ATE200223T1 - Sampangin-derivate zur verwendung als antimykotische und antimykobakterielle wirkstoffe - Google Patents
Sampangin-derivate zur verwendung als antimykotische und antimykobakterielle wirkstoffeInfo
- Publication number
- ATE200223T1 ATE200223T1 AT92905142T AT92905142T ATE200223T1 AT E200223 T1 ATE200223 T1 AT E200223T1 AT 92905142 T AT92905142 T AT 92905142T AT 92905142 T AT92905142 T AT 92905142T AT E200223 T1 ATE200223 T1 AT E200223T1
- Authority
- AT
- Austria
- Prior art keywords
- sampangin
- antimycobacterial
- actives
- antifungal
- derivatives
- Prior art date
Links
- BWQKHOMAOVUASZ-UHFFFAOYSA-N sampangine Chemical class C1=NC(C(=O)C=2C3=CC=CC=2)=C2C3=NC=CC2=C1 BWQKHOMAOVUASZ-UHFFFAOYSA-N 0.000 title abstract 3
- 230000000843 anti-fungal effect Effects 0.000 title 1
- 230000001355 anti-mycobacterial effect Effects 0.000 title 1
- 229940121375 antifungal agent Drugs 0.000 title 1
- 239000003926 antimycobacterial agent Substances 0.000 title 1
- GVRYUHXXENMGEV-UHFFFAOYSA-N 4-methylbenzo[g]quinoline-5,10-dione Chemical compound O=C1C2=CC=CC=C2C(=O)C2=C1N=CC=C2C GVRYUHXXENMGEV-UHFFFAOYSA-N 0.000 abstract 2
- 206010017533 Fungal infection Diseases 0.000 abstract 1
- 206010062207 Mycobacterial infection Diseases 0.000 abstract 1
- 208000031888 Mycoses Diseases 0.000 abstract 1
- 230000002538 fungal effect Effects 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 208000027531 mycobacterial infectious disease Diseases 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/06—Peri-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
- C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
- C07D221/04—Ortho- or peri-condensed ring systems
- C07D221/06—Ring systems of three rings
- C07D221/08—Aza-anthracenes
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Medicines Containing Plant Substances (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US07/715,776 US5227383A (en) | 1991-06-14 | 1991-06-14 | Compounds and compositions useful as antifungal and antimycobacterial agents |
| PCT/US1991/008319 WO1992022297A1 (en) | 1991-06-14 | 1991-11-06 | New compounds and compositions useful as antifungal and antimycobacterial agents |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE200223T1 true ATE200223T1 (de) | 2001-04-15 |
Family
ID=24875436
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT92905142T ATE200223T1 (de) | 1991-06-14 | 1991-11-06 | Sampangin-derivate zur verwendung als antimykotische und antimykobakterielle wirkstoffe |
Country Status (10)
| Country | Link |
|---|---|
| US (2) | US5227383A (de) |
| EP (1) | EP0588796B1 (de) |
| JP (1) | JP3405540B2 (de) |
| AT (1) | ATE200223T1 (de) |
| CA (1) | CA2111338A1 (de) |
| DE (1) | DE69132575T2 (de) |
| DK (1) | DK0588796T3 (de) |
| ES (1) | ES2157899T3 (de) |
| GR (1) | GR3036159T3 (de) |
| WO (1) | WO1992022297A1 (de) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE4301424A1 (de) * | 1993-01-20 | 1994-07-21 | Basf Ag | Derivate des Azaanthrachinons und des Azaxanthons und diese enthaltende Herbizide und Pflanzenwachstumsregulatoren |
| US5476933A (en) * | 1994-11-16 | 1995-12-19 | State Of Oregon, Acting By And Through The Oregon State Board Of Higher Education, Acting For And On Behalf Of The Oregon Health Sciences University And The University Of Oregon | Azepine synthesis via a diels-alder reaction |
| US20040052868A1 (en) * | 2002-09-12 | 2004-03-18 | William Asiedu | Composition treating for AIDS and associated conditions |
