ZA812085B - Novel 3-(1-piperidinylalkyl)4h-pyrido(1,2-a)pyrimidin-4one derivatives - Google Patents

Novel 3-(1-piperidinylalkyl)4h-pyrido(1,2-a)pyrimidin-4one derivatives

Info

Publication number
ZA812085B
ZA812085B ZA00812085A ZA812085A ZA812085B ZA 812085 B ZA812085 B ZA 812085B ZA 00812085 A ZA00812085 A ZA 00812085A ZA 812085 A ZA812085 A ZA 812085A ZA 812085 B ZA812085 B ZA 812085B
Authority
ZA
South Africa
Prior art keywords
piperidinylalkyl
pyrido
pyrimidin
novel
4one
Prior art date
Application number
ZA00812085A
Other languages
English (en)
Inventor
L Kennis
J Mertens
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of ZA812085B publication Critical patent/ZA812085B/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
ZA00812085A 1980-03-28 1981-03-27 Novel 3-(1-piperidinylalkyl)4h-pyrido(1,2-a)pyrimidin-4one derivatives ZA812085B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US13484580A 1980-03-28 1980-03-28

Publications (1)

Publication Number Publication Date
ZA812085B true ZA812085B (en) 1982-11-24

Family

ID=22465278

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA00812085A ZA812085B (en) 1980-03-28 1981-03-27 Novel 3-(1-piperidinylalkyl)4h-pyrido(1,2-a)pyrimidin-4one derivatives

Country Status (5)

Country Link
JP (1) JPS56150091A (OSRAM)
KR (2) KR850000412B1 (OSRAM)
PL (2) PL132428B1 (OSRAM)
SU (1) SU1093251A3 (OSRAM)
ZA (1) ZA812085B (OSRAM)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0615529B2 (ja) * 1985-04-01 1994-03-02 エーザイ株式会社 新規ピペリジン誘導体
NZ228447A (en) * 1988-03-28 1990-08-28 Janssen Pharmaceutica Nv Cosmetic or pharmaceutical composition possessing serotonin antogonistic activity
CN101970427A (zh) 2008-02-29 2011-02-09 Vm生物医药公司 治疗疼痛症状及其它失调的方法
MX354074B (es) * 2012-02-10 2018-02-12 Ptc Therapeutics Inc Compuestos para tratar la atrofia muscular espinal.
EP4249472A3 (en) 2015-05-30 2023-12-13 PTC Therapeutics, Inc. Methods for modulating rna splicing
MX391850B (es) 2015-12-10 2025-03-19 Ptc Therapeutics Inc Compuestos para usarse en el tratamiento o mejoramiento de la enfermedad de huntington
MX2019005588A (es) 2016-11-28 2019-10-15 Ptc Therapeutics Inc Metodos para modular corte y empalme de arn.
CA3066224A1 (en) 2017-06-05 2018-12-13 Ptc Therapeutics Inc. Compounds for treating huntington's disease
KR20200017476A (ko) 2017-06-14 2020-02-18 피티씨 테라퓨틱스, 인크. Rna 스플라이싱의 변경 방법
MX2019015580A (es) 2017-06-28 2020-07-28 Ptc Therapeutics Inc Metodos para tratar la enfermedad de huntington.
US11382918B2 (en) 2017-06-28 2022-07-12 Ptc Therapeutics, Inc. Methods for treating Huntington's Disease
JP7399870B2 (ja) 2018-03-27 2023-12-18 ピーティーシー セラピューティクス, インコーポレイテッド ハンチントン病を処置するための化合物
KR20210038845A (ko) 2018-06-27 2021-04-08 피티씨 테라퓨틱스, 인크. 헌팅턴병 치료를 위한 헤테로아릴 화합물
US11685746B2 (en) 2018-06-27 2023-06-27 Ptc Therapeutics, Inc. Heteroaryl compounds for treating Huntington's disease
HUE068060T2 (hu) 2018-06-27 2024-12-28 Ptc Therapeutics Inc Heterociklikus és heteroaril vegyületek Huntington-kór kezelésére

Also Published As

Publication number Publication date
PL131162B1 (en) 1984-10-31
PL230364A1 (OSRAM) 1982-03-29
KR850000413B1 (ko) 1985-03-26
PL233902A1 (OSRAM) 1982-07-19
JPH0215550B2 (OSRAM) 1990-04-12
JPS56150091A (en) 1981-11-20
KR830005220A (ko) 1983-08-03
PL132428B1 (en) 1985-03-30
KR850000412B1 (ko) 1985-03-26
SU1093251A3 (ru) 1984-05-15

Similar Documents

Publication Publication Date Title
PT72740A (en) Novel 3-(1-piperidinylalkyl)-4h-pyrido/1,2-a/-pyrimidin-4-one derivatives
AU540840B2 (en) Imidazo(1,2-a)pyridines
GB2035303B (en) 2,3-dicyano-hydroquinone derivatives
AU531348B2 (en) 1,8 naphthyridine derivatives
ZA812085B (en) Novel 3-(1-piperidinylalkyl)4h-pyrido(1,2-a)pyrimidin-4one derivatives
AU7600481A (en) Imidazo (4,5-b)pyridines
AU515352B2 (en) 1, 2-DIHYDRO-3H-PYRROLE (1, 2-a)-PYRROLE-1-NITRILES
GB2098203B (en) Novel 4,5-diaryl-thiazole-2-thiol derivatives
NZ194529A (en) 9,10-dihydro-1h, 4h-pyrazolo (4,3-b)(1,5)benzodiazepin-10-ones
GB2067567B (en) 24,24-difluoro-cyclovitamin d3 derivatives
AU7338081A (en) 1,2,4-triazolylpropenol derivatives
NZ195248A (en) 4-(piperaz-1-yl)-2,10-dihydropyrazolo (3,4-b)(1,5)-benzodiazepines
CS528780A2 (en) Zpusob vyroby substituovanych pyrido-(1,2-a)pyrimidinu
GB2017093B (en) 3,3-dichloro-2-azetidinone derivatives
JPS5732239A (en) 2,3-bis-hydroxybenzyl derivative
NZ197563A (en) 3-(1,2,4-triazinylthiomethyl)-3-cephem-1-sulphoxide derivatives
IL61535A0 (en) 1-oxo-1h-thiazolo(3,2-a)pyrimidine-2-carboxamides
GB2092130B (en) 4-oximino-1,2,3,4-tetrahydroquinoline derivatives
AU521104B2 (en) (1,3-thiazino) (3,4-b)-isoquinolines
GB2080794B (en) 1,6-naphthyridine derivatives
PH14888A (en) 1,2,3,4-tetrahydro-9h-pyrrolo(3,4-b)quinolin-9-one derivative
GB2013678B (en) 1,4 benzoazine derivatives
AU7744681A (en) 2,3-dihydro-4-pyrone derivatives
NZ192622A (en) 4,7-phenanthroline derivatives
AU542710B2 (en) 16-amino-17-phenyl-18,19,20-trinor-prosta-glandin derivatives