DK0799239T3 - Diastereomert rene 3-oxo- og 3-thioxo-4-aza-androstan-derivater og anvendelse deraf som antiandrogener - Google Patents

Diastereomert rene 3-oxo- og 3-thioxo-4-aza-androstan-derivater og anvendelse deraf som antiandrogener

Info

Publication number
DK0799239T3
DK0799239T3 DK95942689T DK95942689T DK0799239T3 DK 0799239 T3 DK0799239 T3 DK 0799239T3 DK 95942689 T DK95942689 T DK 95942689T DK 95942689 T DK95942689 T DK 95942689T DK 0799239 T3 DK0799239 T3 DK 0799239T3
Authority
DK
Denmark
Prior art keywords
antiandrogens
thioxo
aza
oxo
diastereomerically pure
Prior art date
Application number
DK95942689T
Other languages
Danish (da)
English (en)
Inventor
Stefano Poli
Roberto Girardello
Paride Grisenti
Vincenzo Olgiati
Ambrogio Magni
Original Assignee
Polichem Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Polichem Sa filed Critical Polichem Sa
Application granted granted Critical
Publication of DK0799239T3 publication Critical patent/DK0799239T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • C07J73/001—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
    • C07J73/005—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by nitrogen as hetero atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK95942689T 1994-12-23 1995-12-18 Diastereomert rene 3-oxo- og 3-thioxo-4-aza-androstan-derivater og anvendelse deraf som antiandrogener DK0799239T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ITMI942626A IT1271325B (it) 1994-12-23 1994-12-23 Composti diastereomericamente puri derivati da 3-oxo e 3-tioxo-4-azaandrostani e loro uso come antiandrogeni
PCT/EP1995/005008 WO1996020210A2 (en) 1994-12-23 1995-12-18 Diastereomerically pure 3-oxo and 3-thioxo-4-aza-androstan derivatives and the use thereof as antiandrogens

Publications (1)

Publication Number Publication Date
DK0799239T3 true DK0799239T3 (da) 2001-12-10

Family

ID=11370067

Family Applications (1)

Application Number Title Priority Date Filing Date
DK95942689T DK0799239T3 (da) 1994-12-23 1995-12-18 Diastereomert rene 3-oxo- og 3-thioxo-4-aza-androstan-derivater og anvendelse deraf som antiandrogener

Country Status (10)

Country Link
US (1) US6147213A (de)
EP (1) EP0799239B1 (de)
AT (1) ATE207929T1 (de)
AU (1) AU4387296A (de)
DE (1) DE69523622T2 (de)
DK (1) DK0799239T3 (de)
ES (1) ES2163538T3 (de)
IT (1) IT1271325B (de)
PT (1) PT799239E (de)
WO (1) WO1996020210A2 (de)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6645974B2 (en) 2001-07-31 2003-11-11 Merck & Co., Inc. Androgen receptor modulators and methods for use thereof
JP2010510674A (ja) 2006-11-15 2010-04-02 エナジーツー・インコーポレイテッド 電気２重層キャパシタ装置
JP5456669B2 (ja) * 2007-05-03 2014-04-02 エール ユニヴァーシティ 局所活性「ソフト」抗アンドロゲン剤
EP2448748A4 (de) 2009-07-01 2016-04-06 Basf Se Ultrareine synthetische kohlenstoffmaterialien
WO2011072256A1 (en) * 2009-12-11 2011-06-16 Energ2, Inc. Carbon materials comprising an electrochemical modifier
US8916296B2 (en) 2010-03-12 2014-12-23 Energ2 Technologies, Inc. Mesoporous carbon materials comprising bifunctional catalysts
CN103261090A (zh) 2010-09-30 2013-08-21 艾纳G2技术公司 储能颗粒的增强式装填
US9269502B2 (en) 2010-12-28 2016-02-23 Basf Se Carbon materials comprising enhanced electrochemical properties
US20120262127A1 (en) 2011-04-15 2012-10-18 Energ2 Technologies, Inc. Flow ultracapacitor
WO2012167117A2 (en) 2011-06-03 2012-12-06 Energ2 Technologies, Inc. Carbon-lead blends for use in hybrid energy storage devices
WO2013120011A1 (en) 2012-02-09 2013-08-15 Energ2 Technologies, Inc. Preparation of polymeric resins and carbon materials
WO2014143213A1 (en) 2013-03-14 2014-09-18 Energ2 Technologies, Inc. Composite carbon materials comprising lithium alloying electrochemical modifiers
US10195583B2 (en) 2013-11-05 2019-02-05 Group 14 Technologies, Inc. Carbon-based compositions with highly efficient volumetric gas sorption
JP6665121B2 (ja) 2014-03-14 2020-03-13 グループ１４・テクノロジーズ・インコーポレイテッドＧｒｏｕｐ１４ Ｔｅｃｈｎｏｌｏｇｉｅｓ， Ｉｎｃ． 無溶媒中におけるゾル−ゲル重合のための新規方法、及びゾル−ゲル重合由来の可変炭素構造の作製
US20190097222A1 (en) 2015-08-14 2019-03-28 Energ2 Technologies, Inc. Composites of porous nano-featured silicon materials and carbon materials
KR102637617B1 (ko) 2015-08-28 2024-02-19 그룹14 테크놀로지스, 인코포레이티드 극도로 내구성이 우수한 리튬 인터칼레이션을 나타내는 신규 물질 및 그의 제조 방법
KR20230128140A (ko) 2017-03-09 2023-09-01 그룹14 테크놀로지스, 인코포레이티드 다공성 스캐폴드 재료 상의 실리콘 함유 전구체의 분해
US11639292B2 (en) 2020-08-18 2023-05-02 Group14 Technologies, Inc. Particulate composite materials
US11174167B1 (en) 2020-08-18 2021-11-16 Group14 Technologies, Inc. Silicon carbon composites comprising ultra low Z
US11335903B2 (en) 2020-08-18 2022-05-17 Group14 Technologies, Inc. Highly efficient manufacturing of silicon-carbon composites materials comprising ultra low z

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4845104A (en) * 1986-11-20 1989-07-04 Merck & Co., Inc. Oxidized analogs of 17β-N-monosubstituted-carbamoyl-4-aza-5-α-androstan-3-ones
IE76452B1 (en) * 1990-10-29 1997-10-22 Sankyo Co Azasteroid compounds for the treatment of prostatic hypertrophy their preparation and use
GB9216329D0 (en) * 1992-07-31 1992-09-16 Erba Carlo Spa 17beta-substituted 4-aza-5alpha-androstan-3-one derivatives

Also Published As

Publication number Publication date
DE69523622D1 (de) 2001-12-06
ITMI942626A0 (it) 1994-12-23
WO1996020210A3 (en) 1996-09-06
EP0799239A2 (de) 1997-10-08
PT799239E (pt) 2002-02-28
IT1271325B (it) 1997-05-27
ITMI942626A1 (it) 1996-06-23
ATE207929T1 (de) 2001-11-15
AU4387296A (en) 1996-07-19
ES2163538T3 (es) 2002-02-01
EP0799239B1 (de) 2001-10-31
DE69523622T2 (de) 2002-05-29
WO1996020210A2 (en) 1996-07-04
US6147213A (en) 2000-11-14

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