ZA918044B - Pyridine and pyridine n-oxide derivatives of diaryl methyl piperidines of piperazines,and compositions and methods of use thereof - Google Patents

Pyridine and pyridine n-oxide derivatives of diaryl methyl piperidines of piperazines,and compositions and methods of use thereof

Info

Publication number
ZA918044B
ZA918044B ZA918044A ZA918044A ZA918044B ZA 918044 B ZA918044 B ZA 918044B ZA 918044 A ZA918044 A ZA 918044A ZA 918044 A ZA918044 A ZA 918044A ZA 918044 B ZA918044 B ZA 918044B
Authority
ZA
South Africa
Prior art keywords
pyridine
piperazines
methods
pct
oxide derivatives
Prior art date
Application number
ZA918044A
Other languages
English (en)
Inventor
John J Piwinski
J Piwinski John
Jesse Wong
Wong Jesse
Michael J Green
J Green Michael
Vera Seidl
Seidl Vera
Richard Friary
Friary Richard
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corp filed Critical Schering Corp
Publication of ZA918044B publication Critical patent/ZA918044B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
ZA918044A 1990-10-10 1991-10-08 Pyridine and pyridine n-oxide derivatives of diaryl methyl piperidines of piperazines,and compositions and methods of use thereof ZA918044B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US59533090A 1990-10-10 1990-10-10

Publications (1)

Publication Number Publication Date
ZA918044B true ZA918044B (en) 1992-07-29

Family

ID=24382813

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA918044A ZA918044B (en) 1990-10-10 1991-10-08 Pyridine and pyridine n-oxide derivatives of diaryl methyl piperidines of piperazines,and compositions and methods of use thereof

Country Status (22)

Country Link
US (1) US5432175A (cs)
EP (1) EP0553191B1 (cs)
JP (1) JPH089596B2 (cs)
KR (1) KR970005927B1 (cs)
AT (1) ATE122673T1 (cs)
AU (1) AU646519B2 (cs)
CA (1) CA2093798C (cs)
CZ (1) CZ280532B6 (cs)
DE (1) DE69109871T2 (cs)
DK (1) DK0553191T3 (cs)
ES (1) ES2072627T3 (cs)
FI (1) FI931600L (cs)
HK (1) HK186596A (cs)
HU (1) HUT66081A (cs)
IE (1) IE67808B1 (cs)
IL (1) IL99676A (cs)
MY (1) MY108616A (cs)
NO (1) NO305028B1 (cs)
PH (1) PH31566A (cs)
SK (1) SK31793A3 (cs)
WO (1) WO1992006971A1 (cs)
ZA (1) ZA918044B (cs)

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Also Published As

Publication number Publication date
AU8849091A (en) 1992-05-20
JPH089596B2 (ja) 1996-01-31
EP0553191A1 (en) 1993-08-04
FI931600A0 (fi) 1993-04-08
NO931312D0 (no) 1993-04-06
HK186596A (en) 1996-10-11
FI931600A7 (fi) 1993-05-17
KR970005927B1 (ko) 1997-04-22
EP0553191B1 (en) 1995-05-17
MY108616A (en) 1996-10-31
AU646519B2 (en) 1994-02-24
IL99676A0 (en) 1992-08-18
HUT66081A (en) 1994-09-28
NO305028B1 (no) 1999-03-22
CA2093798A1 (en) 1992-04-11
IE913571A1 (en) 1992-04-22
US5432175A (en) 1995-07-11
CZ280532B6 (cs) 1996-02-14
FI931600L (fi) 1993-05-17
SK31793A3 (en) 1993-09-08
IE67808B1 (en) 1996-05-01
ATE122673T1 (de) 1995-06-15
ES2072627T3 (es) 1995-07-16
CZ62293A3 (en) 1994-02-16
PH31566A (en) 1998-11-03
IL99676A (en) 1995-11-27
HU9301051D0 (en) 1993-07-28
DK0553191T3 (da) 1995-08-07
NO931312L (no) 1993-06-10
DE69109871T2 (de) 1995-09-14
CA2093798C (en) 2000-02-01
JPH05508660A (ja) 1993-12-02
DE69109871D1 (de) 1995-06-22
WO1992006971A1 (en) 1992-04-30

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