DK0799239T3 - Diastereomert rene 3-oxo- og 3-thioxo-4-aza-androstan-derivater og anvendelse deraf som antiandrogener - Google Patents

Diastereomert rene 3-oxo- og 3-thioxo-4-aza-androstan-derivater og anvendelse deraf som antiandrogener

Info

Publication number
DK0799239T3
DK0799239T3 DK95942689T DK95942689T DK0799239T3 DK 0799239 T3 DK0799239 T3 DK 0799239T3 DK 95942689 T DK95942689 T DK 95942689T DK 95942689 T DK95942689 T DK 95942689T DK 0799239 T3 DK0799239 T3 DK 0799239T3
Authority
DK
Denmark
Prior art keywords
antiandrogens
thioxo
aza
oxo
diastereomerically pure
Prior art date
Application number
DK95942689T
Other languages
English (en)
Inventor
Stefano Poli
Roberto Girardello
Paride Grisenti
Vincenzo Olgiati
Ambrogio Magni
Original Assignee
Polichem Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Polichem Sa filed Critical Polichem Sa
Application granted granted Critical
Publication of DK0799239T3 publication Critical patent/DK0799239T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • C07J73/001—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
    • C07J73/005—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by nitrogen as hetero atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK95942689T 1994-12-23 1995-12-18 Diastereomert rene 3-oxo- og 3-thioxo-4-aza-androstan-derivater og anvendelse deraf som antiandrogener DK0799239T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ITMI942626A IT1271325B (it) 1994-12-23 1994-12-23 Composti diastereomericamente puri derivati da 3-oxo e 3-tioxo-4-azaandrostani e loro uso come antiandrogeni
PCT/EP1995/005008 WO1996020210A2 (en) 1994-12-23 1995-12-18 Diastereomerically pure 3-oxo and 3-thioxo-4-aza-androstan derivatives and the use thereof as antiandrogens

Publications (1)

Publication Number Publication Date
DK0799239T3 true DK0799239T3 (da) 2001-12-10

Family

ID=11370067

Family Applications (1)

Application Number Title Priority Date Filing Date
DK95942689T DK0799239T3 (da) 1994-12-23 1995-12-18 Diastereomert rene 3-oxo- og 3-thioxo-4-aza-androstan-derivater og anvendelse deraf som antiandrogener

Country Status (10)

Country Link
US (1) US6147213A (da)
EP (1) EP0799239B1 (da)
AT (1) ATE207929T1 (da)
AU (1) AU4387296A (da)
DE (1) DE69523622T2 (da)
DK (1) DK0799239T3 (da)
ES (1) ES2163538T3 (da)
IT (1) IT1271325B (da)
PT (1) PT799239E (da)
WO (1) WO1996020210A2 (da)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6645974B2 (en) 2001-07-31 2003-11-11 Merck & Co., Inc. Androgen receptor modulators and methods for use thereof
BRPI0718811B1 (pt) 2006-11-15 2020-05-19 Basf Se dispositivo elétrico de capacitância de camada dupla
US8552061B2 (en) * 2007-05-03 2013-10-08 Yale University Locally active “soft” antiandrogens
HRP20241382T1 (hr) 2009-07-01 2024-12-20 Basf Mobile Emissions Catalysts Llc Ultračisti sintetički ugljični materijali
BR112012014092A2 (pt) * 2009-12-11 2016-07-05 Energ2 Technologies Inc materiais de carvão compreendendo um modificador eletroquímico.
US8916296B2 (en) 2010-03-12 2014-12-23 Energ2 Technologies, Inc. Mesoporous carbon materials comprising bifunctional catalysts
US8654507B2 (en) 2010-09-30 2014-02-18 Energ2 Technologies, Inc. Enhanced packing of energy storage particles
CN108538625B (zh) 2010-12-28 2020-12-08 巴斯福股份公司 包含增强的电化学特性的碳材料
US20120262127A1 (en) 2011-04-15 2012-10-18 Energ2 Technologies, Inc. Flow ultracapacitor
CN103947017B (zh) 2011-06-03 2017-11-17 巴斯福股份公司 用于混合能量存储装置中的碳‑铅共混物
US9409777B2 (en) 2012-02-09 2016-08-09 Basf Se Preparation of polymeric resins and carbon materials
WO2014143213A1 (en) 2013-03-14 2014-09-18 Energ2 Technologies, Inc. Composite carbon materials comprising lithium alloying electrochemical modifiers
US10195583B2 (en) 2013-11-05 2019-02-05 Group 14 Technologies, Inc. Carbon-based compositions with highly efficient volumetric gas sorption
KR102663138B1 (ko) 2014-03-14 2024-05-03 그룹14 테크놀로지스, 인코포레이티드 용매의 부재하의 졸-겔 중합을 위한 신규한 방법 및 그러한 방법으로부터의 가변형 탄소 구조의 생성
US20190097222A1 (en) 2015-08-14 2019-03-28 Energ2 Technologies, Inc. Composites of porous nano-featured silicon materials and carbon materials
US10147950B2 (en) 2015-08-28 2018-12-04 Group 14 Technologies, Inc. Materials with extremely durable intercalation of lithium and manufacturing methods thereof
KR102798089B1 (ko) 2017-03-09 2025-04-21 그룹14 테크놀로지스, 인코포레이티드 다공성 스캐폴드 재료 상의 실리콘 함유 전구체의 분해
KR20230052901A (ko) 2020-08-10 2023-04-20 그룹14 테크놀로지스, 인코포레이티드 열진동 보조 화학 기상 침투
US11639292B2 (en) 2020-08-18 2023-05-02 Group14 Technologies, Inc. Particulate composite materials
US11335903B2 (en) 2020-08-18 2022-05-17 Group14 Technologies, Inc. Highly efficient manufacturing of silicon-carbon composites materials comprising ultra low z
US11174167B1 (en) 2020-08-18 2021-11-16 Group14 Technologies, Inc. Silicon carbon composites comprising ultra low Z
CN116457309B (zh) 2020-09-30 2025-02-14 14集团技术公司 控制硅-碳复合材料的氧含量和反应性的钝化方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4845104A (en) * 1986-11-20 1989-07-04 Merck & Co., Inc. Oxidized analogs of 17β-N-monosubstituted-carbamoyl-4-aza-5-α-androstan-3-ones
IE76452B1 (en) * 1990-10-29 1997-10-22 Sankyo Co Azasteroid compounds for the treatment of prostatic hypertrophy their preparation and use
GB9216329D0 (en) * 1992-07-31 1992-09-16 Erba Carlo Spa 17beta-substituted 4-aza-5alpha-androstan-3-one derivatives

