AP2774A - Substituted (pyrazolylcarbonyl) imidazolidinones and their uses - Google Patents

Substituted (pyrazolylcarbonyl) imidazolidinones and their uses

Info

Publication number
AP2774A
AP2774A AP2010005422A AP2010005422A AP2774A AP 2774 A AP2774 A AP 2774A AP 2010005422 A AP2010005422 A AP 2010005422A AP 2010005422 A AP2010005422 A AP 2010005422A AP 2774 A AP2774 A AP 2774A
Authority
AP
ARIPO
Prior art keywords
pyrazolylcarbonyl
imidazolidinones
substituted
Prior art date
Application number
AP2010005422A
Other languages
English (en)
Other versions
AP2010005422A0 (en
Inventor
Kai Thede
Susanne Greschat
Steffen Wildum
Original Assignee
Aicuris Gmbh & Co Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aicuris Gmbh & Co Kg filed Critical Aicuris Gmbh & Co Kg
Publication of AP2010005422A0 publication Critical patent/AP2010005422A0/en
Application granted granted Critical
Publication of AP2774A publication Critical patent/AP2774A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Molecular Biology (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AP2010005422A 2008-03-17 2009-03-10 Substituted (pyrazolylcarbonyl) imidazolidinones and their uses AP2774A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102008015033A DE102008015033A1 (de) 2008-03-17 2008-03-17 Substituierte (Pyrazolyl-carbonyl)imidazolidinone und ihre Verwendung
PCT/EP2009/001714 WO2009115213A1 (de) 2008-03-17 2009-03-10 (pyrazolyl-carbonyl) imidazolidinone-derivate zur behandlung retroviraler erkrankungen

Publications (2)

Publication Number Publication Date
AP2010005422A0 AP2010005422A0 (en) 2010-10-31
AP2774A true AP2774A (en) 2013-09-30

Family

ID=40565083

Family Applications (1)

Application Number Title Priority Date Filing Date
AP2010005422A AP2774A (en) 2008-03-17 2009-03-10 Substituted (pyrazolylcarbonyl) imidazolidinones and their uses

Country Status (22)

Country Link
US (1) US8399682B2 (es)
EP (1) EP2254885B1 (es)
JP (1) JP5576853B2 (es)
KR (1) KR20100124337A (es)
CN (1) CN101977908B (es)
AP (1) AP2774A (es)
AR (1) AR070919A1 (es)
AU (1) AU2009226656A1 (es)
CA (1) CA2718685C (es)
CL (1) CL2009000636A1 (es)
DE (1) DE102008015033A1 (es)
IL (1) IL207649A0 (es)
MA (1) MA32224B1 (es)
MX (1) MX2010010230A (es)
NZ (1) NZ588141A (es)
PE (1) PE20091718A1 (es)
RU (1) RU2010141578A (es)
TW (1) TW200951125A (es)
UA (1) UA102390C2 (es)
UY (1) UY31717A1 (es)
WO (1) WO2009115213A1 (es)
ZA (1) ZA201007361B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102008015032A1 (de) * 2008-03-17 2009-09-24 Aicuris Gmbh & Co. Kg Substituierte Pyrazolamide und ihre Verwendung
DE102008015033A1 (de) 2008-03-17 2009-09-24 Aicuris Gmbh & Co. Kg Substituierte (Pyrazolyl-carbonyl)imidazolidinone und ihre Verwendung
DE102008062878A1 (de) 2008-12-17 2010-06-24 Aicuris Gmbh & Co. Kg Substituierte Furancarboxamide und ihre Verwendung
DE102008062863A1 (de) 2008-12-17 2010-06-24 Aicuris Gmbh & Co. Kg Substituierte (Thiophenyl-carbonyl)imidazolidinone und ihre Verwendung
EP2295038B1 (en) * 2009-09-11 2013-05-29 AiCuris GmbH & Co. KG Solid dispersion comprising an anti-HIV agent
DE102011055815A1 (de) 2011-11-29 2013-05-29 Aicuris Gmbh & Co. Kg Carboxamid-substituierte Heteroaryl-Pyrazole und ihre Verwendung
DE102012016908A1 (de) 2012-08-17 2014-02-20 Aicuris Gmbh & Co. Kg Tris-(Hetero)Aryl-Pyrazole und ihre Verwendung

