ZA913092B - Process for the synthesis of n-(3-(1h-imidazol-1-yl)phenyl-4-(substituted)-2-pyrimidinamines - Google Patents
Process for the synthesis of n-(3-(1h-imidazol-1-yl)phenyl-4-(substituted)-2-pyrimidinaminesInfo
- Publication number
- ZA913092B ZA913092B ZA913092A ZA913092A ZA913092B ZA 913092 B ZA913092 B ZA 913092B ZA 913092 A ZA913092 A ZA 913092A ZA 913092 A ZA913092 A ZA 913092A ZA 913092 B ZA913092 B ZA 913092B
- Authority
- ZA
- South Africa
- Prior art keywords
- imidazol
- substituted
- phenyl
- dihydrohalide
- pyridinyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Photoreceptors In Electrophotography (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US07/514,455 US5064963A (en) | 1990-04-25 | 1990-04-25 | Process for the synthesis of n-(3-(1h-imidazol-1-yl)phenyl-4-(substituted)-2-pyrimidinamines |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA913092B true ZA913092B (en) | 1992-02-26 |
Family
ID=24047219
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA913092A ZA913092B (en) | 1990-04-25 | 1991-04-24 | Process for the synthesis of n-(3-(1h-imidazol-1-yl)phenyl-4-(substituted)-2-pyrimidinamines |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US5064963A (hu) |
| EP (1) | EP0453731B1 (hu) |
| JP (1) | JPH04225975A (hu) |
| KR (1) | KR0168679B1 (hu) |
| AT (1) | ATE170184T1 (hu) |
| AU (1) | AU630849B2 (hu) |
| CA (1) | CA2041031A1 (hu) |
| DE (1) | DE69130029T2 (hu) |
| DK (1) | DK0453731T3 (hu) |
| ES (1) | ES2121757T3 (hu) |
| FI (1) | FI100533B (hu) |
| GR (1) | GR3027762T3 (hu) |
| HU (1) | HU211774B (hu) |
| IE (1) | IE911366A1 (hu) |
| NO (1) | NO177567C (hu) |
| NZ (1) | NZ237870A (hu) |
| SG (1) | SG47565A1 (hu) |
| TW (1) | TW215087B (hu) |
| ZA (1) | ZA913092B (hu) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5521184A (en) * | 1992-04-03 | 1996-05-28 | Ciba-Geigy Corporation | Pyrimidine derivatives and processes for the preparation thereof |
| US5516775A (en) * | 1992-08-31 | 1996-05-14 | Ciba-Geigy Corporation | Further use of pyrimidine derivatives |
| DE69943247D1 (de) * | 1998-03-27 | 2011-04-14 | Janssen Pharmaceutica Nv | HIV hemmende Pyrimidin Derivate |
| JP4919566B2 (ja) * | 1999-09-24 | 2012-04-18 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | 抗ウイルス組成物 |
| WO2007053776A1 (en) * | 2005-11-03 | 2007-05-10 | Sgx Pharmaceuticals, Inc. | Pyrimidinyl-thiophene kinase modulators |
| CA2686379A1 (en) * | 2007-05-04 | 2008-11-13 | Irm Llc | Phenylaminopyrimidine derivatives and compositions thereof as c-kit and pdgfr kinase inhibitors |
| US9242984B2 (en) | 2012-06-20 | 2016-01-26 | Merck Sharp & Dohme Corp. | Pyrazolyl derivatives as Syk inhibitors |
| WO2013192128A1 (en) * | 2012-06-20 | 2013-12-27 | Merck Sharp & Dohme Corp. | Imidazolyl analogs as syk inhibitors |
| CN110330447B (zh) * | 2019-07-16 | 2022-04-15 | 北京赛升药业股份有限公司 | 一种甲磺酸萘莫司他中间体的制备方法及其应用 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU5319479A (en) * | 1978-12-22 | 1980-06-26 | Ici Australia Limited | Pyrimidinyl amino phenoxy carboxylate derivatives |
| EP0164204A1 (en) * | 1984-05-12 | 1985-12-11 | FISONS plc | Novel pharmaceutically useful pyrimidines |
| US4788195A (en) * | 1986-01-13 | 1988-11-29 | American Cyanamid Company | 4,5,6-substituted-N-(substituted-phenyl)-2-pyrimidinamines |
-
1990
- 1990-04-25 US US07/514,455 patent/US5064963A/en not_active Expired - Fee Related
-
1991
- 1991-02-27 AT AT91102859T patent/ATE170184T1/de active
- 1991-02-27 EP EP91102859A patent/EP0453731B1/en not_active Expired - Lifetime
- 1991-02-27 DE DE69130029T patent/DE69130029T2/de not_active Expired - Fee Related
- 1991-02-27 ES ES91102859T patent/ES2121757T3/es not_active Expired - Lifetime
- 1991-02-27 SG SG1996002850A patent/SG47565A1/en unknown
- 1991-02-27 DK DK91102859T patent/DK0453731T3/da active
- 1991-03-22 TW TW080102248A patent/TW215087B/zh active
- 1991-04-18 NZ NZ237870A patent/NZ237870A/xx unknown
- 1991-04-23 JP JP3117918A patent/JPH04225975A/ja active Pending
- 1991-04-23 CA CA002041031A patent/CA2041031A1/en not_active Abandoned
- 1991-04-24 ZA ZA913092A patent/ZA913092B/xx unknown
- 1991-04-24 NO NO911632A patent/NO177567C/no unknown
- 1991-04-24 HU HU911373A patent/HU211774B/hu not_active IP Right Cessation
- 1991-04-24 AU AU75905/91A patent/AU630849B2/en not_active Ceased
- 1991-04-24 IE IE136691A patent/IE911366A1/en unknown
- 1991-04-24 KR KR1019910006612A patent/KR0168679B1/ko not_active IP Right Cessation
- 1991-04-24 FI FI911983A patent/FI100533B/fi active
-
1998
- 1998-08-27 GR GR980401941T patent/GR3027762T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| DE69130029T2 (de) | 1999-02-18 |
| HU211774B (en) | 1995-12-28 |
| EP0453731B1 (en) | 1998-08-26 |
| EP0453731A2 (en) | 1991-10-30 |
| FI911983A (fi) | 1991-10-26 |
| FI100533B (fi) | 1997-12-31 |
| NO177567B (no) | 1995-07-03 |
| SG47565A1 (en) | 1998-04-17 |
| EP0453731A3 (en) | 1992-09-02 |
| ATE170184T1 (de) | 1998-09-15 |
| US5064963A (en) | 1991-11-12 |
| KR0168679B1 (ko) | 1999-01-15 |
| CA2041031A1 (en) | 1991-10-26 |
| AU7590591A (en) | 1991-11-07 |
| HUT57719A (en) | 1991-12-30 |
| NO911632L (no) | 1991-10-28 |
| NO911632D0 (no) | 1991-04-24 |
| IE911366A1 (en) | 1991-11-06 |
| NZ237870A (en) | 1993-05-26 |
| FI911983A0 (fi) | 1991-04-24 |
| DE69130029D1 (de) | 1998-10-01 |
| GR3027762T3 (en) | 1998-11-30 |
| ES2121757T3 (es) | 1998-12-16 |
| HU911373D0 (en) | 1991-10-28 |
| TW215087B (hu) | 1993-10-21 |
| JPH04225975A (ja) | 1992-08-14 |
| NO177567C (no) | 1995-10-11 |
| AU630849B2 (en) | 1992-11-05 |
| KR910018375A (ko) | 1991-11-30 |
| DK0453731T3 (da) | 1999-02-15 |
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