RO69617A - PROCESS FOR THE PREPARATION OF 2-TETRAHYDRO-FURFURYL-6,7-BENZOMORPHANS - Google Patents

PROCESS FOR THE PREPARATION OF 2-TETRAHYDRO-FURFURYL-6,7-BENZOMORPHANS

Info

Publication number
RO69617A
RO69617A RO7589653A RO8965375A RO69617A RO 69617 A RO69617 A RO 69617A RO 7589653 A RO7589653 A RO 7589653A RO 8965375 A RO8965375 A RO 8965375A RO 69617 A RO69617 A RO 69617A
Authority
RO
Romania
Prior art keywords
benzomorphans
furfuryl
tetrahydro
preparation
Prior art date
Application number
RO7589653A
Other languages
French (fr)
Romanian (ro)
Inventor
Herbert Merz
Adolf Langbein
Gerhard Walther
Klaus Steckhaus
Original Assignee
C.H.Boehringer Sohn,De
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by C.H.Boehringer Sohn,De filed Critical C.H.Boehringer Sohn,De
Publication of RO69617A publication Critical patent/RO69617A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D221/00Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/22Bridged ring systems
    • C07D221/26Benzomorphans
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Neurosurgery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pain & Pain Management (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
RO7589653A 1974-03-09 1975-03-07 PROCESS FOR THE PREPARATION OF 2-TETRAHYDRO-FURFURYL-6,7-BENZOMORPHANS RO69617A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2411382A DE2411382C3 (en) 1974-03-09 1974-03-09 2-Tetrahydrofurfuryl-6,7-benzomorphane, process for the preparation and their use

Publications (1)

Publication Number Publication Date
RO69617A true RO69617A (en) 1980-08-15

Family

ID=5909593

Family Applications (2)

Application Number Title Priority Date Filing Date
RO7589653A RO69617A (en) 1974-03-09 1975-03-07 PROCESS FOR THE PREPARATION OF 2-TETRAHYDRO-FURFURYL-6,7-BENZOMORPHANS
RO7589654A RO70051A (en) 1974-03-09 1975-03-07 PROCESS FOR THE PREPARATION OF 2-TETRA-HYDROFURFURIL-6,7-BENZOMORPHANES

Family Applications After (1)

Application Number Title Priority Date Filing Date
RO7589654A RO70051A (en) 1974-03-09 1975-03-07 PROCESS FOR THE PREPARATION OF 2-TETRA-HYDROFURFURIL-6,7-BENZOMORPHANES

Country Status (25)

