ZA795508B - Derivatives of polyene macrolide antibiotics containing an amino sugar moiety, process for the preparation thereof, and pharmaceutical compositions containing them - Google Patents

Derivatives of polyene macrolide antibiotics containing an amino sugar moiety, process for the preparation thereof, and pharmaceutical compositions containing them

Info

Publication number
ZA795508B
ZA795508B ZA00795508A ZA795508A ZA795508B ZA 795508 B ZA795508 B ZA 795508B ZA 00795508 A ZA00795508 A ZA 00795508A ZA 795508 A ZA795508 A ZA 795508A ZA 795508 B ZA795508 B ZA 795508B
Authority
ZA
South Africa
Prior art keywords
hydrogen
zero
polyene macrolide
compounds
phenylpropargyl
Prior art date
Application number
ZA00795508A
Other languages
English (en)
Inventor
J Wright
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corp filed Critical Schering Corp
Priority to ES485140A priority Critical patent/ES8102146A1/es
Priority to ES492083A priority patent/ES492083A0/es
Priority to ES492082A priority patent/ES8200373A1/es
Publication of ZA795508B publication Critical patent/ZA795508B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
ZA00795508A 1978-10-23 1979-10-16 Derivatives of polyene macrolide antibiotics containing an amino sugar moiety, process for the preparation thereof, and pharmaceutical compositions containing them ZA795508B (en)

Priority Applications (3)

Application Number Priority Date Filing Date Title
ES485140A ES8102146A1 (es) 1978-10-23 1979-10-18 Procedimiento para la preparacion de derivados de antibioti-co de polienmacrolida
ES492083A ES492083A0 (es) 1979-10-16 1980-06-02 Procedimiento para la preparacion de esteres de antibiotico de polienmacrolida
ES492082A ES8200373A1 (es) 1978-10-23 1980-06-02 Procedimiento para la preparacion de derivados de antibioti-co de polienmacrolida

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US95382478A 1978-10-23 1978-10-23

Publications (1)

Publication Number Publication Date
ZA795508B true ZA795508B (en) 1981-05-27

Family

ID=25494578

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA00795508A ZA795508B (en) 1978-10-23 1979-10-16 Derivatives of polyene macrolide antibiotics containing an amino sugar moiety, process for the preparation thereof, and pharmaceutical compositions containing them

Country Status (14)

Country Link
EP (1) EP0010297B1 (no)
JP (1) JPS5557600A (no)
AT (1) ATE3046T1 (no)
AU (1) AU5190079A (no)
CA (1) CA1132542A (no)
DE (1) DE2965212D1 (no)
DK (1) DK439879A (no)
FI (1) FI793236A (no)
GR (1) GR74128B (no)
HU (1) HU181506B (no)
IL (1) IL58490A (no)
NO (1) NO147840C (no)
PT (1) PT70341A (no)
ZA (1) ZA795508B (no)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS59104326A (ja) * 1982-12-04 1984-06-16 Toyo Jozo Co Ltd マクロライド抗生物質の安定な経口用製剤および安定化法
FR2574075B1 (fr) * 1984-12-04 1987-09-18 Poudres & Explosifs Ste Nale Procede de synthese d'esters actifs d'acides carboxyliques, nouveaux carbonates alpha-halogenes utiles pour cette synthese et leur mode d'obtention
MX9706283A (es) * 1996-08-19 1998-02-28 Hoechst Ag Nuevos antibioticos de polieno, 3874 hi a h6, procedimientos para su preparacion y empleo.
EP0987273A4 (en) * 1997-06-03 2001-11-07 Ajinomoto Kk PROCESS FOR PRODUCING ANTIFUNGAL V-28-3M
US5981721A (en) * 1997-10-23 1999-11-09 Karykion Corporation Polyene macrolide schiff bases, their alkyl esters and processes for preparing polyene macrolide alkyl ester salts thereof
JP2010534688A (ja) * 2007-07-30 2010-11-11 上海医薬工業研究院 ポリエン類抗生物質ジエステル化合物
WO2020119773A1 (zh) * 2018-12-13 2020-06-18 上海医药工业研究院 两性霉素b肽衍生物

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3244590A (en) * 1960-12-23 1966-04-05 Rutgers Res And Educational Fo Polyenic compounds and procedures related thereto
US4038382A (en) 1972-07-24 1977-07-26 Spa-Societe Prodotti Antibiotici S.P.A. Alkyl esters of polyene antibiotics
GB1399139A (en) 1972-07-24 1975-06-25 Prodotti Antibiotici Spa Alkyl esters of polyene antibiotics
US4041232A (en) * 1976-02-23 1977-08-09 E. R. Squibb & Sons, Inc. Amphotericin B methyl ester salts

Also Published As

Publication number Publication date
HU181506B (en) 1983-10-28
ATE3046T1 (de) 1983-04-15
IL58490A (en) 1983-07-31
AU5190079A (en) 1980-05-01
CA1132542A (en) 1982-09-28
EP0010297A1 (en) 1980-04-30
IL58490A0 (en) 1980-01-31
GR74128B (no) 1984-06-06
EP0010297B1 (en) 1983-04-13
NO793354L (no) 1980-04-24
NO147840B (no) 1983-03-14
DE2965212D1 (en) 1983-05-19
JPS5557600A (en) 1980-04-28
NO147840C (no) 1983-06-22
DK439879A (da) 1980-04-24
PT70341A (en) 1979-11-01
FI793236A (fi) 1980-04-24

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