AT344332B - METHOD FOR PRODUCING NEW 2-TETRAHYDROFURFURYL-6,7-BENZOMORPHANES AND THEIR ACID ADDITION SALTS - Google Patents
METHOD FOR PRODUCING NEW 2-TETRAHYDROFURFURYL-6,7-BENZOMORPHANES AND THEIR ACID ADDITION SALTSInfo
- Publication number
- AT344332B AT344332B AT153875A AT153875A AT344332B AT 344332 B AT344332 B AT 344332B AT 153875 A AT153875 A AT 153875A AT 153875 A AT153875 A AT 153875A AT 344332 B AT344332 B AT 344332B
- Authority
- AT
- Austria
- Prior art keywords
- benzomorphanes
- tetrahydrofurfuryl
- acid addition
- addition salts
- producing new
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
- C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
- C07D221/22—Bridged ring systems
- C07D221/26—Benzomorphans
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Neurosurgery (AREA)
- Life Sciences & Earth Sciences (AREA)
- Neurology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pain & Pain Management (AREA)
- Pharmacology & Pharmacy (AREA)
- Biomedical Technology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE2411382A DE2411382C3 (en) | 1974-03-09 | 1974-03-09 | 2-Tetrahydrofurfuryl-6,7-benzomorphane, process for the preparation and their use |
Publications (2)
Publication Number | Publication Date |
---|---|
ATA153875A ATA153875A (en) | 1977-11-15 |
AT344332B true AT344332B (en) | 1978-07-10 |
Family
ID=5909593
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT153875A AT344332B (en) | 1974-03-09 | 1975-02-28 | METHOD FOR PRODUCING NEW 2-TETRAHYDROFURFURYL-6,7-BENZOMORPHANES AND THEIR ACID ADDITION SALTS |
Country Status (25)
Country | Link |
---|---|
JP (1) | JPS5827275B2 (en) |
AT (1) | AT344332B (en) |
BE (1) | BE826440A (en) |
BG (3) | BG24814A4 (en) |
CA (1) | CA1049511A (en) |
CH (8) | CH612425A5 (en) |
CS (1) | CS188221B2 (en) |
DD (1) | DD119236A5 (en) |
DE (1) | DE2411382C3 (en) |
DK (1) | DK137188C (en) |
ES (6) | ES440345A1 (en) |
FI (1) | FI63571C (en) |
FR (1) | FR2262984B1 (en) |
GB (1) | GB1496418A (en) |
HU (1) | HU177408B (en) |
IE (1) | IE40945B1 (en) |
IL (1) | IL46760A (en) |
NL (1) | NL7502724A (en) |
NO (1) | NO141800C (en) |
PH (1) | PH14127A (en) |
PL (3) | PL93499B1 (en) |
RO (2) | RO69617A (en) |
SE (1) | SE421919B (en) |
SU (3) | SU577982A3 (en) |
ZA (1) | ZA751394B (en) |
Families Citing this family (26)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2716687A1 (en) * | 1977-04-15 | 1978-10-19 | Boehringer Sohn Ingelheim | 2'-HYDROXY-2- (5-ISOXAZOLYLMETHYL) -6.7BENZOMORPHANES, THEIR ACID ADDITIONAL SALTS AND MEDICINAL PRODUCTS CONTAINING THEM |
DE2828039A1 (en) * | 1978-06-26 | 1980-01-10 | Boehringer Sohn Ingelheim | 2- (2-ALKOXYETHYL) -2'-HYDROXY-6,7-BENZOMORPHANES THEIR ACID ADDITION SALTS, THESE MEDICINAL PRODUCTS, AND METHOD FOR THE PRODUCTION THEREOF |
US6492420B2 (en) | 1995-03-10 | 2002-12-10 | Photocure As | Esters of 5-aminolevulinic acid as photosensitizing agents in photochemotherapy |
EP0820432B1 (en) * | 1995-03-10 | 2001-06-13 | PhotoCure ASA | Esters of 5-aminolevulinic acid as photosensitizing agents in photochemotherapy |
US6992107B1 (en) | 1995-03-10 | 2006-01-31 | Photocure Asa | Esters of 5-aminolevulinic acid and their use as photosensitizing compounds in photochemotherapy |
US7530461B2 (en) | 1995-03-10 | 2009-05-12 | Photocure Asa | Esters of 5-aminolevulinic acid as photosensitizing agents in photochemotherapy |
