ZA834371B - 3-phenoxy-1-azetidinecarboxamides - Google Patents

3-phenoxy-1-azetidinecarboxamides

Info

Publication number
ZA834371B
ZA834371B ZA834371A ZA834371A ZA834371B ZA 834371 B ZA834371 B ZA 834371B ZA 834371 A ZA834371 A ZA 834371A ZA 834371 A ZA834371 A ZA 834371A ZA 834371 B ZA834371 B ZA 834371B
Authority
ZA
South Africa
Prior art keywords
azetidinecarboxamides
phenoxy
Prior art date
Application number
ZA834371A
Other languages
English (en)
Inventor
Chen Teng Lina
Original Assignee
Robins Co Inc A H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Robins Co Inc A H filed Critical Robins Co Inc A H
Publication of ZA834371B publication Critical patent/ZA834371B/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/04Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
ZA834371A 1982-08-19 1983-06-14 3-phenoxy-1-azetidinecarboxamides ZA834371B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US40947682A 1982-08-19 1982-08-19

Publications (1)

Publication Number Publication Date
ZA834371B true ZA834371B (en) 1984-03-28

Family

ID=23620657

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA834371A ZA834371B (en) 1982-08-19 1983-06-14 3-phenoxy-1-azetidinecarboxamides

Country Status (25)

Country Link
EP (1) EP0102194B1 (pm)
JP (1) JPH0643388B2 (pm)
KR (1) KR900001210B1 (pm)
AU (1) AU553528B2 (pm)
CA (1) CA1173841A (pm)
CS (1) CS236796B2 (pm)
DE (1) DE3367089D1 (pm)
DK (1) DK165741C (pm)
EG (1) EG16472A (pm)
ES (1) ES523193A0 (pm)
FI (1) FI77225C (pm)
GR (1) GR79634B (pm)
HK (1) HK47487A (pm)
HU (1) HU190608B (pm)
IE (1) IE55769B1 (pm)
IL (1) IL68699A (pm)
IN (1) IN157045B (pm)
MX (1) MX9203639A (pm)
NO (1) NO157976C (pm)
NZ (1) NZ205317A (pm)
PH (1) PH19595A (pm)
PL (1) PL140765B1 (pm)
PT (1) PT77217B (pm)
YU (1) YU44854B (pm)
ZA (1) ZA834371B (pm)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4594189A (en) * 1983-07-06 1986-06-10 A. H. Robins Company, Inc. Process for preparing 3-phenoxy-1-azetidines and carboxamide derivatives
US5151418A (en) * 1985-02-28 1992-09-29 A. H. Robins Company, Incorporated Method of treating muscular tension, muscle spasticity and anxiety with 3-aryloxy and 3-arylthioazetidinecarboxamides
US4956359A (en) * 1985-02-28 1990-09-11 A. H. Robins Company, Inc. 3-aryloxy and 3-arylthioazetidinecarboxamides as anticonvulsants and antiepileptics
FI87559C (fi) * 1985-02-28 1993-01-25 Robins Co Inc A H Foerfarande foer framstaellning av aktiva 3-fenyloxiazetidinkarboxamider
ZA861210B (en) * 1985-02-28 1987-10-28 Robins Co Inc A H 3-aryloxyazetidinecarboxamides as anticonvulsants and antiepileptics
US5183902A (en) * 1985-02-28 1993-02-02 A. H. Robins Company, Incorporated Method of treating muscular tension, muscle spasticity and anxiety with 3-aryloxy and 3-arylthioazetidinecarboxamides
US5068231A (en) * 1985-02-28 1991-11-26 A. H. Robins Company Incorporated Method of treating muscular tension, muscle spasticity and anxiety with 3-aryloxy and 3-arylthioazetidinecarboxamides
IN162808B (pm) * 1985-02-28 1988-07-09 Robins Co Inc A H
US5183903A (en) * 1991-11-26 1993-02-02 A. H. Robins Company, Incorporated Urea fusion process for the synthesis of 3-phenoxy-1-azetidinecarboxamides
WO1999037612A1 (en) * 1998-01-23 1999-07-29 Vernalis Research Limited Azetidinecarboxamide derivatives for treating cns disorders
ES2181387T3 (es) * 1998-01-23 2003-02-16 Vernalis Res Ltd Derivados de azetidinocarboxamida para el tratamiento de trastornos del sistema nervioso central.
GB9917386D0 (en) * 1999-07-23 1999-09-22 Cerebrus Ltd Chemical compounds-II
CN113754541B (zh) * 2020-06-02 2025-01-03 深圳湾实验室 靶向eb病毒核抗原蛋白的小分子抑制剂、制备方法及其应用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB872447A (en) * 1958-12-23 1961-07-12 Lepetit Spa 1-carbamyl-3-substituted azetidines
US4226861A (en) * 1978-04-18 1980-10-07 A. H. Robins Company, Inc. N-Lower-alkyl 3-phenoxy-1-azetidinecarboxamides

Also Published As

Publication number Publication date
DK376183D0 (da) 1983-08-17
AU553528B2 (en) 1986-07-17
IE55769B1 (en) 1991-01-16
JPH0643388B2 (ja) 1994-06-08
KR900001210B1 (ko) 1990-02-28
ES8500225A1 (es) 1984-10-01
YU158683A (en) 1985-12-31
FI77225C (fi) 1989-02-10
CS236796B2 (en) 1985-05-15
PL243255A1 (en) 1984-08-27
PT77217B (en) 1986-02-04
IL68699A0 (en) 1983-09-30
HU190608B (en) 1986-09-29
PT77217A (en) 1983-09-01
NO157976B (no) 1988-03-14
KR840005715A (ko) 1984-11-15
IE831651L (en) 1984-02-19
DK165741C (da) 1993-06-07
GR79634B (pm) 1984-10-31
IN157045B (pm) 1986-01-04
AU1459783A (en) 1984-02-23
NO832971L (no) 1984-02-20
EP0102194B1 (en) 1986-10-22
CA1173841A (en) 1984-09-04
IL68699A (en) 1986-08-31
NZ205317A (en) 1985-08-30
NO157976C (no) 1988-06-22
HK47487A (en) 1987-06-26
MX9203639A (es) 1992-07-01
DK165741B (da) 1993-01-11
DE3367089D1 (en) 1986-11-27
FI77225B (fi) 1988-10-31
PL140765B1 (en) 1987-05-30
PH19595A (en) 1986-05-26
JPS5980657A (ja) 1984-05-10
YU44854B (en) 1991-04-30
ES523193A0 (es) 1984-10-01
FI832956A0 (fi) 1983-08-18
FI832956L (fi) 1984-02-20
EG16472A (en) 1987-03-30
EP0102194A1 (en) 1984-03-07
DK376183A (da) 1984-02-20

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