ATE119881T1 - 3-(2-(dimethylamino)ethyl>-n-methyl-1h-indol-5- methansulfonamid sulfat (2:1). - Google Patents

3-(2-(dimethylamino)ethyl>-n-methyl-1h-indol-5- methansulfonamid sulfat (2:1).

Info

Publication number
ATE119881T1
ATE119881T1 AT91311583T AT91311583T ATE119881T1 AT E119881 T1 ATE119881 T1 AT E119881T1 AT 91311583 T AT91311583 T AT 91311583T AT 91311583 T AT91311583 T AT 91311583T AT E119881 T1 ATE119881 T1 AT E119881T1
Authority
AT
Austria
Prior art keywords
indole
dimethylamino
ethyl
methyl
methanesulfonamide
Prior art date
Application number
AT91311583T
Other languages
German (de)
English (en)
Inventor
Joanne Craig
Derek Leslie Crookes
Stephen John Skittrall
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Application granted granted Critical
Publication of ATE119881T1 publication Critical patent/ATE119881T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • C07D209/16—Tryptamines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A61P29/02—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Indole Compounds (AREA)
AT91311583T 1990-12-12 1991-12-12 3-(2-(dimethylamino)ethyl>-n-methyl-1h-indol-5- methansulfonamid sulfat (2:1). ATE119881T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB909026998A GB9026998D0 (en) 1990-12-12 1990-12-12 Medicaments

Publications (1)

Publication Number Publication Date
ATE119881T1 true ATE119881T1 (de) 1995-04-15

Family

ID=10686904

Family Applications (1)

Application Number Title Priority Date Filing Date
AT91311583T ATE119881T1 (de) 1990-12-12 1991-12-12 3-(2-(dimethylamino)ethyl>-n-methyl-1h-indol-5- methansulfonamid sulfat (2:1).

Country Status (36)

Country Link
US (2) US5554639A (https=)
EP (1) EP0490689B1 (https=)
JP (1) JP2994037B2 (https=)
KR (1) KR100211479B1 (https=)
CN (2) CN1030890C (https=)
AP (1) AP230A (https=)
AT (1) ATE119881T1 (https=)
AU (1) AU650706B2 (https=)
BE (1) BE1005085A3 (https=)
CA (1) CA2098302C (https=)
CH (1) CH684192A5 (https=)
CY (1) CY2005A (https=)
CZ (1) CZ281931B6 (https=)
DE (1) DE69108200T2 (https=)
DK (1) DK0490689T3 (https=)
EG (1) EG20219A (https=)
ES (1) ES2069836T3 (https=)
FR (1) FR2670487B1 (https=)
GB (2) GB9026998D0 (https=)
GR (1) GR3015430T3 (https=)
HK (1) HK82697A (https=)
HU (1) HU211937A9 (https=)
IE (1) IE62894B1 (https=)
IL (1) IL100330A (https=)
IS (1) IS1706B (https=)
IT (1) IT1252868B (https=)
MX (1) MX9102501A (https=)
MY (1) MY109265A (https=)
NL (1) NL9102071A (https=)
NZ (1) NZ240942A (https=)
PT (1) PT99757B (https=)
RU (1) RU2108328C1 (https=)
TW (2) TW205035B (https=)
WO (1) WO1992010477A1 (https=)
YU (1) YU48926B (https=)
ZA (1) ZA919750B (https=)

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KR20080012360A (ko) 2005-05-20 2008-02-11 얀센 파마슈티카 엔.브이. 설파미드 유도체의 제조 방법
WO2007070504A2 (en) * 2005-12-13 2007-06-21 Morton Grove Pharmaceuticals, Inc. Stable and palatable oral liquid sumatriptan compositions
US8716231B2 (en) 2005-12-19 2014-05-06 Janssen Pharmaceutica Nv Use of benzo-fused heterocycle sulfamide derivatives for the treatment of pain
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JP2011526889A (ja) * 2008-06-30 2011-10-20 アフギン ファーマ，エルエルシー 局所局部的神経作用療法
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HK1244715A1 (zh) 2015-03-02 2018-08-17 阿福金制药有限责任公司 用大麻素的局部区域神经影响性疗法
US10383816B2 (en) 2015-03-02 2019-08-20 Afgin Pharma, Llc Topical regional neuro-affective therapy with cannabinoid combination products
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US20220096438A1 (en) 2018-09-07 2022-03-31 Upsher-Smith Laboratories, Llc Methods of treating migraine
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GB2162522B (en) * 1984-08-01 1988-02-24 Glaxo Group Ltd An indole derivative
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GB8928208D0 (en) * 1989-12-13 1990-02-14 Glaxo Group Ltd Medicaments

Also Published As

Publication number Publication date
BE1005085A3 (fr) 1993-04-13
EG20219A (en) 1997-11-30
CZ114093A3 (en) 1994-02-16
ZA919750B (en) 1992-10-28
MX9102501A (es) 1992-09-01
GR3015430T3 (en) 1995-06-30
DK0490689T3 (da) 1995-05-22
DE69108200D1 (de) 1995-04-20
JP2994037B2 (ja) 1999-12-27
IE914317A1 (en) 1992-06-17
WO1992010477A1 (en) 1992-06-25
IL100330A (en) 1996-06-18
IL100330A0 (en) 1992-09-06
US5554639A (en) 1996-09-10
EP0490689B1 (en) 1995-03-15
CY2005A (en) 1997-12-05
TW205035B (https=) 1993-05-01
AU650706B2 (en) 1994-06-30
ES2069836T3 (es) 1995-05-16
MY109265A (en) 1996-12-31
US5705520A (en) 1998-01-06
DE69108200T2 (de) 1995-07-20
CN1050831C (zh) 2000-03-29
PT99757A (pt) 1992-12-31
CA2098302C (en) 2001-10-16
AP9100339A0 (en) 1992-01-31
HK82697A (en) 1997-06-27
GB2251614A (en) 1992-07-15
CH684192A5 (fr) 1994-07-29
ITRM910922A0 (it) 1991-12-11
CN1128259A (zh) 1996-08-07
TW300886B (https=) 1997-03-21
ITRM910922A1 (it) 1993-06-11
CZ281931B6 (cs) 1997-04-16
NZ240942A (en) 1994-03-25
AP230A (en) 1993-01-27
FR2670487B1 (fr) 1993-08-20
CN1030890C (zh) 1996-02-07
IT1252868B (it) 1995-06-28
PT99757B (pt) 1999-05-31
GB2251614B (en) 1994-12-14
AU9072091A (en) 1992-07-08
CN1063099A (zh) 1992-07-29
IE62894B1 (en) 1995-03-08
NL9102071A (nl) 1992-07-01
GB9126297D0 (en) 1992-02-12
GB9026998D0 (en) 1991-01-30
KR100211479B1 (ko) 1999-08-02
HU211937A9 (en) 1996-01-29
JPH06503560A (ja) 1994-04-21
FR2670487A1 (fr) 1992-06-19
YU48926B (sh) 2002-12-10
IS3790A7 (is) 1992-06-13
EP0490689A1 (en) 1992-06-17
CA2098302A1 (en) 1992-06-13
RU2108328C1 (ru) 1998-04-10
YU191491A (sh) 1994-04-05
IS1706B (is) 1998-12-10

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Legal Events

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EELA Cancelled due to lapse of time