GB0018528D0 (en) | 2000-07-27 | 2000-09-13 | Photocure Asa | Compounds |
US6723750B2 (en) | 2002-03-15 | 2004-04-20 | Allergan, Inc. | Photodynamic therapy for pre-melanomas |
CL2008002199A1 (en) | 2007-07-26 | 2009-10-23 | Vitae Pharmaceuticals Inc | Compounds derived from 1,3-oxazin-2-one; pharmaceutical composition comprising said compounds; and use to treat a disease associated with the activity of 11beta-hydroxysteroid dehydrogenase type 1 (11beta-hsd1) such as dyslipidemia, hyperlipidemia, hypertension, obesity and cardiovascular disease, among others. |
AR069545A1 (en) | 2007-11-16 | 2010-02-03 | Boehringer Ingelheim Pharma | DERIVATIVES OF ARIL AND HETEROARILCARBONILO OF RELATED BENZOMORPHANS AND RELATED STRUCTURES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, OBTAINING THEMSELVES, THEIR USE IN THE TREATMENT OF DISEASES MEDIATED BY THE INHIBITION OF THE HIDDEN AND DISEASE |
JP5490014B2 (en) | 2007-12-11 | 2014-05-14 | ヴァイティー ファーマシューティカルズ,インコーポレイテッド | 11β-hydroxysteroid dehydrogenase type 1 cyclic urea inhibitor |
TW200934490A (en) | 2008-01-07 | 2009-08-16 | Vitae Pharmaceuticals Inc | Lactam inhibitors of 11 &abgr;-hydroxysteroid dehydrogenase 1 |
EP2252601B1 (en) | 2008-01-24 | 2012-12-19 | Vitae Pharmaceuticals, Inc. | Cyclic carbazate and semicarbazide inhibitors of 11beta-hydroxysteroid dehydrogenase 1 |
EP2254872A2 (en) | 2008-02-15 | 2010-12-01 | Vitae Pharmaceuticals, Inc. | Cycloalkyl lactame derivatives as inhibitors of 11-beta-hydroxysteroid dehydrogenase 1 |
CL2009001058A1 (en) | 2008-05-01 | 2010-09-10 | Vitae Pharmaceuticals Inc | Compounds derived from substituted oxazines, inhibitors of 11b-hydroxysteroid dehydrogenase type-1; pharmaceutical composition; and use of the compound to inhibit the activity of 11b-hsd1, as in the treatment of diabetes, dyslipidemia, hypertension, obesity, cancer, glaucoma, among others. |
BRPI0911764A2 (en) | 2008-05-01 | 2015-10-06 | Boehringer Ingelheim Int | cyclic inhibitors of 11betahydroxysteroid desigrogenase 1 |
CA2723034A1 (en) | 2008-05-01 | 2009-11-05 | Vitae Pharmaceuticals, Inc. | Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1 |
AR071719A1 (en) | 2008-05-13 | 2010-07-07 | Boehringer Ingelheim Int | ALICICLIC DERIVATIVES OF CARBOXILIC ACID OF BENZOMORPHANS AND RELATED STRUCTURES, MEDICINES CONTAINING THESE COMPOUNDS AND THEIR USE. OBTAINING PROCESSES |
TW201016691A (en) | 2008-07-25 | 2010-05-01 | Boehringer Ingelheim Int | Inhibitors of 11beta-hydroxysteroid dehydrogenase 1 |
US8114868B2 (en) | 2008-07-25 | 2012-02-14 | Boehringer Ingelheim International Gmbh | Cyclic inhibitors of 11β-hydroxysteroid dehydrogenase 1 |
MA33216B1 (en) | 2009-04-30 | 2012-04-02 | Boehringer Ingelheim Int | CYCLIC INHIBITORS OF 11BETA-HYDROXYSTEROID DEHYDROGENASE 1 |
US8927539B2 (en) | 2009-06-11 | 2015-01-06 | Vitae Pharmaceuticals, Inc. | Cyclic inhibitors of 11β-hydroxysteroid dehydrogenase 1 based on the 1,3-oxazinan-2-one structure |
AR078887A1 (en) | 2009-11-06 | 2011-12-07 | Boehringer Ingelheim Int | ARILO AND HETEROARILCARBONILO DERIVATIVES OF HEXAHYDROINDENOPIRIDINE AND OCTAHYDROBENZOQUINOLINE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM. |
EP2582698B1 (en) | 2010-06-16 | 2016-09-14 | Vitae Pharmaceuticals, Inc. | Substituted 5-,6- and 7-membered heterocycles, medicaments containing such compounds, and their use |
