CR20150387A - Proceso para producir compuesto de piridazinona y producción de sus intermediarios - Google Patents

Proceso para producir compuesto de piridazinona y producción de sus intermediarios

Info

Publication number
CR20150387A
CR20150387A CR20150387A CR20150387A CR20150387A CR 20150387 A CR20150387 A CR 20150387A CR 20150387 A CR20150387 A CR 20150387A CR 20150387 A CR20150387 A CR 20150387A CR 20150387 A CR20150387 A CR 20150387A
Authority
CR
Costa Rica
Prior art keywords
piridazinone
intermediaries
composite
produce
production
Prior art date
Application number
CR20150387A
Other languages
English (en)
Inventor
Yasuyuki Nakae
Akio Manabe
Takashi Miyamoto
Original Assignee
Sumitomo Chemical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sumitomo Chemical Co filed Critical Sumitomo Chemical Co
Publication of CR20150387A publication Critical patent/CR20150387A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
    • C07D237/06—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D237/10—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D237/12—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C51/00—Preparation of carboxylic acids or their salts, halides or anhydrides
    • C07C51/347—Preparation of carboxylic acids or their salts, halides or anhydrides by reactions not involving formation of carboxyl groups
    • C07C51/353—Preparation of carboxylic acids or their salts, halides or anhydrides by reactions not involving formation of carboxyl groups by isomerisation; by change of size of the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C51/00—Preparation of carboxylic acids or their salts, halides or anhydrides
    • C07C51/347—Preparation of carboxylic acids or their salts, halides or anhydrides by reactions not involving formation of carboxyl groups
    • C07C51/373—Preparation of carboxylic acids or their salts, halides or anhydrides by reactions not involving formation of carboxyl groups by introduction of functional groups containing oxygen only in doubly bound form
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/40—Unsaturated compounds
    • C07C59/76—Unsaturated compounds containing keto groups
    • C07C59/88—Unsaturated compounds containing keto groups containing halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/40—Unsaturated compounds
    • C07C59/76—Unsaturated compounds containing keto groups
    • C07C59/90—Unsaturated compounds containing keto groups containing singly bound oxygen-containing groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C67/00—Preparation of carboxylic acid esters
    • C07C67/30—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group
    • C07C67/333—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group by isomerisation; by change of size of the carbon skeleton
    • C07C67/343—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C67/00—Preparation of carboxylic acid esters
    • C07C67/475—Preparation of carboxylic acid esters by splitting of carbon-to-carbon bonds and redistribution, e.g. disproportionation or migration of groups between different molecules
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
    • C07C69/66—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety
    • C07C69/67—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety of saturated acids
    • C07C69/675—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety of saturated acids of saturated hydroxy-carboxylic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
    • C07C69/66—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety
    • C07C69/73—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety of unsaturated acids
    • C07C69/738—Esters of keto-carboxylic acids or aldehydo-carboxylic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
    • C07D237/06—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D237/08—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
    • C07D237/06—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D237/10—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D237/14—Oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D307/60—Two oxygen atoms, e.g. succinic anhydride

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Materials Engineering (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

La presente invención se refiere a un proceso para producir un compuesto de la fórmula (1) en donde X representa un átomo de hidrógeno, etc., e Y representa un átomo de hidrógeno, etc., que comprende la etapa 1 de reacción de un compuesto de la fórmula (2) y un compuesto de la fórmula (3) en presencia de un ácido de Lewis en donde R representa un átomo de hidrógeno, etc., para obtener un aducto, y la etapa 2 de reacción del aducto obtenido en la etapa 1 e hidrazina para obtener el compuesto de la fórmula.
CR20150387A 2013-02-21 2015-07-22 Proceso para producir compuesto de piridazinona y producción de sus intermediarios CR20150387A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2013031766 2013-02-21
PCT/JP2014/054251 WO2014129612A1 (en) 2013-02-21 2014-02-18 Process for producing pyridazinone compound and production intermediates thereof

Publications (1)

Publication Number Publication Date
CR20150387A true CR20150387A (es) 2015-11-02

Family

ID=51391391

Family Applications (1)

Application Number Title Priority Date Filing Date
CR20150387A CR20150387A (es) 2013-02-21 2015-07-22 Proceso para producir compuesto de piridazinona y producción de sus intermediarios

