AR063646A1 - Proceso para la sulfinilacion de un derivado de pirazol - Google Patents
Proceso para la sulfinilacion de un derivado de pirazolInfo
- Publication number
- AR063646A1 AR063646A1 ARP070105012A ARP070105012A AR063646A1 AR 063646 A1 AR063646 A1 AR 063646A1 AR P070105012 A ARP070105012 A AR P070105012A AR P070105012 A ARP070105012 A AR P070105012A AR 063646 A1 AR063646 A1 AR 063646A1
- Authority
- AR
- Argentina
- Prior art keywords
- acid
- trifluoromethylsulfinic
- trifluoromethyl
- sulfinilation
- salt
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/44—Oxygen and nitrogen or sulfur and nitrogen atoms
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Communicable Diseases (AREA)
- Zoology (AREA)
- Oncology (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- Wood Science & Technology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Environmental Sciences (AREA)
- Epidemiology (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Catalysts (AREA)
Abstract
Un proceso para la sulfinilación de un derivado de pirazol, caracterizado porque se hace reaccionar 5-amino-1-[2,6-dicloro-4-(trifluorometil)fenil]-1H-pirazol-3-carbonitrilo de fórmula (2) con un agente de sulfinilación seleccionado de árido trifluorometilsulfínico, anhídrido de ácido trifluorometilsulfínico y una sal de metal trifluorometilsulfinato alcalino o alcalinotérreo y mezclas del ácido y/o de la(s) sal(es), en presencia de al menos un complejo de amina ácida, en donde la(s) amina(s) es/son seleccionada(s) de aminas terciarias y el/los ácido(s) es/son seleccionado(s) de ácido fluorhídrico, clorhídrico, bromhídrico y yodhídrico, y derivados del ácido sulfónico, y con la adición de un agente halogenante.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US86517806P | 2006-11-10 | 2006-11-10 | |
| US91361707P | 2007-04-24 | 2007-04-24 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR063646A1 true AR063646A1 (es) | 2009-02-04 |
Family
ID=39167843
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP070105012A AR063646A1 (es) | 2006-11-10 | 2007-11-09 | Proceso para la sulfinilacion de un derivado de pirazol |
Country Status (22)
| Country | Link |
|---|---|
| US (2) | US8263783B2 (es) |
| EP (1) | EP2081908B1 (es) |
| JP (1) | JP5450077B2 (es) |
| KR (1) | KR20090083453A (es) |
| CN (1) | CN102746233A (es) |
| AR (1) | AR063646A1 (es) |
| AU (1) | AU2007316718B2 (es) |
| BR (1) | BRPI0718774A2 (es) |
| CA (1) | CA2667559A1 (es) |
| DK (1) | DK2081908T3 (es) |
| EA (1) | EA200900629A1 (es) |
| ES (1) | ES2422296T3 (es) |
| HR (1) | HRP20130582T1 (es) |
| IL (1) | IL198259A (es) |
| MA (1) | MA30917B1 (es) |
| MX (1) | MX2009004262A (es) |
| NZ (1) | NZ576594A (es) |
| PL (1) | PL2081908T3 (es) |
| PT (1) | PT2081908E (es) |
| TW (1) | TWI413498B (es) |
| WO (1) | WO2008055877A1 (es) |
| ZA (1) | ZA200903968B (es) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5396085B2 (ja) | 2005-12-14 | 2014-01-22 | マクテシム・ケミカル・ワークス・リミテツド | ５−アミノ−１−［２，６−ジクロロ−４−（トリフルオロメチル）フェニル］−４−［（トリフルオロメチル）スルフィニル］−１ｈ−ピラゾール−３−カルボニトリルの多形および非晶形 |
| CA2667562A1 (en) | 2006-11-10 | 2008-05-15 | Basf Se | Process for the sulfinylation of a pyrazole derivative |
| DK2349987T3 (da) * | 2008-10-02 | 2013-03-11 | Basf Se | Fremgangsmåde til fremstilling og oprensning af trifluormethansulfinsyre |
| EP3412658A1 (en) * | 2017-06-09 | 2018-12-12 | Solvay Sa | Processes for the manufacture of sulfur-substitued pyrazole derivatives |
| EP3412659A1 (en) * | 2017-06-09 | 2018-12-12 | Solvay Sa | Processes for the manufacture of sulfur-substituted pyrazole derivatives |
| EP3941907A4 (en) * | 2019-03-19 | 2023-01-04 | Gharda Chemicals Limited | FIPRONIL SYNTHESIS METHOD |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2716453B1 (fr) * | 1994-02-22 | 1996-03-29 | Rhone Poulenc Agrochimie | Procédé de sulfinylation de composés hétérocycliques. |
| DE3568455D1 (en) | 1984-05-23 | 1989-04-06 | Rhone Poulenc Chimie | Detergent compositions containing copolymers based on polyoxyethylene and polyoxyalkylene used as antisoil redeposition agents, and process for their preparation |
| GB8713768D0 (en) * | 1987-06-12 | 1987-07-15 | May & Baker Ltd | Compositions of matter |
| ATE208752T1 (de) * | 1996-08-01 | 2001-11-15 | Rhone Poulenc Chimie | Verfahren zum anbringen einer substituierten difluormethylgruppe |