Country Link
JP (1) JPS5827275B2 (en)
AT (1) AT344332B (en)
BE (1) BE826440A (en)
BG (3) BG24814A4 (en)
CA (1) CA1049511A (en)
CH (8) CH612425A5 (en)
CS (1) CS188221B2 (en)
DD (1) DD119236A5 (en)
DE (1) DE2411382C3 (en)
DK (1) DK137188C (en)
ES (6) ES440345A1 (en)
FI (1) FI63571C (en)
FR (1) FR2262984B1 (en)
GB (1) GB1496418A (en)
HU (1) HU177408B (en)
IE (1) IE40945B1 (en)
IL (1) IL46760A (en)
NL (1) NL7502724A (en)
NO (1) NO141800C (en)
PH (1) PH14127A (en)
PL (3) PL93499B1 (en)
RO (2) RO69617A (en)
SE (1) SE421919B (en)
SU (3) SU577982A3 (en)
ZA (1) ZA751394B (en)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2716687A1 (en) * 1977-04-15 1978-10-19 Boehringer Sohn Ingelheim 2'-HYDROXY-2- (5-ISOXAZOLYLMETHYL) -6.7BENZOMORPHANES, THEIR ACID ADDITIONAL SALTS AND MEDICINAL PRODUCTS CONTAINING THEM
DE2828039A1 (en) * 1978-06-26 1980-01-10 Boehringer Sohn Ingelheim 2- (2-ALKOXYETHYL) -2'-HYDROXY-6,7-BENZOMORPHANES THEIR ACID ADDITION SALTS, THESE MEDICINAL PRODUCTS, AND METHOD FOR THE PRODUCTION THEREOF
US6492420B2 (en) 1995-03-10 2002-12-10 Photocure As Esters of 5-aminolevulinic acid as photosensitizing agents in photochemotherapy
EP0820432B1 (en) * 1995-03-10 2001-06-13 PhotoCure ASA Esters of 5-aminolevulinic acid as photosensitizing agents in photochemotherapy
US6992107B1 (en) 1995-03-10 2006-01-31 Photocure Asa Esters of 5-aminolevulinic acid and their use as photosensitizing compounds in photochemotherapy
US7530461B2 (en) 1995-03-10 2009-05-12 Photocure Asa Esters of 5-aminolevulinic acid as photosensitizing agents in photochemotherapy
GB0018528D0 (en) 2000-07-27 2000-09-13 Photocure Asa Compounds
US6723750B2 (en) 2002-03-15 2004-04-20 Allergan, Inc. Photodynamic therapy for pre-melanomas
CL2008002199A1 (en) 2007-07-26 2009-10-23 Vitae Pharmaceuticals Inc Compounds derived from 1,3-oxazin-2-one; pharmaceutical composition comprising said compounds; and use to treat a disease associated with the activity of 11beta-hydroxysteroid dehydrogenase type 1 (11beta-hsd1) such as dyslipidemia, hyperlipidemia, hypertension, obesity and cardiovascular disease, among others.
AR069545A1 (en) 2007-11-16 2010-02-03 Boehringer Ingelheim Pharma DERIVATIVES OF ARIL AND HETEROARILCARBONILO OF RELATED BENZOMORPHANS AND RELATED STRUCTURES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, OBTAINING THEMSELVES, THEIR USE IN THE TREATMENT OF DISEASES MEDIATED BY THE INHIBITION OF THE HIDDEN AND DISEASE
JP5490014B2 (en) 2007-12-11 2014-05-14 ヴァイティー ファーマシューティカルズ,インコーポレイテッド 11β-hydroxysteroid dehydrogenase type 1 cyclic urea inhibitor
TW200934490A (en) 2008-01-07 2009-08-16 Vitae Pharmaceuticals Inc Lactam inhibitors of 11 &abgr;-hydroxysteroid dehydrogenase 1
EP2252601B1 (en) 2008-01-24 2012-12-19 Vitae Pharmaceuticals, Inc. Cyclic carbazate and semicarbazide inhibitors of 11beta-hydroxysteroid dehydrogenase 1
EP2254872A2 (en) 2008-02-15 2010-12-01 Vitae Pharmaceuticals, Inc. Cycloalkyl lactame derivatives as inhibitors of 11-beta-hydroxysteroid dehydrogenase 1
CL2009001058A1 (en) 2008-05-01 2010-09-10 Vitae Pharmaceuticals Inc Compounds derived from substituted oxazines, inhibitors of 11b-hydroxysteroid dehydrogenase type-1; pharmaceutical composition; and use of the compound to inhibit the activity of 11b-hsd1, as in the treatment of diabetes, dyslipidemia, hypertension, obesity, cancer, glaucoma, among others.
BRPI0911764A2 (en) 2008-05-01 2015-10-06 Boehringer Ingelheim Int cyclic inhibitors of 11betahydroxysteroid desigrogenase 1
CA2723034A1 (en) 2008-05-01 2009-11-05 Vitae Pharmaceuticals, Inc. Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
AR071719A1 (en) 2008-05-13 2010-07-07 Boehringer Ingelheim Int ALICICLIC DERIVATIVES OF CARBOXILIC ACID OF BENZOMORPHANS AND RELATED STRUCTURES, MEDICINES CONTAINING THESE COMPOUNDS AND THEIR USE. OBTAINING PROCESSES
TW201016691A (en) 2008-07-25 2010-05-01 Boehringer Ingelheim Int Inhibitors of 11beta-hydroxysteroid dehydrogenase 1
US8114868B2 (en) 2008-07-25 2012-02-14 Boehringer Ingelheim International Gmbh Cyclic inhibitors of 11β-hydroxysteroid dehydrogenase 1
MA33216B1 (en) 2009-04-30 2012-04-02 Boehringer Ingelheim Int CYCLIC INHIBITORS OF 11BETA-HYDROXYSTEROID DEHYDROGENASE 1
US8927539B2 (en) 2009-06-11 2015-01-06 Vitae Pharmaceuticals, Inc. Cyclic inhibitors of 11β-hydroxysteroid dehydrogenase 1 based on the 1,3-oxazinan-2-one structure
AR078887A1 (en) 2009-11-06 2011-12-07 Boehringer Ingelheim Int ARILO AND HETEROARILCARBONILO DERIVATIVES OF HEXAHYDROINDENOPIRIDINE AND OCTAHYDROBENZOQUINOLINE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM.
EP2582698B1 (en) 2010-06-16 2016-09-14 Vitae Pharmaceuticals, Inc. Substituted 5-,6- and 7-membered heterocycles, medicaments containing such compounds, and their use
TWI537258B (en) 2010-11-05 2016-06-11 百靈佳殷格翰國際股份有限公司 Aryl-and heteroarylcarbonyl derivatives of hexahydroindenopyridine and octahydrobenzoquinoline
JP2014524438A (en) 2011-08-17 2014-09-22 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Indenopyridine derivatives

