AR094706A1 - Proceso para producir compuesto de piridazinona y producción de sus intermediarios - Google Patents
Proceso para producir compuesto de piridazinona y producción de sus intermediariosInfo
- Publication number
- AR094706A1 AR094706A1 ARP140100519A ARP140100519A AR094706A1 AR 094706 A1 AR094706 A1 AR 094706A1 AR P140100519 A ARP140100519 A AR P140100519A AR P140100519 A ARP140100519 A AR P140100519A AR 094706 A1 AR094706 A1 AR 094706A1
- Authority
- AR
- Argentina
- Prior art keywords
- atom
- piridazinone
- intermediaries
- composite
- produce
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 2
- 239000002131 composite material Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 3
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 3
- WKBOTKDWSSQWDR-UHFFFAOYSA-N Bromine atom Chemical group [Br] WKBOTKDWSSQWDR-UHFFFAOYSA-N 0.000 abstract 2
- OAKJQQAXSVQMHS-UHFFFAOYSA-N Hydrazine Chemical compound NN OAKJQQAXSVQMHS-UHFFFAOYSA-N 0.000 abstract 2
- 229910052801 chlorine Inorganic materials 0.000 abstract 2
- 125000001309 chloro group Chemical group Cl* 0.000 abstract 2
- 229910052731 fluorine Inorganic materials 0.000 abstract 2
- 125000004178 (C1-C4) alkyl group Chemical group 0.000 abstract 1
- PXGOKWXKJXAPGV-UHFFFAOYSA-N Fluorine Chemical compound FF PXGOKWXKJXAPGV-UHFFFAOYSA-N 0.000 abstract 1
- 239000002841 Lewis acid Substances 0.000 abstract 1
- 125000004429 atom Chemical group 0.000 abstract 1
- 239000011737 fluorine Substances 0.000 abstract 1
- 125000001153 fluoro group Chemical group F* 0.000 abstract 1
- 150000007517 lewis acids Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
- C07D237/06—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D237/10—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D237/12—Halogen atoms or nitro radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
- C07D237/06—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D237/10—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D237/14—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C51/00—Preparation of carboxylic acids or their salts, halides or anhydrides
- C07C51/347—Preparation of carboxylic acids or their salts, halides or anhydrides by reactions not involving formation of carboxyl groups
- C07C51/353—Preparation of carboxylic acids or their salts, halides or anhydrides by reactions not involving formation of carboxyl groups by isomerisation; by change of size of the carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C51/00—Preparation of carboxylic acids or their salts, halides or anhydrides
- C07C51/347—Preparation of carboxylic acids or their salts, halides or anhydrides by reactions not involving formation of carboxyl groups
- C07C51/373—Preparation of carboxylic acids or their salts, halides or anhydrides by reactions not involving formation of carboxyl groups by introduction of functional groups containing oxygen only in doubly bound form
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
- C07C59/40—Unsaturated compounds
- C07C59/76—Unsaturated compounds containing keto groups
- C07C59/88—Unsaturated compounds containing keto groups containing halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
- C07C59/40—Unsaturated compounds
- C07C59/76—Unsaturated compounds containing keto groups
- C07C59/90—Unsaturated compounds containing keto groups containing singly bound oxygen-containing groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C67/00—Preparation of carboxylic acid esters
- C07C67/30—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group
- C07C67/333—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group by isomerisation; by change of size of the carbon skeleton
- C07C67/343—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C67/00—Preparation of carboxylic acid esters
- C07C67/475—Preparation of carboxylic acid esters by splitting of carbon-to-carbon bonds and redistribution, e.g. disproportionation or migration of groups between different molecules
