AR213705A1 - Procedimiento para preparar(2-imidazolin-2-ilamino)-quinolinas,quinoxalinas y-quinazolinas sustituidas - Google Patents

Procedimiento para preparar(2-imidazolin-2-ilamino)-quinolinas,quinoxalinas y-quinazolinas sustituidas

Info

Publication number
AR213705A1
AR213705A1 AR246774A AR24677473A AR213705A1 AR 213705 A1 AR213705 A1 AR 213705A1 AR 246774 A AR246774 A AR 246774A AR 24677473 A AR24677473 A AR 24677473A AR 213705 A1 AR213705 A1 AR 213705A1
Authority
AR
Argentina
Prior art keywords
ilamine
quinoxalines
quinazolines
imidazolin
quinolines
Prior art date
Application number
AR246774A
Other languages
English (en)
Spanish (es)
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of AR213705A1 publication Critical patent/AR213705A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/18Halogen atoms or nitro radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38Nitrogen atoms
    • C07D215/40Nitrogen atoms attached in position 8
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D241/00Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/36Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems
    • C07D241/38Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems with only hydrogen or carbon atoms directly attached to the ring nitrogen atoms
    • C07D241/40Benzopyrazines
    • C07D241/42Benzopyrazines with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Cardiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
AR246774A 1972-02-29 1973-02-23 Procedimiento para preparar(2-imidazolin-2-ilamino)-quinolinas,quinoxalinas y-quinazolinas sustituidas AR213705A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB919672A GB1381979A (en) 1972-02-29 1972-02-29 Amino derivatives of quinoline quinoxaline and quinazoline
GB5162972 1972-11-08

Publications (1)

Publication Number Publication Date
AR213705A1 true AR213705A1 (es) 1979-03-15

Family

ID=26242776

Family Applications (1)

Application Number Title Priority Date Filing Date
AR246774A AR213705A1 (es) 1972-02-29 1973-02-23 Procedimiento para preparar(2-imidazolin-2-ilamino)-quinolinas,quinoxalinas y-quinazolinas sustituidas

Country Status (16)

Country Link
US (1) US3890319A (US06653308-20031125-C00199.png)
JP (2) JPS5754516B2 (US06653308-20031125-C00199.png)
AR (1) AR213705A1 (US06653308-20031125-C00199.png)
AU (1) AU471598B2 (US06653308-20031125-C00199.png)
BE (1) BE795970A (US06653308-20031125-C00199.png)
CA (1) CA981678A (US06653308-20031125-C00199.png)
CH (2) CH577500A5 (US06653308-20031125-C00199.png)
DE (1) DE2309160A1 (US06653308-20031125-C00199.png)
ES (2) ES411804A1 (US06653308-20031125-C00199.png)
FI (1) FI63757C (US06653308-20031125-C00199.png)
FR (1) FR2181776B1 (US06653308-20031125-C00199.png)
GB (1) GB1381979A (US06653308-20031125-C00199.png)
IE (1) IE37519B1 (US06653308-20031125-C00199.png)
MX (1) MX3042E (US06653308-20031125-C00199.png)
NL (1) NL159102B (US06653308-20031125-C00199.png)
SE (1) SE417204B (US06653308-20031125-C00199.png)

Families Citing this family (84)

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GB1463520A (en) * 1974-09-06 1977-02-02 Pfizer Ltd Process for the production of imidazolines
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US4188393A (en) 1977-04-22 1980-02-12 Sandoz Ltd. Treating spastic conditions or relaxing muscles
US4145421A (en) 1977-04-22 1979-03-20 Sandoz Ltd. Treating spastic conditions
FR2449087A2 (fr) * 1979-02-16 1980-09-12 Rhone Poulenc Ind Nouveaux derives de l'isoquinoleine, leur preparation et les compositions pharmaceutiques qui les contiennent
US4486432A (en) * 1982-09-30 1984-12-04 Eli Lilly And Company Quinoxalinedione leukotriene release inhibitors
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JPS6118950U (ja) * 1984-07-10 1986-02-03 財団法人鉄道総合技術研究所 トロリ線の給油装置
JPS63296814A (ja) * 1987-05-29 1988-12-02 Ishigaki Kiko Kk 集塵装置における濾材の目詰り除去装置
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US5326763A (en) * 1989-10-12 1994-07-05 Allergan, Inc. Methods for using (2-imidazolin-2-ylamino) quinoxaline derivatives
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US5077292A (en) * 1989-10-12 1991-12-31 Allergan, Inc. (2-imidazolin-2-ylamino) tetrahydroquinoxalines and methods for using same
US5204347A (en) * 1989-10-12 1993-04-20 Allergan, Inc. Methods for using (2-imidazolin-2-ylamino) tetrahydroquinoxalines
US5198442A (en) * 1989-10-12 1993-03-30 Allergan, Inc. (2-imidazolin-2-ylamino) quinoxaline derivatives and methods for using same
US5231096A (en) * 1989-10-12 1993-07-27 Allergan, Inc. Methods for using (2-imidazolin-2-ylamino) quinoxaline derivatives
US5021416A (en) * 1989-10-31 1991-06-04 Allergan, Inc. Method for using (2-imidazolin-2-ylamino) quinoxalines to reduce or maintain intraocular pressure
US5215991A (en) * 1990-01-26 1993-06-01 Allergan, Inc. Combination of selective alpha-adrenergic agonists and Na+ /H+ ex
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CN103827107A (zh) 2011-07-25 2014-05-28 阿勒根公司 作为α2肾上腺素能受体的调节剂的N-(咪唑烷-2-亚基)喹啉衍生物
GR1009419B (el) 2017-11-07 2018-12-14 Φαρματεν Αβεε Οφθαλμικο φαρμακευτικο σκευασμα που περιεχει εναν συνδυασμο βρινζολαμιδης και βριμονιδινης και μεθοδος για την παρασκευη αυτου

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Also Published As

Publication number Publication date
CA981678A (en) 1976-01-13
ES411804A1 (es) 1976-05-01
AU5198573A (en) 1974-08-08
MX3042E (es) 1980-03-04
NL159102B (nl) 1979-01-15
IE37519B1 (en) 1977-08-17
GB1381979A (en) 1975-01-29
JPS5625176A (en) 1981-03-10
CH577500A5 (US06653308-20031125-C00199.png) 1976-07-15
FR2181776A1 (US06653308-20031125-C00199.png) 1973-12-07
FI63757C (fi) 1983-08-10
CH576975A5 (US06653308-20031125-C00199.png) 1976-06-30
FR2181776B1 (US06653308-20031125-C00199.png) 1976-08-13
JPS5754516B2 (US06653308-20031125-C00199.png) 1982-11-18
NL7302799A (US06653308-20031125-C00199.png) 1973-08-31
DE2309160A1 (de) 1973-09-27
SE417204B (sv) 1981-03-02
ES412102A1 (es) 1976-05-16
JPS5745439B2 (US06653308-20031125-C00199.png) 1982-09-28
JPS4897878A (US06653308-20031125-C00199.png) 1973-12-13
IE37519L (en) 1973-08-29
FI63757B (fi) 1983-04-29
AU471598B2 (en) 1976-04-29
BE795970A (fr) 1973-08-27
US3890319A (en) 1975-06-17

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