ATE197249T1 - Stabiles arzneimittel enthaltend oxaliplatin - Google Patents

Stabiles arzneimittel enthaltend oxaliplatin

Info

Publication number
ATE197249T1
ATE197249T1 AT95925976T AT95925976T ATE197249T1 AT E197249 T1 ATE197249 T1 AT E197249T1 AT 95925976 T AT95925976 T AT 95925976T AT 95925976 T AT95925976 T AT 95925976T AT E197249 T1 ATE197249 T1 AT E197249T1
Authority
AT
Austria
Prior art keywords
pct
product containing
oxaliplatinum
medicinal product
containing oxaliplatin
Prior art date
Application number
AT95925976T
Other languages
English (en)
Inventor
Houssam Ibrahim
Rolland-Yves Mauvernay
Original Assignee
Debiopharm Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=50845249&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE197249(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Debiopharm Sa filed Critical Debiopharm Sa
Application granted granted Critical
Publication of ATE197249T1 publication Critical patent/ATE197249T1/de

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/28Compounds containing heavy metals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/28Compounds containing heavy metals
    • A61K31/282Platinum compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K33/00Medicinal preparations containing inorganic active ingredients
    • A61K33/24Heavy metals; Compounds thereof
    • A61K33/243Platinum; Compounds thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Inorganic Chemistry (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
AT95925976T 1994-08-08 1995-08-07 Stabiles arzneimittel enthaltend oxaliplatin ATE197249T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH246294 1994-08-08
PCT/IB1995/000614 WO1996004904A1 (fr) 1994-08-08 1995-08-07 Preparation pharmaceutiquement stable d'oxaliplatine

Publications (1)

Publication Number Publication Date
ATE197249T1 true ATE197249T1 (de) 2000-11-15

Family

ID=50845249

Family Applications (1)

Application Number Title Priority Date Filing Date
AT95925976T ATE197249T1 (de) 1994-08-08 1995-08-07 Stabiles arzneimittel enthaltend oxaliplatin

Country Status (17)

Country Link
US (1) US5716988A (de)
EP (1) EP0774963B1 (de)
JP (1) JP3547755B2 (de)
KR (1) KR100365171B1 (de)
CN (1) CN1138541C (de)
AT (1) ATE197249T1 (de)
AU (2) AU2989695A (de)
BR (1) BR9508554A (de)
CA (1) CA2196922C (de)
CZ (1) CZ286714B6 (de)
DE (1) DE69519300T2 (de)
DK (1) DK0774963T3 (de)
ES (1) ES2152412T3 (de)
IL (1) IL114852A (de)
RU (1) RU2148400C1 (de)
UA (1) UA42779C2 (de)
WO (1) WO1996004904A1 (de)

