GB8519261D0 - Chemical compounds - Google Patents

Chemical compounds

Info

Publication number
GB8519261D0
GB8519261D0 GB858519261A GB8519261A GB8519261D0 GB 8519261 D0 GB8519261 D0 GB 8519261D0 GB 858519261 A GB858519261 A GB 858519261A GB 8519261 A GB8519261 A GB 8519261A GB 8519261 D0 GB8519261 D0 GB 8519261D0
Authority
GB
United Kingdom
Prior art keywords
group
chained
branched
straight
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
GB858519261A
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Roussel Laboratories Ltd
Original Assignee
Roussel Laboratories Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Laboratories Ltd filed Critical Roussel Laboratories Ltd
Priority to GB858519261A priority Critical patent/GB8519261D0/en
Publication of GB8519261D0 publication Critical patent/GB8519261D0/en
Priority to ZA865170A priority patent/ZA865170B/en
Priority to JP61171948A priority patent/JPS6229592A/en
Priority to DK361286A priority patent/DK361286A/en
Priority to ES8600714A priority patent/ES2002111A6/en
Priority to GR862015A priority patent/GR862015B/en
Priority to CA000514995A priority patent/CA1286290C/en
Priority to AU60687/86A priority patent/AU586010B2/en
Priority to SU864027859A priority patent/SU1544191A3/en
Priority to GB8618641A priority patent/GB2178429B/en
Priority to PT83099A priority patent/PT83099B/en
Priority to FI863118A priority patent/FI863118A/en
Priority to NZ217026A priority patent/NZ217026A/en
Priority to DE8686401707T priority patent/DE3678764D1/en
Priority to AT86401707T priority patent/ATE62689T1/en
Priority to HU863299A priority patent/HU194895B/en
Priority to EP86401707A priority patent/EP0211759B1/en
Priority to KR1019860006314A priority patent/KR870001221A/en
Priority to US06/892,771 priority patent/US4762840A/en
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/22—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D277/26—Radicals substituted by sulfur atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Immunology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

The present invention relates to compounds of formula I <IMAGE> [wherein R and R3,which may be the same or different, each represents a hydrogen atom or a straight-chained or branched C1-6 alkyl group or together with the intervening carbon atom represent a C3-6 cycloalkyl group; R1 represents a C7-12 straight-chained, branched or cyclic alkoxy group; and R2 represents a hydrogen atom, a straight-chained or branched C1-6 alkyl group, a C2-7 alkoxycarbonyl group, a C3-6 cycloalkyl group, an aralkyl group, an aryl group (unsubstituted or substituted by one or more halogen atoms or C1-6 alkyl, C1-6 alkoxy or nitro groups) or a heteroaryl group] and acid addition salts thereof, to processes for their preparation and to their application as drugs. Compounds 1 have anti-allergy activity.
GB858519261A 1984-02-13 1985-07-31 Chemical compounds Pending GB8519261D0 (en)

Priority Applications (19)

Application Number Priority Date Filing Date Title
GB858519261A GB8519261D0 (en) 1985-07-31 1985-07-31 Chemical compounds
ZA865170A ZA865170B (en) 1985-07-31 1986-07-10 Derivatives of pyrimido/2,1-b/benzothiazole and their salts,process of preparation,application as medicaments and compositions containing them
JP61171948A JPS6229592A (en) 1985-07-31 1986-07-23 Novel pyrimido(2,1 b)benzothiazoles and salts, manufacture and use as drugs
ES8600714A ES2002111A6 (en) 1985-07-31 1986-07-30 Pyrimido[2,1-b]benzothiazole derivatives and their salts, process for their preparation, use as medicaments and compositions containing them.
SU864027859A SU1544191A3 (en) 1985-07-31 1986-07-30 Method of producing derivatives of pyrimido(2,1-b)benzthiazol
NZ217026A NZ217026A (en) 1985-07-31 1986-07-30 Pyrimido (1,2-b) benzothiazole derivatives and pharmaceutical compositions
GR862015A GR862015B (en) 1985-07-31 1986-07-30 Chemical compositions
CA000514995A CA1286290C (en) 1985-07-31 1986-07-30 Anti-allergic pyrimido[2,1-l-b]benzothiazoles
AU60687/86A AU586010B2 (en) 1985-07-31 1986-07-30 Pyrimido``2,1-b`` benzothiazole derivatives
DK361286A DK361286A (en) 1985-07-31 1986-07-30 PYRAMIDO (2,1-B) BENZOTHIAZOLES AND SALTS THEREOF, PROCEDURE FOR THEIR PREPARATION AND MEDICINES WITH CONTENTS
GB8618641A GB2178429B (en) 1985-07-31 1986-07-30 Pyrimido [2,1-6]-benzothiazole-8-acetic acid derivitives
PT83099A PT83099B (en) 1985-07-31 1986-07-30 PROCESS FOR THE PREPARATION OF NEW PYRIMIDES (2,1-B} BENZOTIAZOES WITH ANTI-ALLERGIC PROPERTIES
FI863118A FI863118A (en) 1985-07-31 1986-07-30 CHEMICAL FOERENINGAR.
DE8686401707T DE3678764D1 (en) 1985-07-31 1986-07-31 PYRIMIDO (2,1-B) BENZOTHIAZOLE DERIVATIVES AND THEIR SALTS, METHOD FOR THE PRODUCTION THEREOF, USE AS MEDICINAL PRODUCTS AND THE PREPARATIONS CONTAINING THE SAME.
US06/892,771 US4762840A (en) 1984-02-13 1986-07-31 Pyrimido[2,1-b]benzothiazoles having antiallergic activity
AT86401707T ATE62689T1 (en) 1985-07-31 1986-07-31 PYRIMIDO(2,1-B>BENZOTHIAZOLE DERIVATIVES AND THEIR SALTS, PROCESS FOR THEIR MANUFACTURE, USE AS MEDICINAL PRODUCTS AND THE PREPARATIONS CONTAINING THEM.
HU863299A HU194895B (en) 1985-07-31 1986-07-31 Process for production of new pyrimide /2,1-b/ benzothiasoles and medical preparatives containing these substances
EP86401707A EP0211759B1 (en) 1985-07-31 1986-07-31 Pyrimido[2,1-b]benzothiazole derivatives and their salts, process for their preparation, use as medicaments and compositions containing them
KR1019860006314A KR870001221A (en) 1985-07-31 1986-07-31 Method for preparing pyrimido- [2,1-b] benzothiazole and salts thereof

