AR113965A1 - Triazol azoles ciclohexil ácidos como antagonistas de lpa - Google Patents

Triazol azoles ciclohexil ácidos como antagonistas de lpa

Info

Publication number
AR113965A1
AR113965A1 ARP180103701A ARP180103701A AR113965A1 AR 113965 A1 AR113965 A1 AR 113965A1 AR P180103701 A ARP180103701 A AR P180103701A AR P180103701 A ARP180103701 A AR P180103701A AR 113965 A1 AR113965 A1 AR 113965A1
Authority
AR
Argentina
Prior art keywords
alkyl
nrcrc
nrbc
orb
haloalkyl
Prior art date
Application number
ARP180103701A
Other languages
English (en)
Spanish (es)
Inventor
Shiwei Tao
Lawrence J Kennedy
Hao Zhang
Jun Shi
James R Corte
Tianan Fang
Jun Li
Ying Wang
Peter Tai Wah Cheng
Yan Shi
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of AR113965A1 publication Critical patent/AR113965A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
ARP180103701A 2017-12-19 2018-12-18 Triazol azoles ciclohexil ácidos como antagonistas de lpa AR113965A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201762607488P 2017-12-19 2017-12-19

Publications (1)

Publication Number Publication Date
AR113965A1 true AR113965A1 (es) 2020-07-01

Family

ID=65003581

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP180103701A AR113965A1 (es) 2017-12-19 2018-12-18 Triazol azoles ciclohexil ácidos como antagonistas de lpa

Country Status (16)

Country Link
US (1) US11319315B2 (enExample)
EP (1) EP3728224B1 (enExample)
JP (1) JP7280881B2 (enExample)
KR (1) KR20200100713A (enExample)
CN (1) CN111712492B (enExample)
AR (1) AR113965A1 (enExample)
AU (1) AU2018392325A1 (enExample)
BR (1) BR112020012177A2 (enExample)
CA (1) CA3085938A1 (enExample)
EA (1) EA202091505A1 (enExample)
ES (1) ES2938863T3 (enExample)
IL (1) IL275363A (enExample)
MX (1) MX2020005818A (enExample)
SG (1) SG11202005703TA (enExample)
TW (1) TW201927778A (enExample)
WO (1) WO2019126094A1 (enExample)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11312706B2 (en) * 2017-12-19 2022-04-26 Bristol-Myers Squibb Company Cyclohexyl acid pyrazole azines as LPA antagonists
WO2019126090A1 (en) 2017-12-19 2019-06-27 Bristol-Myers Squibb Company Triazole n-linked carbamoyl cyclohexyl acids as lpa antagonists
WO2020081410A2 (en) * 2018-10-15 2020-04-23 Bristol-Myers Squibb Company Radioligands for imaging the lpa1 receptor
CN111434653A (zh) * 2019-01-15 2020-07-21 武汉朗来科技发展有限公司 三氮唑类化合物及其制备方法与用途
EP3986553A1 (en) 2019-06-18 2022-04-27 Bristol-Myers Squibb Company Cyclobutyl carboxylic acids as lpa antagonists
CA3158743A1 (en) 2019-11-15 2021-05-20 Gilead Sciences, Inc. Triazole carbamate pyridyl sulfonamides as lpa receptor antagonists and uses thereof
TWI843503B (zh) 2020-06-03 2024-05-21 美商基利科學股份有限公司 Lpa受體拮抗劑及其用途
CA3185689A1 (en) 2020-06-03 2021-12-09 Gilead Sciences, Inc. Lpa receptor antagonists and uses thereof
EP4196220A1 (en) * 2020-08-11 2023-06-21 Viva Star Biosciences Limited Triazole-pyridinyl substituted azacyclohexyl acetic acid compounds as lpa receptor antagonists
EP4232431B1 (en) * 2020-10-22 2025-08-13 Lhotse Bio, Inc. Compounds and compositions for treating conditions associated with lpa receptor activity
CN114621135B (zh) * 2020-12-11 2024-01-30 上海拓界生物医药科技有限公司 一种lpa1小分子拮抗剂
CA3218917A1 (en) 2021-05-11 2022-11-17 Gilead Sciences, Inc. Lpa receptor antagonists and uses thereof
IL310708A (en) * 2021-08-12 2024-04-01 Shanghai Simr Biotechnology Co Ltd The history of converted triazole, a method for its preparation, its pharmaceutical preparation and its use
AU2022405082B2 (en) 2021-12-08 2025-09-25 Gilead Sciences, Inc. Lpa receptor antagonists and uses thereof
AR128613A1 (es) 2022-02-25 2024-05-29 Lhotse Bio Inc Compuestos y composiciones para el tratamiento de afecciones asociadas con la actividad del receptor de lpa
CN115785014B (zh) * 2022-12-27 2025-01-24 瑞石生物医药有限公司 四唑衍生物及其用途
WO2025029733A1 (en) 2023-08-01 2025-02-06 Discovery Energy, Llc Convertible silencer