Families Citing this family (48)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69519300T2 (de) 1994-08-08 2001-05-31 Debiopharm Sa Stabiles arzneimittel enthaltend oxaliplatin
GB9804013D0 (en) * 1998-02-25 1998-04-22 Sanofi Sa Formulations
WO2000021527A2 (fr) * 1998-10-14 2000-04-20 Debiopharm S.A. Conditionnement d'une preparation d'oxaliplatine
GB9904386D0 (en) * 1999-02-25 1999-04-21 Pharmacia & Upjohn Spa Antitumour synergistic composition
BRPI0013613B8 (pt) * 1999-08-30 2021-05-25 Debiopharm Sa composição farmacêuticamente estável de oxaliplatina para administração parenteral.
US7070796B1 (en) * 1999-08-30 2006-07-04 Debiopharm S.A. Pharmaceutically stable oxaliplatinum preparation for parenteral administration
US7012072B2 (en) * 2000-12-12 2006-03-14 Debiopharm S.A. Pharmaceutical oxaliplatinum preparation for parenteral administration and method for obtaining same
SI1368022T1 (sl) * 2001-03-02 2007-10-31 Debiopharm Sa Uporaba stekleničke, ki vsebuje raztopino oksaliplatina
EP1404689A1 (de) * 2001-07-02 2004-04-07 Debiopharm S.A. Aktive oxiplatinverbindung mit sehr niedrigem oxalsaüregehalt
TWI315982B (en) 2001-07-19 2009-10-21 Novartis Ag Combinations comprising epothilones and pharmaceutical uses thereof
US6476068B1 (en) 2001-12-06 2002-11-05 Pharmacia Italia, S.P.A. Platinum derivative pharmaceutical formulations
CA2388352A1 (en) * 2002-05-31 2003-11-30 Voiceage Corporation A method and device for frequency-selective pitch enhancement of synthesized speed
US20040022842A1 (en) * 2002-06-03 2004-02-05 Mebiopharm Co., Ltd. Liposome preparations containing oxaliplatin
JP2007504098A (ja) 2003-08-28 2007-03-01 メイン・ファーマ・リミテッド 酸を含むオキサリプラチン製剤
EP2330110A1 (de) 2003-11-25 2011-06-08 Platco Technologies (Proprietary) Limited Platin(II) Komplexe, Herstellung und Verwendung
CN100471493C (zh) * 2003-12-17 2009-03-25 梅比欧法姆股份有限公司 含有奥沙利铂的脂质体制剂
JP5578753B2 (ja) * 2004-06-09 2014-08-27 大鵬薬品工業株式会社 抗腫瘍効果増強剤、抗腫瘍剤及び癌治療方法
ES2327346T3 (es) 2004-09-01 2009-10-28 Platco Technologies (Proprietary) Limited Preparacion de complejos de platino (ii).
US20060063720A1 (en) * 2004-09-22 2006-03-23 Edgar Schridde Oxaliplatin solution concentrate
US20060063833A1 (en) * 2004-09-22 2006-03-23 Edgar Schridde Ready-to-use oxaliplatin solutions
DE102004052877B4 (de) * 2004-11-02 2008-06-19 Ebewe Pharma Ges.M.B.H. Nfg.Kg Stabile wässrige Formulierungen eines Platin-Derivats
JP2006248978A (ja) * 2005-03-10 2006-09-21 Mebiopharm Co Ltd 新規なリポソーム製剤
WO2007029268A2 (en) 2005-09-05 2007-03-15 Dabur Pharma Limited Stable oxaliplatin formulation
US7956208B2 (en) * 2006-01-30 2011-06-07 Platco Technologies (Proprietary) Limited Preparation of platinum (II) complexes
CA2647297A1 (en) * 2006-03-16 2007-09-27 Bionumerik Pharmaceuticals, Inc. Anti-cancer activity augmentation compounds and formulations and methods of use thereof
