AR028991A1 - METODO PARA PREPARAR UN ANALOGO DE beta- NUCLEOSIDO. - Google Patents

METODO PARA PREPARAR UN ANALOGO DE beta- NUCLEOSIDO.

Info

Publication number
AR028991A1
AR028991A1 ARP000102222A ARP000102222A AR028991A1 AR 028991 A1 AR028991 A1 AR 028991A1 AR P000102222 A ARP000102222 A AR P000102222A AR P000102222 A ARP000102222 A AR P000102222A AR 028991 A1 AR028991 A1 AR 028991A1
Authority
AR
Argentina
Prior art keywords
group
hydrogen
beta
substituted
alkyl
Prior art date
Application number
ARP000102222A
Other languages
English (en)
Spanish (es)
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of AR028991A1 publication Critical patent/AR028991A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H21/00Compounds containing two or more mononucleotide units having separate phosphate or polyphosphate groups linked by saccharide radicals of nucleoside groups, e.g. nucleic acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/14Pyrrolo-pyrimidine radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Genetics & Genomics (AREA)
  • General Health & Medical Sciences (AREA)
  • Biotechnology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
ARP000102222A 1999-05-11 2000-05-09 METODO PARA PREPARAR UN ANALOGO DE beta- NUCLEOSIDO. AR028991A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US13365199P 1999-05-11 1999-05-11

Publications (1)

Publication Number Publication Date
AR028991A1 true AR028991A1 (es) 2003-06-04

Family

ID=22459680

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP000102222A AR028991A1 (es) 1999-05-11 2000-05-09 METODO PARA PREPARAR UN ANALOGO DE beta- NUCLEOSIDO.

Country Status (22)

Country Link
US (1) US6271370B1 (OSRAM)
EP (1) EP1052264B1 (OSRAM)
JP (1) JP2001011092A (OSRAM)
KR (1) KR100403900B1 (OSRAM)
CN (1) CN1275575A (OSRAM)
AR (1) AR028991A1 (OSRAM)
AT (1) ATE291582T1 (OSRAM)
AU (1) AU3401100A (OSRAM)
BR (1) BR0002089A (OSRAM)
CA (1) CA2307951A1 (OSRAM)
CZ (1) CZ20001710A3 (OSRAM)
DE (1) DE60018833D1 (OSRAM)
HU (1) HUP0001843A3 (OSRAM)
ID (1) ID25992A (OSRAM)
IL (1) IL136027A0 (OSRAM)
IN (1) IN186850B (OSRAM)
MX (1) MXPA00004532A (OSRAM)
PL (1) PL340109A1 (OSRAM)
RU (1) RU2200738C2 (OSRAM)
TR (1) TR200001340A2 (OSRAM)
YU (1) YU25500A (OSRAM)
ZA (1) ZA200002263B (OSRAM)

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EP2673277A1 (en) 2011-02-10 2013-12-18 Novartis AG [1, 2, 4]triazolo [4, 3 -b]pyridazine compounds as inhibitors of the c-met tyrosine kinase
JP5808826B2 (ja) 2011-02-23 2015-11-10 インテリカイン, エルエルシー 複素環化合物およびその使用
CA2828219A1 (en) 2011-02-25 2012-08-30 Irm Llc Pyrazolo [1,5-a] pyridines as trk inhibitors
US9062045B2 (en) 2011-09-15 2015-06-23 Novartis Ag Triazolopyridine compounds
US20130209543A1 (en) 2011-11-23 2013-08-15 Intellikine Llc Enhanced treatment regimens using mtor inhibitors
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WO2014151147A1 (en) 2013-03-15 2014-09-25 Intellikine, Llc Combination of kinase inhibitors and uses thereof
AR096532A1 (es) 2013-06-06 2016-01-13 Chiesi Farm Spa Inhibidores de quinasa
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JP6487921B2 (ja) 2013-12-17 2019-03-20 ファイザー・インク LRRK2阻害薬としての新規の3,4−二置換−1H−ピロロ[2,3−b]ピリジンおよび4,5−二置換−7H−ピロロ[2,3−c]ピリダジン
WO2016011658A1 (en) 2014-07-25 2016-01-28 Novartis Ag Combination therapy
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EP3630767A1 (en) 2017-05-22 2020-04-08 H. Hoffnabb-La Roche Ag Therapeutic compounds and compositions, and methods of use thereof
KR20200010390A (ko) 2017-05-22 2020-01-30 에프. 호프만-라 로슈 아게 치료 화합물 및 조성물, 및 이의 사용 방법
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JP7339263B2 (ja) 2018-01-15 2023-09-05 エフ. ホフマン-ラ ロシュ アーゲー Jak阻害剤としてのピラゾロピリミジン化合物
CA3102279A1 (en) 2018-06-01 2019-12-05 Cornell University Combination therapy for pi3k-associated disease or disorder
JP7657740B2 (ja) 2019-06-18 2025-04-07 エフ・ホフマン-ラ・ロシュ・アクチェンゲゼルシャフト Jakキナーゼのピラゾロピリミジンスルホン阻害剤およびその使用
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Also Published As

Publication number Publication date
KR100403900B1 (ko) 2003-11-01
KR20010069193A (ko) 2001-07-23
US6271370B1 (en) 2001-08-07
EP1052264A2 (en) 2000-11-15
EP1052264A3 (en) 2001-06-13
IL136027A0 (en) 2001-05-20
JP2001011092A (ja) 2001-01-16
ATE291582T1 (de) 2005-04-15
HUP0001843A3 (en) 2001-09-28
HU0001843D0 (en) 2000-07-28
EP1052264B1 (en) 2005-03-23
BR0002089A (pt) 2001-01-02
TR200001340A2 (tr) 2000-12-21
IN186850B (OSRAM) 2001-11-24
RU2200738C2 (ru) 2003-03-20
CN1275575A (zh) 2000-12-06
ZA200002263B (en) 2001-12-24
YU25500A (sh) 2003-08-29
HUP0001843A2 (hu) 2001-06-28
CZ20001710A3 (cs) 2001-09-12
DE60018833D1 (de) 2005-04-28
PL340109A1 (en) 2000-11-20
CA2307951A1 (en) 2000-11-11
MXPA00004532A (es) 2002-03-08
AU3401100A (en) 2000-11-16
ID25992A (id) 2000-11-16

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