Also Published As

Publication number Publication date
DE69523622D1 (de) 2001-12-06
ATE207929T1 (de) 2001-11-15
PT799239E (pt) 2002-02-28
US6147213A (en) 2000-11-14
EP0799239B1 (en) 2001-10-31
ITMI942626A1 (it) 1996-06-23
AU4387296A (en) 1996-07-19
WO1996020210A2 (en) 1996-07-04
WO1996020210A3 (en) 1996-09-06
ITMI942626A0 (it) 1994-12-23
ES2163538T3 (es) 2002-02-01
DE69523622T2 (de) 2002-05-29
EP0799239A2 (en) 1997-10-08
IT1271325B (it) 1997-05-27

Similar Documents

Publication Publication Date Title
DK0799239T3 (da) Diastereomert rene 3-oxo- og 3-thioxo-4-aza-androstan-derivater og anvendelse deraf som antiandrogener
NO962286D0 (no) N-substituerte azabicykloalkanderivater som neuroleptika etc.
ES2124424T3 (es) Azadioxacicloalquenos substituidos y su empleo como fungicidas.
AR003955A1 (es) Derivados de n-(indol-2-carbonil)-glicinamidas, procedimiento para su obtencion y composiciones que los contienen.
ES2083595T3 (es) Derivados de indol que inhiben la biosintesis de leucotrienos.
ES2132415T3 (es) Nuevos derivados de 5-pirrolil-2-piridilmetilsulfinilbencimidazol.
NO943100L (no) Forbindelser for anvendelse i kontrastmidler for radiografi
NO20002676L (no) Androgene steroidforbindelser og en fremgangsmÕte for fremstilling og anvendelse av samme
NO970473L (no) N-substituerte 3-azabicyklo (3.2.0)heptanderivater egnet som neuroleptika
WO1995018821A3 (en) Novel antiandrogenic agents and related pharmaceutical compositions and methods of use
NO981393L (no) Guanidinoproteasehemmere
NO962285D0 (no) N-substituerte azabicykloheptan-derivater anvendt for eksempel som neuroleptika
NO990914L (no) Amorfe benzotiofener, fremgangsmÕter for fremstilling og fremgangsmÕter for anvendelse
FI970449A0 (fi) N-substituoituja atsabisykloheptaanijohdannaisia, jotka ovat käyttökelpoisia neuroleptisinä aineina
DK0970042T3 (da) 5-hydroxymethyl-2-aminotetraliner som kardiovaskulære midler
ZA849159B (en) N-(methoxyphenacyl)-amine derivatives
FI962301A0 (fi) Substituoidut aminoalkyyliaminopyridiinit
ATE277614T1 (de) Anxiolytischer wirkstoff
DK0883628T3 (da) 17beta- (2-oxo-tetrahydrofuran-4-yl) -thioandrostanderivater (17beta- (gamma-smørsyrelacton) -thioderivater) til behandling
NO20053117L (no) Cyklopenta[c]isoksazol-3-aminer anvendt som materialbeskyttelsesmidler..
AR000385A1 (es) Proceso para la producción de derivados de 4-alcoxiimino-6-(5-hidroxipi razol-4-il)-tiocromano-1,1-dioxido y compuestos intermediarios de aplicación en dicho proceso y preparación de dichos compuestos intermediarios
ES2107281T3 (es) Nuevos derivados de acetaldehido, su procedimiento de preparacion y su aplicacion.
UA70975C2 (uk) Похідні 1,4-діарил-2-фтор-1-бутен-3-олу, спосіб їх одержання та способи одержання похідних 1,4-діарил-2-фтор-1,3-бутадієну і 1,4-діарил-2-фтор-2-бутену
ATE293605T1 (de) Fluorierte 3,4-dihydrochinolin-derivative als nos-inhibitoren
YU49004B (sh) LANOSTA-7,9-DIEN-3Гџ, 32-DIOL I POSTUPAK ZA NJEGOVO DOBIJANJE