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB858519261A GB8519261D0 (en) 1985-07-31 1985-07-31 Chemical compounds

Publications (1)

Publication Number Publication Date
GB8519261D0 true GB8519261D0 (en) 1985-09-04

Family

ID=10583097

Family Applications (2)

Application Number Title Priority Date Filing Date
GB858519261A Pending GB8519261D0 (en) 1984-02-13 1985-07-31 Chemical compounds
GB8618641A Expired GB2178429B (en) 1985-07-31 1986-07-30 Pyrimido [2,1-6]-benzothiazole-8-acetic acid derivitives

Family Applications After (1)

Application Number Title Priority Date Filing Date
GB8618641A Expired GB2178429B (en) 1985-07-31 1986-07-30 Pyrimido [2,1-6]-benzothiazole-8-acetic acid derivitives

Country Status (17)

Country Link
EP (1) EP0211759B1 (en)
JP (1) JPS6229592A (en)
KR (1) KR870001221A (en)
AT (1) ATE62689T1 (en)
AU (1) AU586010B2 (en)
CA (1) CA1286290C (en)
DE (1) DE3678764D1 (en)
DK (1) DK361286A (en)
ES (1) ES2002111A6 (en)
FI (1) FI863118A (en)
GB (2) GB8519261D0 (en)
GR (1) GR862015B (en)
HU (1) HU194895B (en)
NZ (1) NZ217026A (en)
PT (1) PT83099B (en)
SU (1) SU1544191A3 (en)
ZA (1) ZA865170B (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8403739D0 (en) * 1984-02-13 1984-03-14 Roussel Lab Ltd Chemical compounds
GB8522186D0 (en) * 1985-09-06 1985-10-09 Erba Farmitalia Cycloalkyl-substituted 4-aminophenyl derivatives

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3919201A (en) * 1970-09-30 1975-11-11 Lilly Industries Ltd 2-({62 -Aminoacryloyl)iminobenzothiazolines
DE2810863A1 (en) * 1978-03-13 1979-09-27 Boehringer Mannheim Gmbh 1-OXO-1H-PYRIMIDO ANGLE CLAMP ON 6.1-B ANGLE CLAMP ON BENZTHIAZOLE DERIVATIVES AND METHOD FOR THE PRODUCTION THEREOF
GB8403739D0 (en) * 1984-02-13 1984-03-14 Roussel Lab Ltd Chemical compounds

Also Published As

Publication number Publication date
EP0211759B1 (en) 1991-04-17
AU586010B2 (en) 1989-06-29
ATE62689T1 (en) 1991-05-15
FI863118A0 (en) 1986-07-30
GB2178429A (en) 1987-02-11
PT83099A (en) 1986-08-01
FI863118A (en) 1987-02-01
NZ217026A (en) 1989-02-24
KR870001221A (en) 1987-03-12
GB8618641D0 (en) 1986-09-10
GR862015B (en) 1986-12-23
EP0211759A3 (en) 1988-03-30
CA1286290C (en) 1991-07-16
HUT42776A (en) 1987-08-28
JPS6229592A (en) 1987-02-07
HU194895B (en) 1988-03-28
DK361286D0 (en) 1986-07-30
SU1544191A3 (en) 1990-02-15
DK361286A (en) 1987-02-01
GB2178429B (en) 1989-09-13
EP0211759A2 (en) 1987-02-25
ES2002111A6 (en) 1988-07-16
AU6068786A (en) 1987-02-05
PT83099B (en) 1988-11-30
DE3678764D1 (en) 1991-05-23
ZA865170B (en) 1987-09-30

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