JP2009536180A (ja) 2006-05-09 2009-10-08 ノバルティス アクチエンゲゼルシャフト 鉄キレート剤と抗新生物剤を含む組合せ剤およびそれらの使用
PT2101805E (pt) * 2007-01-18 2013-01-31 Merck Patent Gmbh Terapia específica e medicamento usando ligandos integrina para tratar o cancro
US20090076139A1 (en) * 2007-09-19 2009-03-19 Protia, Llc Deuterium-enriched oxalplatin
US20100267824A1 (en) * 2007-11-12 2010-10-21 Intas Pharmaceuticals Limited Stable oxaliplatin composition for parenteral administration
JP5694782B2 (ja) 2008-03-14 2015-04-01 バイオニューメリック・ファーマスーティカルズ・インコーポレイテッド 肺癌、腺癌及び他の病状のための治療方法及び組成物
WO2009113989A1 (en) 2008-03-14 2009-09-17 Bionumerik Pharmaceuticals, Inc. Compositions and methods of use of compounds to increase cancer patient survival time
JP5759464B2 (ja) 2009-09-21 2015-08-05 ジェイダブリュー ファーマシューティカル コーポレイション オキサリプラチンのナノ粒子及びその製造方法
US20130096170A1 (en) 2011-10-14 2013-04-18 Hospira, Inc. Methods of treating pediatric patients using dexmedetomidine
AU2013202575B1 (en) * 2012-01-04 2013-05-16 Hospira, Inc. Dexmedetomidine premix formulation
US8242158B1 (en) 2012-01-04 2012-08-14 Hospira, Inc. Dexmedetomidine premix formulation
JP5314790B1 (ja) * 2012-07-09 2013-10-16 東和薬品株式会社 オキサリプラチン含有医薬組成物
ES2733061T3 (es) 2012-08-10 2019-11-27 Taiho Pharmaceutical Co Ltd Dispersión acuosa de liposomas encapsulantes de oxaliplatino estable y método para estabilización de la misma
KR102238677B1 (ko) 2012-09-07 2021-04-12 코히러스 바이오사이언시즈, 인코포레이티드 아달리무맙의 안정한 수성 제형
CN103690494B (zh) * 2013-11-29 2015-04-15 杭州华东医药集团新药研究院有限公司 一种低杂质含有奥沙利铂的组合物及其制备方法
BR112016030310A2 (pt) 2014-06-23 2017-08-22 Placon Therapeutics Inc Compostos de platina, composições e seus usos
AU2016289856B2 (en) 2015-07-07 2020-11-26 H. Lundbeck A/S PDE9 inhibitors with imidazo triazinone backbone and imidazo pyrazinone backbone for treatment of peripheral diseases
CN104940151A (zh) * 2015-07-23 2015-09-30 青岛蓝盛洋医药生物科技有限责任公司 一种抗癌药物奥沙利铂冻干粉针剂组合物
US11229702B1 (en) 2015-10-28 2022-01-25 Coherus Biosciences, Inc. High concentration formulations of adalimumab
US11071782B2 (en) 2016-04-20 2021-07-27 Coherus Biosciences, Inc. Method of filling a container with no headspace
WO2017192290A1 (en) 2016-05-04 2017-11-09 The Wistar Institute Of Anatomy And Biology Methods of treating cancers overexpressing carm1 with ezh2 inhibitors and platinum-based antineoplastic drugs
EP3481398A1 (de) 2016-07-06 2019-05-15 Imara, Inc. Pde9 -hemmer zur behandlung von peripheren erkrankungen
HRP20240146T1 (hr) 2017-05-26 2024-04-12 Cardurion Pharmaceuticals, Inc. Postupci dobivanja i upotrebe inhibitora pde9
SI3801526T1 (sl) 2018-05-25 2024-05-31 Cardurion Pharmaceuticals, Inc. Monohidratne in kristalinične oblike 6-((3s, 4s)-4-metil-1-(pirimidin-2-ilmetil)pirolidin-3-il)-3-tetrahidropiran-4- il-7h-imidazo (1.5 - a) pirazin-8-ona