| JPH11246555A (ja) * | 1997-10-31 | 1999-09-14 | Sumitomo Chem Co Ltd | フッ素置換ベンゾヘテロ環化合物 |
| DE69720082T2 (de) | 1997-12-22 | 2003-12-11 | Minnesota Mining & Mfg | Verfahren zur herstellung von fluorierten sulfinaten |
| DE19853560A1 (de) | 1998-11-20 | 2000-05-25 | Bayer Ag | Verfahren zur Herstellung von 5-Amino-3-(thio)carbamoylpyrazolen |
| PL206482B1 (pl) | 1999-10-22 | 2010-08-31 | Basf Agro B V Arnhem Nl | Sposób wytwarzania pochodnych 4-trifluorometylosulfinylopirazolu |
| JP2001220386A (ja) * | 1999-11-30 | 2001-08-14 | Takeda Chem Ind Ltd | オキサジアゾリン誘導体の製造方法 |
| JP2002020364A (ja) * | 2000-07-06 | 2002-01-23 | Konica Corp | スルフィン酸ナトリウム、スルフィン酸カリウムの製造方法およびそれらを用いた写真用カプラーの製造方法 |
| EP1331222A1 (en) | 2002-01-28 | 2003-07-30 | Virbac S.A. | Environment friendly reagents and process for halogenoalkylsulfinylation of organic compounds |
| CN1176078C (zh) | 2002-03-27 | 2004-11-17 | 江苏省农药研究所 | 带三氟甲基亚磺酰基的吡唑类化合物的亚磺酰化方法 |
| CA2667562A1 (en) | 2006-11-10 | 2008-05-15 | Basf Se | Process for the sulfinylation of a pyrazole derivative |
| AU2007316721B2 (en) | 2006-11-10 | 2013-05-09 | Basf Se | Process for the sulfinylation of a pyrazole derivative |
| FR2924115B1 (fr) | 2007-11-27 | 2010-02-26 | Rhodia Operations | Procede de preparation d'un acide trifluoromethanesulfinique |
| DK2349987T3 (da) * | 2008-10-02 | 2013-03-11 | Basf Se | Fremgangsmåde til fremstilling og oprensning af trifluormethansulfinsyre |
-
2007
- 2007-11-05 MX MX2009004262A patent/MX2009004262A/es active IP Right Grant
- 2007-11-05 NZ NZ576594A patent/NZ576594A/en not_active IP Right Cessation
- 2007-11-05 CA CA002667559A patent/CA2667559A1/en not_active Abandoned
- 2007-11-05 DK DK07822220.5T patent/DK2081908T3/da active
- 2007-11-05 EA EA200900629A patent/EA200900629A1/ru unknown
- 2007-11-05 PT PT78222205T patent/PT2081908E/pt unknown
- 2007-11-05 JP JP2009535702A patent/JP5450077B2/ja not_active Expired - Fee Related
- 2007-11-05 PL PL07822220T patent/PL2081908T3/pl unknown
- 2007-11-05 KR KR1020097011871A patent/KR20090083453A/ko not_active Application Discontinuation
- 2007-11-05 EP EP07822220.5A patent/EP2081908B1/en active Active
- 2007-11-05 ES ES07822220T patent/ES2422296T3/es active Active
- 2007-11-05 US US12/514,098 patent/US8263783B2/en active Active
- 2007-11-05 CN CN2012102449529A patent/CN102746233A/zh active Pending
- 2007-11-05 WO PCT/EP2007/061891 patent/WO2008055877A1/en active Application Filing
- 2007-11-05 BR BRPI0718774-2A patent/BRPI0718774A2/pt not_active Application Discontinuation
- 2007-11-05 AU AU2007316718A patent/AU2007316718B2/en active Active
- 2007-11-09 AR ARP070105012A patent/AR063646A1/es not_active Application Discontinuation
- 2007-11-09 TW TW096142570A patent/TWI413498B/zh not_active IP Right Cessation
-
2009
- 2009-04-21 IL IL198259A patent/IL198259A/en not_active IP Right Cessation
- 2009-05-25 MA MA31913A patent/MA30917B1/fr unknown
- 2009-06-08 ZA ZA2009/03968A patent/ZA200903968B/en unknown
-
2012
- 2012-08-14 US US13/585,233 patent/US20120309806A1/en not_active Abandoned
-
2013
- 2013-06-24 HR HRP20130582TT patent/HRP20130582T1/hr unknown
Also Published As
| Publication number | Publication date |
|---|---|
| JP2010509271A (ja) | 2010-03-25 |
| BRPI0718774A2 (pt) | 2013-12-03 |
| DK2081908T3 (da) | 2013-07-29 |
| CA2667559A1 (en) | 2008-05-15 |
| JP5450077B2 (ja) | 2014-03-26 |
| IL198259A0 (en) | 2009-12-24 |
| KR20090083453A (ko) | 2009-08-03 |
| HRP20130582T1 (en) | 2013-08-31 |
| MX2009004262A (es) | 2009-05-05 |
| AU2007316718A1 (en) | 2008-05-15 |
| PL2081908T3 (pl) | 2013-09-30 |
| MA30917B1 (fr) | 2009-11-02 |
| CN102746233A (zh) | 2012-10-24 |
| EP2081908B1 (en) | 2013-04-24 |
| US8263783B2 (en) | 2012-09-11 |
| NZ576594A (en) | 2011-12-22 |
| WO2008055877A1 (en) | 2008-05-15 |
| US20120309806A1 (en) | 2012-12-06 |
| IL198259A (en) | 2013-10-31 |
| EP2081908A1 (en) | 2009-07-29 |
| TW200829169A (en) | 2008-07-16 |
| ZA200903968B (en) | 2012-02-29 |
| PT2081908E (pt) | 2013-06-28 |
| EA200900629A1 (ru) | 2009-10-30 |
| US20100137395A1 (en) | 2010-06-03 |
| AU2007316718B2 (en) | 2013-03-28 |
| ES2422296T3 (es) | 2013-09-10 |
| TWI413498B (zh) | 2013-11-01 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |