AR197237A1 - Un procedimiento para preparar tiometilcefalosporinas 7-p-hidroxilfenilacetamido-3-heterociclicos - Google Patents

Un procedimiento para preparar tiometilcefalosporinas 7-p-hidroxilfenilacetamido-3-heterociclicos

Info

Publication number
AR197237A1
AR197237A1 AR248585A AR24858573A AR197237A1 AR 197237 A1 AR197237 A1 AR 197237A1 AR 248585 A AR248585 A AR 248585A AR 24858573 A AR24858573 A AR 24858573A AR 197237 A1 AR197237 A1 AR 197237A1
Authority
AR
Argentina
Prior art keywords
thyometilcefalosporins
hydroxylphenylacetamido
heterociclicos
preparing
procedure
Prior art date
Application number
AR248585A
Other languages
English (en)
Spanish (es)
Original Assignee
Smith Kline French Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US262903A external-priority patent/US3867380A/en
Priority claimed from US00289499A external-priority patent/US3855213A/en
Application filed by Smith Kline French Lab filed Critical Smith Kline French Lab
Application granted granted Critical
Publication of AR197237A1 publication Critical patent/AR197237A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/207-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/247-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/36Methylene radicals, substituted by sulfur atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/041,2,3-Triazoles; Hydrogenated 1,2,3-triazoles
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AR248585A 1972-06-14 1973-06-14 Un procedimiento para preparar tiometilcefalosporinas 7-p-hidroxilfenilacetamido-3-heterociclicos AR197237A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US262903A US3867380A (en) 1971-02-18 1972-06-14 3-Heterocyclic thiomethylcephalosporins
US00289499A US3855213A (en) 1971-02-18 1972-09-15 3-heterocyclic thiomethyl-cephalosporins

Publications (1)

Publication Number Publication Date
AR197237A1 true AR197237A1 (es) 1974-03-22

Family

ID=26949532

Family Applications (1)

Application Number Title Priority Date Filing Date
AR248585A AR197237A1 (es) 1972-06-14 1973-06-14 Un procedimiento para preparar tiometilcefalosporinas 7-p-hidroxilfenilacetamido-3-heterociclicos

Country Status (20)

Country Link
JP (2) JPS5518716B2 (da)
AR (1) AR197237A1 (da)
AT (1) AT324560B (da)
AU (1) AU464107B2 (da)
CA (2) CA1076560A (da)
CH (2) CH589093A5 (da)
DD (1) DD105238A5 (da)
DE (1) DE2316867C2 (da)
DK (1) DK142913B (da)
ES (2) ES412207A1 (da)
FI (1) FI56843C (da)
FR (2) FR2187298B1 (da)
GB (2) GB1363833A (da)
HU (1) HU168689B (da)
IE (2) IE37409B1 (da)
IL (1) IL42126A (da)
NL (2) NL7302817A (da)
PH (1) PH9941A (da)
PL (1) PL91074B1 (da)
SE (2) SE416472B (da)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR780000197B1 (en) * 1972-12-26 1978-05-26 Bristol Myers Co Method for preparing antibacterial agent
CA1035353A (en) * 1973-01-31 1978-07-25 Lee C. Cheney 3-thiolated-7-acylamidocephalosporanic acids
GB1476981A (en) * 1974-06-05 1977-06-16 Bristol Myers Co Substituted penicillanic acids
CA1074784A (en) * 1974-09-06 1980-04-01 Sumitomo Chemical Company N-ACYLAMINO-.alpha.-ARYLACETAMIDO CEPHALOSPORINS
JPS5346995A (en) * 1976-10-12 1978-04-27 Sangyo Kagaku Kenkyu Kyokai Antibacterial agents
NL162387C (nl) * 1977-09-06 1980-05-16 Gist Brocades Nv Werkwijze voor het bereiden van 6-(d-alpha-amino-p- -hydroxyfenylacetamido)penicillanzuur.
JPS6010226U (ja) * 1983-06-30 1985-01-24 松下電工株式会社 昇降装置
JPS6182606A (ja) * 1984-09-29 1986-04-26 東芝ライテック株式会社 昇降装置

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA698494B (en) * 1969-02-26 1971-07-28 Lilly Co Eli Sulfur-containing cephalosporing antibiotics
US3641021A (en) * 1969-04-18 1972-02-08 Lilly Co Eli 3 7-(ring-substituted) cephalosporin compounds