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE60234318D1 (de) 2001-02-08 2009-12-24 Ono Pharmaceutical Co Mittel zur behandlung von harnwegserkrankungen, umfassend mittel zur kontrolle des lpa-rezeptors
DE102004038403B4 (de) 2004-08-07 2006-08-31 Sanofi-Aventis Deutschland Gmbh Verfahren zur Herstellung der enantiomeren Formen von cis-konfigurierten 3-Hydroxycyclohexancarbonsäure-Derivaten
US20080186971A1 (en) 2007-02-02 2008-08-07 Tarari, Inc. Systems and methods for processing access control lists (acls) in network switches using regular expression matching logic
CA2720490A1 (en) * 2008-04-04 2009-10-08 Irm Llc Compounds and compositions as itpkb inhibitors
EP2462128B1 (en) 2009-08-04 2016-09-21 Amira Pharmaceuticals, Inc. Compounds as lysophosphatidic acid receptor antagonists
GB2474748B (en) 2009-10-01 2011-10-12 Amira Pharmaceuticals Inc Polycyclic compounds as lysophosphatidic acid receptor antagonists
GB2474120B (en) 2009-10-01 2011-12-21 Amira Pharmaceuticals Inc Compounds as Lysophosphatidic acid receptor antagonists
BR112013014019A2 (pt) 2010-12-07 2016-09-13 Amira Pharmaceuticals Inc antagonistas do receptor do ácido lisofosfatídico e seus usos
US8785442B2 (en) 2011-01-30 2014-07-22 Curegenix, Inc. Compound as antagonist of lysophosphatidic acid receptor, composition, and use thereof
WO2012137982A2 (en) 2011-04-05 2012-10-11 Takeda Pharmaceutical Company Limited Sulfonamide derivative and use thereof
WO2012138648A1 (en) * 2011-04-06 2012-10-11 Irm Llc Compositions and methods for modulating lpa receptors
CA2848518C (en) * 2011-09-27 2019-06-18 Genfit Derivatives of 6-substituted triazolopyridazines as rev-erb agonists
WO2013070879A1 (en) 2011-11-10 2013-05-16 Bristol-Myers Squibb Company Methods for treating spinal cord injury with lpa receptor antagonists
US20140329871A1 (en) 2011-12-04 2014-11-06 Angion Biomedica Corp. Small molecule anti-fibrotic compounds and uses thereof
WO2013134298A1 (en) 2012-03-07 2013-09-12 Deciphera Pharmaceuticals, Llc Raf inhibitor compounds
PE20142305A1 (es) 2012-06-20 2015-01-16 Hoffmann La Roche Compuestos de n-ariltriazol como antagonistas de lpar
EP2864300A1 (en) * 2012-06-20 2015-04-29 F. Hoffmann-La Roche AG N-alkyltriazole compounds as lpar antagonists
JP6853619B2 (ja) * 2015-01-16 2021-03-31 大塚製薬株式会社 シアノトリアゾール化合物の医薬用途
AR108838A1 (es) 2016-06-21 2018-10-03 Bristol Myers Squibb Co Ácidos de carbamoiloximetil triazol ciclohexilo como antagonistas de lpa
WO2019126090A1 (en) 2017-12-19 2019-06-27 Bristol-Myers Squibb Company Triazole n-linked carbamoyl cyclohexyl acids as lpa antagonists

Also Published As

Publication number Publication date
CN111712492B (zh) 2024-05-31
EA202091505A1 (ru) 2020-09-22
US11319315B2 (en) 2022-05-03
IL275363A (en) 2020-07-30
ES2938863T3 (es) 2023-04-17
JP2021507900A (ja) 2021-02-25
KR20200100713A (ko) 2020-08-26
EP3728224A1 (en) 2020-10-28
CN111712492A (zh) 2020-09-25
WO2019126094A1 (en) 2019-06-27
JP7280881B2 (ja) 2023-05-24
TW201927778A (zh) 2019-07-16
BR112020012177A2 (pt) 2020-11-24
US20210163470A1 (en) 2021-06-03
MX2020005818A (es) 2020-08-20
SG11202005703TA (en) 2020-07-29
CA3085938A1 (en) 2019-06-27
EP3728224B1 (en) 2023-01-11
AU2018392325A1 (en) 2020-07-30

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