AR056026A1 - Derivados de 2-oxo-benzotiazol, como agonistas del adrenoreceptor beta2, un procedimiento para su prepoaracion, composiciones farmaceuticas que los comprenden y su uso en la elaboracion de un medicamento para el tratamiento de enfermedades respiratorias - Google Patents

Derivados de 2-oxo-benzotiazol, como agonistas del adrenoreceptor beta2, un procedimiento para su prepoaracion, composiciones farmaceuticas que los comprenden y su uso en la elaboracion de un medicamento para el tratamiento de enfermedades respiratorias

Info

Publication number
AR056026A1
AR056026A1 ARP060103492A ARP060103492A AR056026A1 AR 056026 A1 AR056026 A1 AR 056026A1 AR P060103492 A ARP060103492 A AR P060103492A AR P060103492 A ARP060103492 A AR P060103492A AR 056026 A1 AR056026 A1 AR 056026A1
Authority
AR
Argentina
Prior art keywords
alkyl
formula
compound
represents hydrogen
hydrogen
Prior art date
Application number
ARP060103492A
Other languages
English (en)
Spanish (es)
Inventor
Alice Flaherty
Garry Pairaudeau
Michael Stocks
Roger V Bonnert
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37727572&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR056026(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of AR056026A1 publication Critical patent/AR056026A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62—Benzothiazoles
    • C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/428—Thiazoles condensed with carbocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Otolaryngology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
ARP060103492A 2005-08-09 2006-08-09 Derivados de 2-oxo-benzotiazol, como agonistas del adrenoreceptor beta2, un procedimiento para su prepoaracion, composiciones farmaceuticas que los comprenden y su uso en la elaboracion de un medicamento para el tratamiento de enfermedades respiratorias AR056026A1 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
SE0501793 2005-08-09
SE0501914 2005-08-30
SE0600515 2006-03-08

Publications (1)

Publication Number Publication Date
AR056026A1 true AR056026A1 (es) 2007-09-12

Family

ID=37727572

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP060103492A AR056026A1 (es) 2005-08-09 2006-08-09 Derivados de 2-oxo-benzotiazol, como agonistas del adrenoreceptor beta2, un procedimiento para su prepoaracion, composiciones farmaceuticas que los comprenden y su uso en la elaboracion de un medicamento para el tratamiento de enfermedades respiratorias

Country Status (17)

Country Link
US (2) US7709511B2 (enExample)
EP (1) EP1915354A4 (enExample)
JP (1) JP4522474B2 (enExample)
KR (1) KR20080033372A (enExample)
AR (1) AR056026A1 (enExample)
AU (2) AU2006277074B2 (enExample)
BR (1) BRPI0614542A2 (enExample)
CA (1) CA2618511C (enExample)
EC (1) ECSP088246A (enExample)
IL (1) IL188857A0 (enExample)
MX (1) MX2008001664A (enExample)
MY (1) MY145647A (enExample)
NO (1) NO20081217L (enExample)
NZ (1) NZ565472A (enExample)
TW (1) TW200738658A (enExample)
UY (1) UY29732A1 (enExample)
WO (1) WO2007018461A1 (enExample)

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TW200745067A (en) * 2006-03-14 2007-12-16 Astrazeneca Ab Novel compounds
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GB0702456D0 (en) * 2007-02-08 2007-03-21 Astrazeneca Ab New combination
GB0702458D0 (en) * 2007-02-08 2007-03-21 Astrazeneca Ab Salts 668
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GB0702457D0 (en) * 2007-02-08 2007-03-21 Astrazeneca Ab New combination 666
WO2009037503A2 (en) * 2007-09-18 2009-03-26 Astrazeneca Ab New combination - 012 for the treatment of respiratory diseases
RU2010147881A (ru) * 2008-05-13 2012-06-20 Астразенека Аб (Se) ФАРМАЦЕВТИЧЕСКИЙ ПРОДУКТ, СОДЕРЖАЩИЙ АНТАГОНИСТ МУСКАРИНОВОГО РЕЦЕПТОРА И АГОНИСТ β2-АДРЕНОРЕЦЕПТОРА
US8329729B2 (en) 2008-05-13 2012-12-11 Astrazeneca Ab Quinuclidine derivatives as muscarinic M3 receptor antagonists
WO2009142568A1 (en) * 2008-05-20 2009-11-26 Astrazeneca Ab Combination of (a) glucocorticoid receptor modulator and (b) a b2-agonist
GB0811100D0 (en) * 2008-06-17 2008-07-23 Astrazeneca Ab New combination
WO2009154557A1 (en) 2008-06-18 2009-12-23 Astrazeneca Ab Benzoxazinone derivatives acting as beta2-adrenoreceptor agonist for the treatment of respiratory disorders
EP2303266A4 (en) * 2008-06-20 2015-01-21 Astrazeneca Ab PHARMACEUTICAL COMPOSITION COMPRISING A 4-HYDROXY-2-OXO-2,3-DIHYDRO-1,3-BENZOTHIAZOL-7-YLE COMPOUND FOR THE MODULATION OF BETA-2-ADRENORECEPTOR ACTIVITY
GB0814728D0 (en) * 2008-08-12 2008-09-17 Argenta Discovery Ltd New combination
GB0913342D0 (en) 2009-07-31 2009-09-16 Astrazeneca Ab Compounds - 801
WO2011061527A1 (en) 2009-11-17 2011-05-26 Astrazeneca Ab Combinations comprising a glucocorticoid receptor modulator for the treatment of respiratory diseases
CN103619816B (zh) 2011-04-18 2016-05-18 联邦科学与工业研究组织 气体捕集方法

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Also Published As

Publication number Publication date
WO2007018461A1 (en) 2007-02-15
US20100210688A1 (en) 2010-08-19
KR20080033372A (ko) 2008-04-16
CA2618511A1 (en) 2007-02-15
ECSP088246A (es) 2008-05-30
CA2618511C (en) 2011-03-15
EP1915354A4 (en) 2010-07-14
AU2010202319B2 (en) 2011-09-22
MX2008001664A (es) 2008-02-19
IL188857A0 (en) 2008-04-13
NO20081217L (no) 2008-04-15
TW200738658A (en) 2007-10-16
JP2009504639A (ja) 2009-02-05
JP4522474B2 (ja) 2010-08-11
AU2006277074A1 (en) 2007-02-15
AU2006277074B2 (en) 2010-03-04
EP1915354A1 (en) 2008-04-30
UY29732A1 (es) 2007-03-30
NZ565472A (en) 2011-03-31
US20080300275A1 (en) 2008-12-04
BRPI0614542A2 (pt) 2012-11-27
AU2010202319A1 (en) 2010-07-01
MY145647A (en) 2012-03-15
US7709511B2 (en) 2010-05-04

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