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6041077B2 (ja) * 1976-09-06 1985-09-13 喜徳 喜谷 1,2‐ジアミノシクロヘキサン異性体のシス白金(2)錯体
IL83380A (en) * 1987-07-30 1991-04-15 Teva Pharma Stable aqueous cisplatin solutions
NL8901433A (nl) * 1989-06-06 1991-01-02 Pharmachemie Bv Carboplatinpreparaat.
JPH04185601A (ja) * 1990-11-20 1992-07-02 Unitika Ltd 白金抗癌剤徐放性製剤
JP2673331B2 (ja) * 1993-01-12 1997-11-05 田中貴金属工業 株式会社 光学的に高純度なシス―オキザラート(トランス―1―1,2―シクロヘキサンジアミン)白金(▲ii▼)
AU5416394A (en) * 1992-11-24 1994-06-22 Debiopharm S.A. Cisplatinum/oxaliplatinum combination
US5455270A (en) * 1993-08-11 1995-10-03 Bristol-Myers Squibb Co. Stabilized solutions of platinum(II) antitumor agents
DE69519300T2 (de) 1994-08-08 2001-05-31 Debiopharm Sa Stabiles arzneimittel enthaltend oxaliplatin

Also Published As

Publication number Publication date
UA42779C2 (uk) 2001-11-15
BR9508554A (pt) 1997-11-25
WO1996004904A1 (fr) 1996-02-22
US5716988A (en) 1998-02-10
IL114852A0 (en) 1995-12-08
EP0774963A1 (de) 1997-05-28
CN1154654A (zh) 1997-07-16
EP0774963B1 (de) 2000-11-02
CN1138541C (zh) 2004-02-18
KR100365171B1 (ko) 2003-02-19
CZ286714B6 (en) 2000-06-14
CA2196922C (fr) 2004-06-01
AU731981B2 (en) 2001-04-12
JPH10508289A (ja) 1998-08-18
KR970704434A (ko) 1997-09-06
RU2148400C1 (ru) 2000-05-10
DE69519300D1 (de) 2000-12-07
CZ37997A3 (en) 1997-06-11
JP3547755B2 (ja) 2004-07-28
DK0774963T3 (da) 2001-01-29
AU2252499A (en) 2000-03-23
CA2196922A1 (fr) 1996-02-22
AU2989695A (en) 2000-03-07
IL114852A (en) 2000-02-29
DE69519300T2 (de) 2001-05-31
ES2152412T3 (es) 2001-02-01

Similar Documents

Publication Publication Date Title
DE69519300D1 (de) Stabiles arzneimittel enthaltend oxaliplatin
HK12495A (en) Pharmaceutical formulations
RU94040387A (ru) Композиция, способствующая прекращению курения, никотиносодержащий распыляемый раствор, способ снижения потребности в курении табака, способ замены курения табака
PL325825A1 (en) Microemulsion for use as a carrier for administering active compounds
IT1270594B (it) Composizione farmaceutica a rilascio controllato di moguisteina in sospensione liquida
AU2001288460A1 (en) Compositions for treating sexual dysfunction, containing an no-donor and an antioxidant
ATE401892T1 (de) Verwendung von pharmazeutischen zubereitungen enthaltend oxcarbazepin im nüchternzustand
NO20023684D0 (no) Pediatrisk formulering
MXPA02008654A (es) Formulaciones de ranolazina de liberacion prolongada.
AU2506388A (en) Azelastine-containing medicaments for application in the nose and/or at the eye
CA2215327A1 (en) Formulations for lipophilic compounds
KR970025615A (ko) 암 전이 억제제
HK1046090A1 (en) Use of l-carnitine and its alkanoyl derivatives asosmotic agents in solutions for medical use
IE790194L (en) Pharmaceutical formulation
IL141232A0 (en) Use of camptothecin derivatives, with reduced gastrointestinal toxicity
KR870009716A (ko) 클로르페니라민 제형
ES404959A1 (es) Un procedimiento para preparar una composicion acuosa es- table de dexiciclina.
AU2001289762A1 (en) Pharmaceutical extemporary compositions
ATE203903T1 (de) Delta-aminolävulinsäure enthaltendes arzneimittel
PL350413A1 (en) Pharmaceutical effervescent formulation containing metamizol
KR900701263A (ko) 이보파민의 수용성 산 부가 염을 포함하는 안과용 약학 조성물
Lin et al. Toxicity of a single oral dose of N-ethylphenylacetamide in rats
AU2001266119A1 (en) Pharmaceutical composition in liquid form for oral administration of an active principle, with unpleasant, in particular bitter, taste
GB1386927A (en) Preparations for combatting swine dysentery
KR900000081A (ko) 트리암테렌의 약학적 액제

Legal Events

Date Code Title Description
UEP Publication of translation of european patent specification
EELV Lapsed due to withdrawal
REZ Deleted due to withdrawal