ZA85696B - Pyrimido(2,1-b)benzothiazoles - Google Patents
Pyrimido(2,1-b)benzothiazolesInfo
- Publication number
- ZA85696B ZA85696B ZA85696A ZA85696A ZA85696B ZA 85696 B ZA85696 B ZA 85696B ZA 85696 A ZA85696 A ZA 85696A ZA 85696 A ZA85696 A ZA 85696A ZA 85696 B ZA85696 B ZA 85696B
- Authority
- ZA
- South Africa
- Prior art keywords
- group
- branched
- straight
- hydrogen atom
- alkyl
- Prior art date
Links
- RWVLSUFUYXWYKA-UHFFFAOYSA-N 4h-pyrimido[2,1-b][1,3]benzothiazole Chemical class C1=CC=C2N3CC=CN=C3SC2=C1 RWVLSUFUYXWYKA-UHFFFAOYSA-N 0.000 title 1
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 3
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 3
- 125000004191 (C1-C6) alkoxy group Chemical group 0.000 abstract 2
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 abstract 2
- 125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 239000000043 antiallergic agent Substances 0.000 abstract 1
- 125000003710 aryl alkyl group Chemical group 0.000 abstract 1
- 125000003118 aryl group Chemical group 0.000 abstract 1
- 229910052799 carbon Inorganic materials 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 125000001072 heteroaryl group Chemical group 0.000 abstract 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
- 125000004573 morpholin-4-yl group Chemical group N1(CCOCC1)* 0.000 abstract 1
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 1
- 229910052757 nitrogen Inorganic materials 0.000 abstract 1
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
- 125000000587 piperidin-1-yl group Chemical group [H]C1([H])N(*)C([H])([H])C([H])([H])C([H])([H])C1([H])[H] 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/82—Nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pulmonology (AREA)
- Public Health (AREA)
- Immunology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Luminescent Compositions (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Saccharide Compounds (AREA)
- Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Polymerisation Methods In General (AREA)
- Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
- Indole Compounds (AREA)
- Compositions Of Macromolecular Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB848403739A GB8403739D0 (en) | 1984-02-13 | 1984-02-13 | Chemical compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA85696B true ZA85696B (en) | 1986-03-26 |
Family
ID=10556508
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA85696A ZA85696B (en) | 1984-02-13 | 1985-01-29 | Pyrimido(2,1-b)benzothiazoles |
Country Status (16)
| Country | Link |
|---|---|
| EP (1) | EP0153230B1 (da) |
| JP (1) | JPS60184086A (da) |
| KR (1) | KR850005847A (da) |
| AT (1) | ATE44745T1 (da) |
| AU (1) | AU574131B2 (da) |
| CA (1) | CA1257259A (da) |
| DE (1) | DE3571621D1 (da) |
| DK (1) | DK63385A (da) |
| ES (2) | ES8702421A1 (da) |
| FI (1) | FI79323C (da) |
| GB (2) | GB8403739D0 (da) |
| GR (1) | GR850369B (da) |
| HU (1) | HU192318B (da) |
| NZ (1) | NZ211104A (da) |
| PT (1) | PT79955B (da) |
| ZA (1) | ZA85696B (da) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8519261D0 (en) * | 1985-07-31 | 1985-09-04 | Roussel Lab Ltd | Chemical compounds |
| US4762840A (en) * | 1984-02-13 | 1988-08-09 | Roussel Uclaf | Pyrimido[2,1-b]benzothiazoles having antiallergic activity |
| AP2013006706A0 (en) | 2010-07-02 | 2013-02-28 | Gilead Sciences Inc | Napht-2-ylacetic acid derivatives to treat AIDS |