TWI537258B (en) | 2010-11-05 | 2016-06-11 | 百靈佳殷格翰國際股份有限公司 | Aryl-and heteroarylcarbonyl derivatives of hexahydroindenopyridine and octahydrobenzoquinoline |
JP2014524438A (en) | 2011-08-17 | 2014-09-22 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | Indenopyridine derivatives |
-
1974
- 1974-03-09 DE DE2411382A patent/DE2411382C3/en not_active Expired
-
1975
- 1975-02-28 AT AT153875A patent/AT344332B/en not_active IP Right Cessation
- 1975-03-05 SU SU7502110984A patent/SU577982A3/en active
- 1975-03-05 CH CH280275A patent/CH612425A5/en not_active IP Right Cessation
- 1975-03-06 FI FI750652A patent/FI63571C/en not_active IP Right Cessation
- 1975-03-07 SE SE7502592A patent/SE421919B/en not_active IP Right Cessation
- 1975-03-07 RO RO7589653A patent/RO69617A/en unknown
- 1975-03-07 FR FR7507239A patent/FR2262984B1/fr not_active Expired
- 1975-03-07 BG BG030538A patent/BG24814A4/en unknown
- 1975-03-07 HU HU75BO1536A patent/HU177408B/en unknown
- 1975-03-07 BG BG029183A patent/BG25087A3/en unknown
- 1975-03-07 RO RO7589654A patent/RO70051A/en unknown
- 1975-03-07 GB GB9633/75A patent/GB1496418A/en not_active Expired
- 1975-03-07 BE BE154138A patent/BE826440A/en not_active IP Right Cessation
- 1975-03-07 IL IL46760A patent/IL46760A/en unknown
- 1975-03-07 CA CA221,554A patent/CA1049511A/en not_active Expired
- 1975-03-07 DK DK92975A patent/DK137188C/en active
- 1975-03-07 ZA ZA751394A patent/ZA751394B/en unknown
- 1975-03-07 NO NO750773A patent/NO141800C/en unknown
- 1975-03-07 NL NL7502724A patent/NL7502724A/en not_active Application Discontinuation
- 1975-03-07 JP JP50027915A patent/JPS5827275B2/en not_active Expired
- 1975-03-07 DD DD184642A patent/DD119236A5/xx unknown
- 1975-03-07 BG BG030537A patent/BG24813A4/en unknown
- 1975-03-07 IE IE505/75A patent/IE40945B1/en unknown
- 1975-03-08 PL PL1975178582A patent/PL93499B1/pl unknown
- 1975-03-08 PL PL1975191318A patent/PL93699B1/pl unknown
- 1975-03-08 PL PL1975191319A patent/PL93700B1/pl unknown
- 1975-03-10 PH PH16895A patent/PH14127A/en unknown
- 1975-03-10 CS CS751583A patent/CS188221B2/en unknown
- 1975-08-20 ES ES440345A patent/ES440345A1/en not_active Expired
- 1975-08-20 ES ES440348A patent/ES440348A1/en not_active Expired
- 1975-08-20 ES ES440349A patent/ES440349A1/en not_active Expired
- 1975-08-20 ES ES440347A patent/ES440347A1/en not_active Expired
- 1975-08-20 ES ES440350A patent/ES440350A1/en not_active Expired
- 1975-08-20 ES ES440346A patent/ES440346A1/en not_active Expired
- 1975-12-19 SU SU752199295A patent/SU588916A3/en active
- 1975-12-19 SU SU7502199294A patent/SU577983A3/en active
-
1979
- 1979-04-24 CH CH384779A patent/CH622016A5/en not_active IP Right Cessation
- 1979-04-24 CH CH384679A patent/CH620440A5/en not_active IP Right Cessation
- 1979-04-24 CH CH384379A patent/CH620439A5/en not_active IP Right Cessation
- 1979-04-24 CH CH384579A patent/CH622015A5/en not_active IP Right Cessation
- 1979-04-24 CH CH384979A patent/CH622017A5/en not_active IP Right Cessation
- 1979-04-24 CH CH384879A patent/CH620681A5/en not_active IP Right Cessation
- 1979-04-24 CH CH384479A patent/CH622014A5/en not_active IP Right Cessation
Also Published As
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
ELJ | Ceased due to non-payment of the annual fee | ||
REN | Ceased due to non-payment of the annual fee |