Also Published As

Publication number Publication date
CA999293A (en) 1976-11-02
SE416472B (sv) 1981-01-05
IE37499L (en) 1973-12-14
DK142913C (da) 1981-09-28
GB1363833A (en) 1974-08-21
NL7305206A (da) 1973-12-18
HU168689B (da) 1976-06-28
PL91074B1 (en) 1977-02-28
AU5234573A (en) 1974-08-22
FI56843B (fi) 1979-12-31
DE2316866A1 (de) 1974-01-03
AU464107B2 (en) 1975-08-14
IL42126A (en) 1975-12-31
JPS4931689A (da) 1974-03-22
IE37499B1 (en) 1977-08-03
DE2316867C2 (de) 1982-05-19
JPS5953274B2 (ja) 1984-12-24
IE37409B1 (en) 1977-07-20
FR2187299B1 (da) 1976-12-03
DE2316866B2 (de) 1976-10-07
FR2187298A1 (da) 1974-01-18
DD105238A5 (da) 1974-04-12
PH9941A (en) 1976-06-14
NL7302817A (da) 1973-12-18
IL42126A0 (en) 1973-06-29
CA1076560A (en) 1980-04-29
SE404190B (sv) 1978-09-25
FR2187298B1 (da) 1976-12-03
GB1358027A (en) 1974-06-26
IE37409L (en) 1973-12-14
JPS4954393A (da) 1974-05-27
ES412207A1 (es) 1976-01-01
FI56843C (fi) 1980-04-10
CH586709A5 (da) 1977-04-15
DK142913B (da) 1981-02-23
DE2316867A1 (de) 1974-01-03
FR2187299A1 (da) 1974-01-18
JPS5518716B2 (da) 1980-05-21
CH589093A5 (da) 1977-06-30
AT324560B (de) 1975-09-10
ES413501A1 (es) 1976-07-16

Similar Documents

Publication Publication Date Title
AR230991A1 (es) Un procedimiento para preparar nuevos derivados benzoxazolicos
AR195350A1 (es) Un procedimiento para preparar tri-p-toluensulfonato de s-adenosil-l-metionina
AR196130A1 (es) Un procedimiento para la preparacion de difenilil-alcanoilaminopiridinas
AR204984A1 (es) Procedimiento para preparar compuestos de 3-alcoxi-7-acilamido-cefem-4-carboxilico
AR194346A1 (es) Un procedimiento para preparar alcanodiaminas sustituidas
AR194803A1 (es) Un procedimiento para preparar urea
AR203004A1 (es) Procedimiento para la preparacion de un 1-aminobencimidazol
AR197237A1 (es) Un procedimiento para preparar tiometilcefalosporinas 7-p-hidroxilfenilacetamido-3-heterociclicos
AR216885A1 (es) Procedimiento para preparar aminonicotinonitrilos
AR198798A1 (es) Un procedimiento para preparar nuevas pirimidonas
AR200024A1 (es) Un procedimiento para preparar un compuesto de amidinourea
AR197206A1 (es) Procedimiento para preparar 6,7-substituido-quinazolinonas
AR192778A1 (es) Un procedimiento para preparar nuevos acidos benzoamidoacetohidroxamicos
AR197500A1 (es) Metodo para preparar un derivado de escopolamina
AR195346A1 (es) Metodo para preparar un polisacarido polihalogenohemiacetalico
AR208650A1 (es) Un procedimiento para la preparacion de 4alpha-aril-transdecahidroisoquinolinas
AR214849A1 (es) Procedimiento para preparar acidos sulfamilbenzoicos
AR203532A1 (es) Un procedimiento para la obtencion de nitroimidazolitriazolopiridazinas
AR210320A1 (es) Un procedimiento para preparar 4-oxo-2-imidazolidinilidenoureas
AR194979A1 (es) Un procedimiento para fabricar pasta
AR203833A1 (es) Procedimiento para preparar compuestos de 16-alfa-ciano-pregn-5-en-20-ona
AR200145A1 (es) Un procedimiento para preparar acidos fenilaceticos 3-alcoxi-5-sustituidos
AR207742A1 (es) Procedimiento para preparar(3-fosfonotioureido)ureidobencenos
AR193266A1 (es) Un procedimiento para preparar un compuesto derivado de proctaglandina
AR206778A1 (es) Procedimiento mejorado para preparar un derivado de cefalosporina