| KR20130124291A (ko) | 2010-07-02 | 2013-11-13 | 길리애드 사이언시즈, 인코포레이티드 | Ｈｉｖ 항바이러스 화합물로서의 2-퀴놀리닐-아세트산 유도체 |
| BR112013027096A2 (pt) | 2011-04-21 | 2016-12-27 | Gilead Sciences Inc | compostos de benzotiazol e seu uso farmacêutico |
| US9284323B2 (en) | 2012-01-04 | 2016-03-15 | Gilead Sciences, Inc. | Naphthalene acetic acid derivatives against HIV infection |
| WO2013103724A1 (en) | 2012-01-04 | 2013-07-11 | Gilead Sciences, Inc. | 2- (tert - butoxy) -2- (7 -methylquinolin- 6 - yl) acetic acid derivatives for treating aids |
| ES2571479T3 (es) | 2012-04-20 | 2016-05-25 | Gilead Sciences Inc | Derivados del ácido benzotiazol-6-il acético y su uso para tratar una infección por VIH |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3919201A (en) * | 1970-09-30 | 1975-11-11 | Lilly Industries Ltd | 2-({62 -Aminoacryloyl)iminobenzothiazolines |
| DE2810863A1 (de) * | 1978-03-13 | 1979-09-27 | Boehringer Mannheim Gmbh | 1-oxo-1h-pyrimido eckige klammer auf 6,1-b eckige klammer zu benzthiazol-derivate und verfahren zu ihrer herstellung |
| GB8519261D0 (en) * | 1985-07-31 | 1985-09-04 | Roussel Lab Ltd | Chemical compounds |
-
1984
- 1984-02-13 GB GB848403739A patent/GB8403739D0/en active Pending
-
1985
- 1985-01-13 KR KR1019850000879A patent/KR850005847A/ko not_active Ceased
- 1985-01-29 ZA ZA85696A patent/ZA85696B/xx unknown
- 1985-02-11 DE DE8585400219T patent/DE3571621D1/de not_active Expired
- 1985-02-11 EP EP85400219A patent/EP0153230B1/fr not_active Expired
- 1985-02-11 AT AT85400219T patent/ATE44745T1/de not_active IP Right Cessation
- 1985-02-12 NZ NZ211104A patent/NZ211104A/en unknown
- 1985-02-12 FI FI850582A patent/FI79323C/fi not_active IP Right Cessation
- 1985-02-12 JP JP60023706A patent/JPS60184086A/ja active Pending
- 1985-02-12 HU HU85529A patent/HU192318B/hu not_active IP Right Cessation
- 1985-02-12 ES ES540332A patent/ES8702421A1/es not_active Expired
- 1985-02-12 GB GB08503541A patent/GB2154583B/en not_active Expired
- 1985-02-12 CA CA000474113A patent/CA1257259A/en not_active Expired
- 1985-02-12 GR GR850369A patent/GR850369B/el unknown
- 1985-02-12 PT PT79955A patent/PT79955B/pt not_active IP Right Cessation
- 1985-02-12 DK DK63385A patent/DK63385A/da not_active Application Discontinuation
- 1985-02-13 AU AU38672/85A patent/AU574131B2/en not_active Ceased
-
1986
- 1986-04-01 ES ES553574A patent/ES8800243A1/es not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| HUT38649A (en) | 1986-06-30 |
| DK63385D0 (da) | 1985-02-12 |
| GR850369B (da) | 1985-06-14 |
| ES540332A0 (es) | 1986-12-16 |
| GB2154583A (en) | 1985-09-11 |
| FI79323C (fi) | 1989-12-11 |
| NZ211104A (en) | 1987-08-31 |
| FI850582L (fi) | 1985-08-14 |
| CA1257259A (en) | 1989-07-11 |
| PT79955A (en) | 1985-03-01 |
| KR850005847A (ko) | 1985-09-26 |
| ES8800243A1 (es) | 1987-10-16 |
| DE3571621D1 (en) | 1989-08-24 |
| JPS60184086A (ja) | 1985-09-19 |
| PT79955B (en) | 1987-02-02 |
| ES553574A0 (es) | 1987-10-16 |
| GB2154583B (en) | 1987-10-28 |
| ATE44745T1 (de) | 1989-08-15 |
| EP0153230B1 (fr) | 1989-07-19 |
| HU192318B (en) | 1987-05-28 |
| EP0153230A3 (en) | 1986-10-01 |
| FI850582A0 (fi) | 1985-02-12 |
| FI79323B (fi) | 1989-08-31 |
| GB8503541D0 (en) | 1985-03-13 |
| AU574131B2 (en) | 1988-06-30 |
| ES8702421A1 (es) | 1986-12-16 |
| GB8403739D0 (en) | 1984-03-14 |
| DK63385A (da) | 1985-08-14 |
| AU3867285A (en) | 1985-08-22 |
| EP0153230A2 (fr) | 1985-08-28 |
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