| AU2011219481B2 (en) * | 2002-09-12 | 2012-09-20 | Willfred-Ramix, Inc. | A composition for treating AIDS and associated conditions |
| JP4794136B2 (ja) * | 2004-04-21 | 2011-10-19 | 阿蘇製薬株式会社 | アクリジン誘導体 |
| US7491721B2 (en) * | 2004-05-12 | 2009-02-17 | Lupin Limited | Antimycobacterial pharmaceutical composition |
| US20170112824A1 (en) * | 2015-10-23 | 2017-04-27 | Wright State University | Combination therapies for the treatment of fungal infections |
| CN106905317B (zh) * | 2017-01-24 | 2019-03-22 | 广西师范大学 | 4-取代Sampangine生物碱衍生物及其合成方法和应用 |
| AU2019289096B2 (en) | 2018-06-18 | 2022-05-26 | Elc Management Llc | Photostabilizing compounds, compositions, and methods |
| CA3104434C (en) | 2018-06-18 | 2023-09-05 | Elc Management Llc | Photostabilizing cyano-containing fused tricyclic compounds, compositions, and methods |
| US11484485B2 (en) | 2018-06-18 | 2022-11-01 | Elc Management Llc | Photostabilizing compounds, compositions, and methods |
| EP3807247A4 (de) | 2018-06-18 | 2021-10-13 | ELC Management LLC | Fotostabilierungsverbindungen, zusammensetzungen und verfahren |
| CN113461506A (zh) * | 2021-06-23 | 2021-10-01 | 苏州求索生物科技有限公司 | 一种2-溴-1,4-萘并醌的制备工艺 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4080456A (en) * | 1971-10-26 | 1978-03-21 | Schering Aktiengesellschaft | Diacylapomorphines |
| AR204011A1 (es) * | 1973-07-27 | 1975-11-12 | Rhone Poulenc Sa | Procedimiento de preparacion de nuevos derivados de 7-h-indolizino(5,6,7-ij)isoquinoleina |
| JPS5337696A (en) * | 1976-08-26 | 1978-04-06 | Omnium Chimique Sa | Hexahydrocantinonee6 derivative |
| US4965272A (en) * | 1988-07-14 | 1990-10-23 | Hufford Charles D | Antimicrobial compound and compositions particularly effective against candida albicans |
| US5128344A (en) * | 1990-11-06 | 1992-07-07 | University Of Mississippi | Sampangine and derivatives useful as an antifungal agent |
-
1991
- 1991-06-14 US US07/715,776 patent/US5227383A/en not_active Expired - Fee Related
- 1991-11-06 ES ES92905142T patent/ES2157899T3/es not_active Expired - Lifetime
- 1991-11-06 EP EP92905142A patent/EP0588796B1/de not_active Expired - Lifetime
- 1991-11-06 WO PCT/US1991/008319 patent/WO1992022297A1/en not_active Ceased
- 1991-11-06 JP JP50518192A patent/JP3405540B2/ja not_active Expired - Fee Related
- 1991-11-06 AT AT92905142T patent/ATE200223T1/de not_active IP Right Cessation
- 1991-11-06 DK DK92905142T patent/DK0588796T3/da active
- 1991-11-06 DE DE69132575T patent/DE69132575T2/de not_active Expired - Fee Related
- 1991-11-06 CA CA002111338A patent/CA2111338A1/en not_active Abandoned
-
1993
- 1993-07-12 US US08/090,594 patent/US5530004A/en not_active Expired - Lifetime
-
2001
- 2001-06-29 GR GR20010401010T patent/GR3036159T3/el not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| DE69132575D1 (de) | 2001-05-10 |
| CA2111338A1 (en) | 1992-12-23 |
| US5530004A (en) | 1996-06-25 |
| EP0588796A4 (en) | 1994-09-14 |
| DK0588796T3 (da) | 2001-05-07 |
| GR3036159T3 (en) | 2001-09-28 |
| EP0588796B1 (de) | 2001-04-04 |
| JPH06508104A (ja) | 1994-09-14 |
| EP0588796A1 (de) | 1994-03-30 |
| ES2157899T3 (es) | 2001-09-01 |
| US5227383A (en) | 1993-07-13 |
| JP3405540B2 (ja) | 2003-05-12 |
| DE69132575T2 (de) | 2001-10-18 |
| WO1992022297A1 (en) | 1992-12-23 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification | ||
| REN | Ceased due to non-payment of the annual fee |