AR049028A1 - Sal solida farmaceuticamente adecuada y que no sublima del enantiomero s de mirtazapina y metodo de fabricacion - Google Patents

Sal solida farmaceuticamente adecuada y que no sublima del enantiomero s de mirtazapina y metodo de fabricacion

Info

Publication number
AR049028A1
AR049028A1 ARP050101549A ARP050101549A AR049028A1 AR 049028 A1 AR049028 A1 AR 049028A1 AR P050101549 A ARP050101549 A AR P050101549A AR P050101549 A ARP050101549 A AR P050101549A AR 049028 A1 AR049028 A1 AR 049028A1
Authority
AR
Argentina
Prior art keywords
mirtazapine
enantiomer
manufacturing
sublimate
solid salt
Prior art date
Application number
ARP050101549A
Other languages
English (en)
Spanish (es)
Inventor
Sytske Hyke Moolenaar
Der Voort Maarschalk Kees Van
Gerardus Johannes Kemperman
Original Assignee
Akzo Nobel Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Akzo Nobel Nv filed Critical Akzo Nobel Nv
Publication of AR049028A1 publication Critical patent/AR049028A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
ARP050101549A 2004-04-21 2005-04-20 Sal solida farmaceuticamente adecuada y que no sublima del enantiomero s de mirtazapina y metodo de fabricacion AR049028A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP04101664 2004-04-21

Publications (1)

Publication Number Publication Date
AR049028A1 true AR049028A1 (es) 2006-06-21

Family

ID=34928990

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP050101549A AR049028A1 (es) 2004-04-21 2005-04-20 Sal solida farmaceuticamente adecuada y que no sublima del enantiomero s de mirtazapina y metodo de fabricacion

Country Status (31)

Country Link
US (1) US20070111993A1 (https=)
EP (1) EP1729777B1 (https=)
JP (2) JP5260959B2 (https=)
CN (2) CN1942191B (https=)
AR (1) AR049028A1 (https=)
AT (1) ATE424210T1 (https=)
AU (1) AU2005235383B2 (https=)
BR (1) BRPI0509953A (https=)
CA (1) CA2561281C (https=)
CY (1) CY1109018T1 (https=)
DE (1) DE602005013066D1 (https=)
DK (1) DK1729777T3 (https=)
EC (1) ECSP066938A (https=)
ES (1) ES2321961T3 (https=)
HR (1) HRP20090190T1 (https=)
IL (1) IL178201A (https=)
LV (1) LV13556B (https=)
MX (1) MXPA06011830A (https=)
MY (1) MY144899A (https=)
NO (1) NO20065077L (https=)
NZ (1) NZ550052A (https=)
PE (1) PE20060400A1 (https=)
PL (1) PL1729777T3 (https=)
PT (1) PT1729777E (https=)
RS (1) RS50764B (https=)
RU (1) RU2375362C2 (https=)
SI (1) SI1729777T1 (https=)
TW (1) TW200538100A (https=)
UA (1) UA89773C2 (https=)
WO (1) WO2005102352A1 (https=)
ZA (1) ZA200608305B (https=)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA83666C2 (ru) * 2003-07-10 2008-08-11 Н.В. Органон Способ получения энантиомерно чистого миртазапина
EP1792618A1 (en) * 2005-11-30 2007-06-06 Rainer Freynhagen R-mirtazapine for the treatment of pain
TW200808804A (en) * 2006-05-22 2008-02-16 Organon Nv Mirtazapine for the treatment of neuropathic pain
CN104095824B (zh) * 2013-04-09 2016-08-31 上海信谊万象药业股份有限公司 一种米氮平缓释片及其制备方法
PL3261645T3 (pl) 2015-02-27 2021-12-06 Dechra Limited Pobudzanie apetytu, zarządzanie utratą masy ciała, i leczenie anoreksji u psów i kotów
CN111053735A (zh) * 2020-02-25 2020-04-24 上海阶平医院管理有限公司 一种治疗失眠的冷敷凝胶

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL189199C (nl) * 1975-04-05 1993-02-01 Akzo Nv Werkwijze ter bereiding van farmaceutische preparaten met werking op het centraal zenuwstelsel op basis van benz(aryl)azepinederivaten, de verkregen gevormde farmaceutische preparaten, alsmede werkwijze ter bereiding van de toe te passen benz(aryl)azepinederivaten.
US4193828A (en) * 1976-07-27 1980-03-18 Fiber Materials, Inc. Method of forming carbon composites
US4515792A (en) * 1982-09-30 1985-05-07 Ciba-Geigy Corporation Tetracyclic heterocycles and antidepressant compositions thereof
EP0813873B1 (en) * 1996-06-19 2002-02-13 Akzo Nobel N.V. Pharmaceutical composition comprising mirtazapine and one or more selective serotonin reuptake inhibitors
IL121076A (en) * 1996-06-19 2000-10-31 Akzo Nobel Nv Pharmaceutical combinations comprising mirtazapine and one or more selective serotonin reuptake inhibitors
WO1999051237A1 (en) * 1998-04-02 1999-10-14 Akzo Nobel N.V. Oral liquid antidepressant solution
WO2001000196A2 (en) * 1999-06-25 2001-01-04 University Of South Florida Mirtazapine for weight gain in wasting diseases
US6281207B1 (en) * 1999-09-15 2001-08-28 Reed Richter Treatment of movement disorders by administration of mirtazapine
WO2001042239A1 (en) * 1999-12-13 2001-06-14 Sumika Fine Chemicals Co., Ltd. Process for the preparation of a pyridinemethanol compound
SK14162002A3 (sk) * 2000-04-05 2003-03-04 Akzo Nobel N.V. Kombinácia obsahujúca paracetamol alebo nesteroidné protizápalové liečivo, použitie mirtazapínu, paracetamolu a pacientský balíček

Also Published As

Publication number Publication date
EP1729777B1 (en) 2009-03-04
CN1942191A (zh) 2007-04-04
EP1729777A1 (en) 2006-12-13
PL1729777T3 (pl) 2009-07-31
TW200538100A (en) 2005-12-01
CA2561281C (en) 2013-04-02
ZA200608305B (en) 2008-08-27
BRPI0509953A (pt) 2007-09-25
CN1942191B (zh) 2011-02-02
US20070111993A1 (en) 2007-05-17
AU2005235383A1 (en) 2005-11-03
NO20065077L (no) 2006-11-14
CN101824035A (zh) 2010-09-08
SI1729777T1 (sl) 2009-08-31
CA2561281A1 (en) 2005-11-03
CY1109018T1 (el) 2014-07-02
IL178201A (en) 2010-06-30
PE20060400A1 (es) 2006-05-27
WO2005102352A1 (en) 2005-11-03
UA89773C2 (ru) 2010-03-10
IL178201A0 (en) 2006-12-31
LV13556B (en) 2007-07-20
RS50764B (sr) 2010-08-31
MY144899A (en) 2011-11-30
ECSP066938A (es) 2006-12-20
JP5260959B2 (ja) 2013-08-14
JP2007533705A (ja) 2007-11-22
HRP20090190T1 (en) 2009-05-31
DK1729777T3 (da) 2009-06-08
NZ550052A (en) 2010-02-26
ATE424210T1 (de) 2009-03-15
MXPA06011830A (es) 2007-03-23
ES2321961T3 (es) 2009-06-15
AU2005235383B2 (en) 2010-05-27
RU2006140988A (ru) 2008-05-27
JP2013136626A (ja) 2013-07-11
DE602005013066D1 (de) 2009-04-16
RU2375362C2 (ru) 2009-12-10
PT1729777E (pt) 2009-04-27

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