatives and the use thereof as antiandrogens
DK95942689T DK0799239T3 (da) 1994-12-23 1995-12-18 Diastereomert rene 3-oxo- og 3-thioxo-4-aza-androstan-derivater og anvendelse deraf som antiandrogener
EP95942689A EP0799239B1 (en) 1994-12-23 1995-12-18 Diastereomerically pure 3-oxo and 3-thioxo-4-aza-androstan derivatives and the use thereof as antiandrogens
AU43872/96A AU4387296A (en) 1994-12-23 1995-12-18 Diastereomerically pure 3-oxo and 3-thioxo-4-aza-androstan derivatives and the use thereof as antiandrogens
DE69523622T DE69523622T2 (de) 1994-12-23 1995-12-18 Diastereomerenreine 3-oxo und 3-thioxo-4-aza-androstanderivate und ihre verwendung als antiandrogene
US08/879,442 US6147213A (en) 1994-12-23 1995-12-18 Diastereomerically pure 3-oxo and 3-thioxo-4-aza-androstan derivatives and the use thereof as antiandrogens
PT95942689T PT799239E (pt) 1994-12-23 1995-12-18 Derivados diastereomericamente puros de 3-oxo e 3-tioxo-4-aza-androstano e a sua utilizacao como anti-androgenos

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ITMI942626A IT1271325B (it) 1994-12-23 1994-12-23 Composti diastereomericamente puri derivati da 3-oxo e 3-tioxo-4-azaandrostani e loro uso come antiandrogeni

Publications (3)

Publication Number Publication Date
ITMI942626A0 ITMI942626A0 (it) 1994-12-23
ITMI942626A1 ITMI942626A1 (it) 1996-06-23
IT1271325B true IT1271325B (it) 1997-05-27

Family

ID=11370067

Family Applications (1)

Application Number Title Priority Date Filing Date
ITMI942626A IT1271325B (it) 1994-12-23 1994-12-23 Composti diastereomericamente puri derivati da 3-oxo e 3-tioxo-4-azaandrostani e loro uso come antiandrogeni

Country Status (10)

Country Link
US (1) US6147213A (it)
EP (1) EP0799239B1 (it)
AT (1) ATE207929T1 (it)
AU (1) AU4387296A (it)
DE (1) DE69523622T2 (it)
DK (1) DK0799239T3 (it)
ES (1) ES2163538T3 (it)
IT (1) IT1271325B (it)
PT (1) PT799239E (it)
WO (1) WO1996020210A2 (it)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6645974B2 (en) 2001-07-31 2003-11-11 Merck & Co., Inc. Androgen receptor modulators and methods for use thereof
BRPI0718811B1 (pt) 2006-11-15 2020-05-19 Basf Se dispositivo elétrico de capacitância de camada dupla
WO2008137038A1 (en) * 2007-05-03 2008-11-13 Yale University Locally active 'soft' antiandrogens
KR102139269B1 (ko) 2009-07-01 2020-08-11 바스프 에스이 초고순도의 합성 탄소 물질
EP2510569B1 (en) * 2009-12-11 2020-07-22 Basf Se Carbon materials comprising an electrochemical modifier
US8916296B2 (en) 2010-03-12 2014-12-23 Energ2 Technologies, Inc. Mesoporous carbon materials comprising bifunctional catalysts
WO2012045002A1 (en) 2010-09-30 2012-04-05 Energ2 Technologies, Inc. Enhanced packing of energy storage particles
CN108538625B (zh) 2010-12-28 2020-12-08 巴斯福股份公司 包含增强的电化学特性的碳材料
US20120262127A1 (en) 2011-04-15 2012-10-18 Energ2 Technologies, Inc. Flow ultracapacitor
WO2012167117A2 (en) 2011-06-03 2012-12-06 Energ2 Technologies, Inc. Carbon-lead blends for use in hybrid energy storage devices
US9409777B2 (en) 2012-02-09 2016-08-09 Basf Se Preparation of polymeric resins and carbon materials
CN110112377A (zh) 2013-03-14 2019-08-09 14族科技公司 包含锂合金化的电化学改性剂的复合碳材料
US10195583B2 (en) 2013-11-05 2019-02-05 Group 14 Technologies, Inc. Carbon-based compositions with highly efficient volumetric gas sorption
EP4496080A3 (en) 2014-03-14 2025-05-07 Group14 Technologies, Inc. Novel methods for sol-gel polymerization in absence of solvent and creation of tunable carbon structure from same
US20190097222A1 (en) 2015-08-14 2019-03-28 Energ2 Technologies, Inc. Composites of porous nano-featured silicon materials and carbon materials
JP7115976B2 (ja) 2015-08-28 2022-08-09 グループ１４・テクノロジーズ・インコーポレイテッド リチウムの非常に耐久性のある挿入を有する新規な材料およびその製造方法
JP7376360B2 (ja) 2017-03-09 2023-11-08 グループ１４・テクノロジーズ・インコーポレイテッド 多孔質足場材料の上のケイ素含有前駆体の分解
US11335903B2 (en) 2020-08-18 2022-05-17 Group14 Technologies, Inc. Highly efficient manufacturing of silicon-carbon composites materials comprising ultra low z
US11639292B2 (en) 2020-08-18 2023-05-02 Group14 Technologies, Inc. Particulate composite materials
US11174167B1 (en) 2020-08-18 2021-11-16 Group14 Technologies, Inc. Silicon carbon composites comprising ultra low Z
JP2023544717A (ja) 2020-09-30 2023-10-25 グループ１４・テクノロジーズ・インコーポレイテッド シリコン－カーボン複合材料の酸素含有量及び反応性制御のための不動態化の方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4845104A (en) * 1986-11-20 1989-07-04 Merck & Co., Inc. Oxidized analogs of 17β-N-monosubstituted-carbamoyl-4-aza-5-α-androstan-3-ones
IE76452B1 (en) * 1990-10-29 1997-10-22 Sankyo Co Azasteroid compounds for the treatment of prostatic hypertrophy their preparation and use
GB9216329D0 (en) * 1992-07-31 1992-09-16 Erba Carlo Spa 17beta-substituted 4-aza-5alpha-androstan-3-one derivatives

Also Published As

Publication number Publication date
PT799239E (pt) 2002-02-28
WO1996020210A2 (en) 1996-07-04
EP0799239A2 (en) 1997-10-08
ATE207929T1 (de) 2001-11-15
ITMI942626A0 (it) 1994-12-23
DK0799239T3 (da) 2001-12-10
AU4387296A (en) 1996-07-19
DE69523622T2 (de) 2002-05-29
EP0799239B1 (en) 2001-10-31
WO1996020210A3 (en) 1996-09-06
DE69523622D1 (de) 2001-12-06
ITMI942626A1 (it) 1996-06-23
US6147213A (en) 2000-11-14
ES2163538T3 (es) 2002-02-01

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Legal Events

Date Code Title Description
0001 Granted
TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19971223