ZA945340B - 4-Aryloxy-and 4-arylthiopiperidine derivatives - Google Patents

4-Aryloxy-and 4-arylthiopiperidine derivatives

Info

Publication number
ZA945340B
ZA945340B ZA945340A ZA945340A ZA945340B ZA 945340 B ZA945340 B ZA 945340B ZA 945340 A ZA945340 A ZA 945340A ZA 945340 A ZA945340 A ZA 945340A ZA 945340 B ZA945340 B ZA 945340B
Authority
ZA
South Africa
Prior art keywords
atoms
aryloxy
action
hal
arylthiopiperidine
Prior art date
Application number
ZA945340A
Other languages
English (en)
Inventor
Helmut Pruecher
Rudolf Gottschlich
Gerd Bartoszyk
Christoph Seyfried
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of ZA945340B publication Critical patent/ZA945340B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)
ZA945340A 1993-07-21 1994-07-20 4-Aryloxy-and 4-arylthiopiperidine derivatives ZA945340B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4324393A DE4324393A1 (de) 1993-07-21 1993-07-21 4-Aryloxy- und 4-Arylthiopiperidinderivate

Publications (1)

Publication Number Publication Date
ZA945340B true ZA945340B (en) 1995-03-01

Family

ID=6493312

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA945340A ZA945340B (en) 1993-07-21 1994-07-20 4-Aryloxy-and 4-arylthiopiperidine derivatives

Country Status (21)

Country Link
US (1) US5561145A (xx)
EP (1) EP0635505B1 (xx)
JP (1) JPH0770117A (xx)
KR (1) KR100354303B1 (xx)
CN (1) CN1055690C (xx)
AT (1) ATE159252T1 (xx)
AU (1) AU683886B2 (xx)
CA (1) CA2128380C (xx)
CZ (1) CZ284544B6 (xx)
DE (2) DE4324393A1 (xx)
DK (1) DK0635505T3 (xx)
ES (1) ES2110660T3 (xx)
GR (1) GR3025880T3 (xx)
HU (1) HU218912B (xx)
NO (1) NO301477B1 (xx)
PL (1) PL177692B1 (xx)
RU (1) RU2135495C1 (xx)
SK (1) SK281630B6 (xx)
TW (1) TW401417B (xx)
UA (1) UA43828C2 (xx)
ZA (1) ZA945340B (xx)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2134870T3 (es) * 1993-05-01 1999-10-16 Merck Patent Gmbh Antagonistas del receptor de adhesion.
DE4332384A1 (de) * 1993-09-23 1995-03-30 Merck Patent Gmbh Adhäsionsrezeptor-Antagonisten III
DK0710657T3 (da) * 1994-11-02 1999-05-25 Merck Patent Gmbh Adhæsionsreceptor-antagonister
DE19504954A1 (de) * 1995-02-15 1996-08-22 Merck Patent Gmbh Adhäsionsrezeptor-Antagonisten
DE19524765A1 (de) * 1995-07-07 1997-01-09 Boehringer Mannheim Gmbh Neue Oxazolidinonderivate, Verfahren zu deren Herstellung und diese Verbindungen enthaltende Arzneimittel
DE19531321A1 (de) * 1995-08-25 1997-02-27 Merck Patent Gmbh Piperidinylmethyloxazolidinone
US5977138A (en) * 1996-08-15 1999-11-02 Schering Corporation Ether muscarinic antagonists
DE19707628A1 (de) * 1997-02-26 1998-08-27 Merck Patent Gmbh Oxazolidinone
EP1467986A1 (en) 2002-01-17 2004-10-20 Eli Lilly And Company Aza-cyclic compounds as modulators of acetylcholine receptors
EP1963261A1 (en) * 2005-12-21 2008-09-03 Decode Genetics EHF Biaryl substituted nitrogen containing heterocycle inhibitors of lta4h for treating inflammation
DE102014010989B4 (de) 2014-07-29 2017-06-14 Kautex Textron Gmbh & Co. Kg Einfüllstutzen für einen Flüssigkeitsbehälter, insbesondere für einen Harnstoffbehälter
WO2018026371A1 (en) * 2016-08-04 2018-02-08 Sunovion Pharmaceuticals Inc. Dual nav1.2/5ht2a inhibitors for treating cns disorders

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0713017B2 (ja) * 1986-06-18 1995-02-15 日本ケミファ株式会社 脳細胞保護作用を有する医薬組成物
DE3723797A1 (de) * 1987-07-18 1989-01-26 Merck Patent Gmbh Oxazolidinone
DE4005371A1 (de) * 1990-02-21 1991-08-22 Merck Patent Gmbh Oxazolidinone
DE4017211A1 (de) * 1990-05-29 1991-12-05 Merck Patent Gmbh Oxazolidinone

Also Published As

Publication number Publication date
SK85294A3 (en) 1995-03-08
TW401417B (en) 2000-08-11
CZ284544B6 (cs) 1998-12-16
CA2128380A1 (en) 1995-01-22
NO942715L (no) 1995-01-23
CN1055690C (zh) 2000-08-23
RU2135495C1 (ru) 1999-08-27
KR100354303B1 (ko) 2002-12-11
AU6753694A (en) 1995-02-02
CA2128380C (en) 2005-04-12
CN1106008A (zh) 1995-08-02
EP0635505A1 (de) 1995-01-25
ATE159252T1 (de) 1997-11-15
HU218912B (hu) 2000-12-28
JPH0770117A (ja) 1995-03-14
EP0635505B1 (de) 1997-10-15
UA43828C2 (uk) 2002-01-15
CZ173894A3 (en) 1995-05-17
AU683886B2 (en) 1997-11-27
GR3025880T3 (en) 1998-04-30
DE59404319D1 (de) 1997-11-20
NO301477B1 (no) 1997-11-03
HU9402154D0 (en) 1994-09-28
RU94026079A (ru) 1996-05-27
US5561145A (en) 1996-10-01
DK0635505T3 (da) 1998-06-02
PL304349A1 (en) 1995-01-23
HUT71110A (en) 1995-11-28
ES2110660T3 (es) 1998-02-16
NO942715D0 (no) 1994-07-20
PL177692B1 (pl) 2000-01-31
SK281630B6 (sk) 2001-06-11
DE4324393A1 (de) 1995-01-26
KR950003290A (ko) 1995-02-16

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