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/66—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety
- C07C69/67—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety of saturated acids
- C07C69/675—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety of saturated acids of saturated hydroxy-carboxylic acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/66—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety
- C07C69/73—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety of unsaturated acids
- C07C69/738—Esters of keto-carboxylic acids or aldehydo-carboxylic acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
- C07D237/06—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D237/08—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D307/60—Two oxygen atoms, e.g. succinic anhydride
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Materials Engineering (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Reivindicación 1: Un proceso para producir un compuesto de la fórmula (1), caracterizado porque X representa un átomo de hidrógeno, un átomo de flúor, un átomo de cloro o un átomo de bromo e Y representa un átomo de hidrógeno, un átomo de flúor, un átomo de cloro o un átomo de bromo; que comprende la etapa 1 de reacción de un compuesto de la fórmula (2) y un compuesto de la fórmula (3) en presencia de un ácido de Lewis para obtener un aducto; en donde R representa un átomo de hidrógeno o un grupo alquilo C₁₋₄ y X tiene el mismo significado que el descrito con anterioridad, en donde Y tiene el mismo significado que el descrito con anterioridad; y la etapa 2 de reacción del aducto obtenido en la etapa 1 e hidrazina
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2013031766 | 2013-02-21 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR094706A1 true AR094706A1 (es) | 2015-08-19 |
Family
ID=51391391
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP140100519A AR094706A1 (es) | 2013-02-21 | 2014-02-19 | Proceso para producir compuesto de piridazinona y producción de sus intermediarios |
Country Status (21)
Country | Link |
---|---|
US (1) | US9650347B2 (es) |
EP (1) | EP2958899B1 (es) |
JP (2) | JP6311719B2 (es) |
KR (1) | KR102136440B1 (es) |
CN (1) | CN105008334B (es) |
AR (1) | AR094706A1 (es) |
AU (1) | AU2014219681B2 (es) |
BR (1) | BR112015019305A2 (es) |
CA (1) | CA2901586A1 (es) |
CR (1) | CR20150387A (es) |
EC (1) | ECSP15035268A (es) |
ES (1) | ES2648662T3 (es) |
GT (1) | GT201500225A (es) |
HU (1) | HUE035927T2 (es) |
IL (1) | IL239987A (es) |
MX (1) | MX359645B (es) |
PH (1) | PH12015501717A1 (es) |
PL (1) | PL2958899T3 (es) |
RU (1) | RU2654058C2 (es) |
TW (1) | TWI603959B (es) |
WO (1) | WO2014129612A1 (es) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BR112015024291A2 (pt) | 2013-03-26 | 2017-07-18 | Sumitomo Chemical Co | método de produção de composto de piridazinona |
US9732042B2 (en) | 2013-05-24 | 2017-08-15 | Sumitomo Chemical Company, Limited | Method for producing pyridazine compound |
TW201922682A (zh) * | 2017-10-27 | 2019-06-16 | 日商住友化學股份有限公司 | 苯甲醯甲酸化合物及嗒化合物之製造方法 |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CS205592B1 (cs) * | 1978-11-27 | 1981-05-29 | Ervin Sohler | Spósob výroby 2-fenyl-4,5-dichlórpyridazín-3-ónu |
PL1767529T3 (pl) * | 2004-06-09 | 2009-10-30 | Sumitomo Chemical Co | Pirydazynowy związek oraz jego zastosowanie |
WO2007044796A2 (en) * | 2005-10-11 | 2007-04-19 | Nps Pharmaceuticals, Inc. | Pyridazinone compounds as calcilytics |
JP2010006722A (ja) * | 2008-06-25 | 2010-01-14 | Hokko Chem Ind Co Ltd | ピリダジン誘導体および殺菌剤 |
AU2009296852A1 (en) | 2008-09-24 | 2010-04-01 | E. I. Du Pont De Nemours And Company | Fungicidal pyridazines |
JP5857511B2 (ja) * | 2010-08-10 | 2016-02-10 | 住友化学株式会社 | 植物病害防除組成物およびその用途 |
BR112015024291A2 (pt) | 2013-03-26 | 2017-07-18 | Sumitomo Chemical Co | método de produção de composto de piridazinona |
US9732042B2 (en) | 2013-05-24 | 2017-08-15 | Sumitomo Chemical Company, Limited | Method for producing pyridazine compound |
-