Also Published As

Publication number Publication date
CH622015A5 (en) 1981-03-13
IL46760A (en) 1978-12-17
PL93700B1 (en) 1977-06-30
NO141800C (en) 1980-06-04
CH620439A5 (en) 1980-11-28
CS188221B2 (en) 1979-02-28
FR2262984B1 (en) 1978-07-28
DK92975A (en) 1975-09-10
PH14127A (en) 1981-02-26
NO141800B (en) 1980-02-04
ES440345A1 (en) 1977-03-01
CH622017A5 (en) 1981-03-13
HU177408B (en) 1981-10-28
DE2411382C3 (en) 1979-09-06
JPS50123675A (en) 1975-09-29
FI63571B (en) 1983-03-31
ES440350A1 (en) 1977-03-16
DK137188B (en) 1978-01-30
SU577983A3 (en) 1977-10-25
FI750652A (en) 1975-09-10
PL93499B1 (en) 1977-05-30
CH612425A5 (en) 1979-07-31
CA1049511A (en) 1979-02-27
BE826440A (en) 1975-09-08
PL93699B1 (en) 1977-06-30
IL46760A0 (en) 1975-05-22
CH620440A5 (en) 1980-11-28
ES440349A1 (en) 1977-03-01
JPS5827275B2 (en) 1983-06-08
DE2411382A1 (en) 1975-09-18
DE2411382B2 (en) 1979-01-18
BG24814A4 (en) 1978-05-12
SU577982A3 (en) 1977-10-25
ATA153875A (en) 1977-11-15
DK137188C (en) 1978-07-03
DD119236A5 (en) 1976-04-12
ES440346A1 (en) 1977-03-01
IE40945B1 (en) 1979-09-12
AT344332B (en) 1978-07-10
AU7894275A (en) 1976-09-16
ES440348A1 (en) 1977-06-01
BG24813A4 (en) 1978-05-12
IE40945L (en) 1975-09-09
FR2262984A1 (en) 1975-10-03
CH622016A5 (en) 1981-03-13
NO750773L (en) 1975-09-10
GB1496418A (en) 1977-12-30
BG25087A3 (en) 1978-07-12
ZA751394B (en) 1976-11-24
SU588916A3 (en) 1978-01-15
CH622014A5 (en) 1981-03-13
SE7502592L (en) 1975-09-10
ES440347A1 (en) 1977-06-01
RO70051A (en) 1980-12-30
SE421919B (en) 1982-02-08
FI63571C (en) 1983-07-11
CH620681A5 (en) 1980-12-15
NL7502724A (en) 1975-09-11

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