Citations (4)

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WO2002100853A1 (en) * 2001-06-04 2002-12-19 F. Hoffmann-La Roche Ag Pyrazole derivatives as hiv reverse transcriptase inhibitors
WO2004024147A1 (en) * 2002-09-16 2004-03-25 Pfizer Limited 4-(3,5-dicyanophenoxy) pyrazole derivatives for use as transcriptase modulators in the treatment of i.a. hiv
WO2004031178A1 (en) * 2002-10-07 2004-04-15 Pfizer Limited Pyrazole derivatives
US20050054707A1 (en) * 2003-09-05 2005-03-10 Pfizer Inc. Pyrazole derivatives

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DE3119796A1 (de) 1981-05-19 1982-12-23 Hoechst Ag, 6000 Frankfurt Substituierte tryptaminderivate von thienyloxpropanolaminen, verfahren zu ihrer herstellung, pharmazeutische praeparate auf basis dieser verbindungen sowie ihre verwendung
FR2538388B1 (fr) 1982-12-24 1985-06-21 Pharmuka Lab Nouveaux derives de naphtalene- ou azanaphtalenecarboxamide, leurs procedes de preparation et leur utilisation comme medicaments
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EE200200715A (et) 2000-06-28 2004-08-16 Astrazeneca Ab Asendatud kinasoliini derivaadid ja nende kasutamine inhibiitoritena
DE60208683T2 (de) 2001-08-01 2006-11-02 Basell Polyolefine Gmbh Verfahren zur herstellung von heterocyclischen pentalen derivaten
EP1451160B1 (en) 2001-11-01 2010-01-13 Icagen, Inc. Pyrazole-amides for use in the treatment of pain
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Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002100853A1 (en) * 2001-06-04 2002-12-19 F. Hoffmann-La Roche Ag Pyrazole derivatives as hiv reverse transcriptase inhibitors
WO2004024147A1 (en) * 2002-09-16 2004-03-25 Pfizer Limited 4-(3,5-dicyanophenoxy) pyrazole derivatives for use as transcriptase modulators in the treatment of i.a. hiv
WO2004031178A1 (en) * 2002-10-07 2004-04-15 Pfizer Limited Pyrazole derivatives
US20050054707A1 (en) * 2003-09-05 2005-03-10 Pfizer Inc. Pyrazole derivatives

Also Published As

Publication number Publication date
CL2009000636A1 (es) 2010-05-07
JP5576853B2 (ja) 2014-08-20
JP2011514366A (ja) 2011-05-06
IL207649A0 (en) 2010-12-30
US20110124618A1 (en) 2011-05-26
AR070919A1 (es) 2010-05-12
PE20091718A1 (es) 2009-12-11
AP2010005422A0 (en) 2010-10-31
NZ588141A (en) 2012-05-25
CN101977908B (zh) 2014-04-23
WO2009115213A1 (de) 2009-09-24
TW200951125A (en) 2009-12-16
US8399682B2 (en) 2013-03-19
EP2254885A1 (de) 2010-12-01
ZA201007361B (en) 2011-12-28
DE102008015033A1 (de) 2009-09-24
EP2254885B1 (de) 2013-12-04
UA102390C2 (ru) 2013-07-10
MA32224B1 (fr) 2011-04-01
AU2009226656A1 (en) 2009-09-24
UY31717A1 (es) 2009-08-31
CA2718685C (en) 2016-11-29
KR20100124337A (ko) 2010-11-26
CN101977908A (zh) 2011-02-16
MX2010010230A (es) 2010-11-09
CA2718685A1 (en) 2009-09-24
RU2010141578A (ru) 2012-04-27

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