2014
- 2014-02-18 PL PL14753644T patent/PL2958899T3/pl unknown
- 2014-02-18 ES ES14753644.5T patent/ES2648662T3/es active Active
- 2014-02-18 US US14/767,533 patent/US9650347B2/en active Active
- 2014-02-18 WO PCT/JP2014/054251 patent/WO2014129612A1/en active Application Filing
- 2014-02-18 HU HUE14753644A patent/HUE035927T2/en unknown
- 2014-02-18 MX MX2015010352A patent/MX359645B/es active IP Right Grant
- 2014-02-18 EP EP14753644.5A patent/EP2958899B1/en not_active Not-in-force
- 2014-02-18 CN CN201480009536.8A patent/CN105008334B/zh active Active
- 2014-02-18 RU RU2015135184A patent/RU2654058C2/ru not_active IP Right Cessation
- 2014-02-18 JP JP2015540943A patent/JP6311719B2/ja active Active
- 2014-02-18 CA CA2901586A patent/CA2901586A1/en active Pending
- 2014-02-18 AU AU2014219681A patent/AU2014219681B2/en not_active Ceased
- 2014-02-18 KR KR1020157022457A patent/KR102136440B1/ko active IP Right Grant
- 2014-02-18 BR BR112015019305A patent/BR112015019305A2/pt active Search and Examination
- 2014-02-19 TW TW103105450A patent/TWI603959B/zh not_active IP Right Cessation
- 2014-02-19 AR ARP140100519A patent/AR094706A1/es not_active Application Discontinuation
-
2015
- 2015-07-16 IL IL239987A patent/IL239987A/en not_active IP Right Cessation
- 2015-07-22 CR CR20150387A patent/CR20150387A/es unknown
- 2015-08-04 PH PH12015501717A patent/PH12015501717A1/en unknown
- 2015-08-12 GT GT201500225A patent/GT201500225A/es unknown
- 2015-08-14 EC ECIEPI201535268A patent/ECSP15035268A/es unknown
-
2017
- 2017-09-11 JP JP2017173777A patent/JP6436204B2/ja active Active
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
MX2015002616A (es) | Sintesis de bis(fluorosulfonil)imida. | |
PE20180327A1 (es) | Proceso para preparar 4-amino-piridazinas | |
CU24410B1 (es) | Benzimidazol-2-aminas como inhibidores de midh1 | |
EA201890752A1 (ru) | Способ получения противогрибковых соединений | |
DOP2015000187A (es) | Proceso de fabricación de vortioxetina | |
MX2016005496A (es) | Sintesis de fluorotrifluorometilsulfonil-imida. | |
CY1118945T1 (el) | Μεθοδος και ενδιαμεσα για την παρασκευη πρεγκαμπαλινης | |
AR105812A1 (es) | Métodos para la preparación de inhibidores de proteína deacetilasa | |
CL2019000016A1 (es) | Procesos novedosos para preparar estimuladores de guanilato ciclasa soluble. | |
AR085052A1 (es) | Metodos para producir un compuesto profarmaco inhibidor de la union al vih e intermediarios | |
TR201904928T4 (tr) | Tereftalik asit diesterlerin resirküle alkol dehidratasyonu ile üretimi için yöntem. | |
AR101136A1 (es) | Proceso para la preparación de ácidos 3-hidroxipicolínicos | |
CY1121116T1 (el) | Νεα μεθοδος για την συνθεση αγομελατινης | |
AR094706A1 (es) | Proceso para producir compuesto de piridazinona y producción de sus intermediarios | |
MX2019004024A (es) | Metodo para preparar acetofenonas sustituidas con ciclopropilo. | |
AR092355A1 (es) | Fluoruros de fluoropicolinoilo y procesos para su preparacion | |
AR098879A1 (es) | Síntesis de ent-progesterona y sus productos intermedios | |
MX2016013586A (es) | Tinturas reactivas fluorescentes, proceso para su produccion y su uso. | |
EA201491463A1 (ru) | Способ получения соединения по новой реакции присоединения михаэля с применением воды или различных кислот в качестве добавки | |
CR20130655A (es) | Métodos de producción de derivados de imidazol | |
MX2015014728A (es) | Sintesis de inhibidores de beta secretasa (bace). | |
BR112017003121A2 (pt) | método para a síntese de um óxido de fosfina de hidrogênio heterocíclico | |
MX2018006638A (es) | Un proceso para la preparacion de acidos de 2-alquilo-4-trifluorom etil-3-alquilosulfonilbenzoico por la oxidacion de tioeter quimoselectivo. | |
MX2015017747A (es) | Proceso para producir 2-fenil-1, 3-benzoxazoles. | |
BR112015017326A2 (pt) | processo para a produção de 2-alquil-3-butin-2-óis |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG | Grant, registration | ||
FD | Application declared void or lapsed, e.g., due to non-payment of fee |