Country Status (21)

Country Link
US (1) US9650347B2 (es)
EP (1) EP2958899B1 (es)
JP (2) JP6311719B2 (es)
KR (1) KR102136440B1 (es)
CN (1) CN105008334B (es)
AR (1) AR094706A1 (es)
AU (1) AU2014219681B2 (es)
BR (1) BR112015019305A2 (es)
CA (1) CA2901586A1 (es)
CR (1) CR20150387A (es)
EC (1) ECSP15035268A (es)
ES (1) ES2648662T3 (es)
GT (1) GT201500225A (es)
HU (1) HUE035927T2 (es)
IL (1) IL239987A (es)
MX (1) MX359645B (es)
PH (1) PH12015501717A1 (es)
PL (1) PL2958899T3 (es)
RU (1) RU2654058C2 (es)
TW (1) TWI603959B (es)
WO (1) WO2014129612A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2014157021A1 (ja) 2013-03-26 2014-10-02 住友化学株式会社 ピリダジノン化合物の製造方法
EP3004065B1 (en) * 2013-05-24 2017-10-18 Sumitomo Chemical Company, Limited Method for producing pyridazine compound
TW201922682A (zh) * 2017-10-27 2019-06-16 日商住友化學股份有限公司 苯甲醯甲酸化合物及嗒化合物之製造方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CS205592B1 (cs) * 1978-11-27 1981-05-29 Ervin Sohler Spósob výroby 2-fenyl-4,5-dichlórpyridazín-3-ónu
ES2324883T3 (es) 2004-06-09 2009-08-18 Sumitomo Chemical Company, Limited Compuesto de piridazina y su utilizacion.
WO2007044796A2 (en) * 2005-10-11 2007-04-19 Nps Pharmaceuticals, Inc. Pyridazinone compounds as calcilytics
JP2010006722A (ja) * 2008-06-25 2010-01-14 Hokko Chem Ind Co Ltd ピリダジン誘導体および殺菌剤
US20110136762A1 (en) 2008-09-24 2011-06-09 E.I. Du Pont De Nemours And Company Fungicidal pyridazines
JP5857511B2 (ja) * 2010-08-10 2016-02-10 住友化学株式会社 植物病害防除組成物およびその用途
WO2014157021A1 (ja) 2013-03-26 2014-10-02 住友化学株式会社 ピリダジノン化合物の製造方法
EP3004065B1 (en) 2013-05-24 2017-10-18 Sumitomo Chemical Company, Limited Method for producing pyridazine compound

Also Published As

Publication number Publication date
KR20150118157A (ko) 2015-10-21
WO2014129612A1 (en) 2014-08-28
EP2958899B1 (en) 2017-10-11
JP6436204B2 (ja) 2018-12-12
GT201500225A (es) 2016-09-23
MX359645B (es) 2018-10-04
PH12015501717B1 (en) 2015-11-09
PH12015501717A1 (en) 2015-11-09
JP2016510718A (ja) 2016-04-11
PL2958899T3 (pl) 2018-01-31
IL239987A (en) 2017-07-31
JP2018027957A (ja) 2018-02-22
AU2014219681A1 (en) 2015-07-30
AU2014219681B2 (en) 2017-07-20
TWI603959B (zh) 2017-11-01
IL239987A0 (en) 2015-09-24
TW201437201A (zh) 2014-10-01
AR094706A1 (es) 2015-08-19
RU2654058C2 (ru) 2018-05-16
KR102136440B1 (ko) 2020-07-21
EP2958899A1 (en) 2015-12-30
CN105008334A (zh) 2015-10-28
US9650347B2 (en) 2017-05-16
BR112015019305A2 (pt) 2017-07-18
HUE035927T2 (en) 2018-05-28
EP2958899A4 (en) 2016-07-06
CN105008334B (zh) 2017-11-03
MX2015010352A (es) 2015-10-09
CA2901586A1 (en) 2014-08-28
ES2648662T3 (es) 2018-01-05
US20150376138A1 (en) 2015-12-31
ECSP15035268A (es) 2015-11-30
RU2015135184A (ru) 2017-03-24
JP6311719B2 (ja) 2018-04-18

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