ZA201608331B - Aminoester derivatives - Google Patents

Aminoester derivatives

Info

Publication number
ZA201608331B
ZA201608331B ZA2016/08331A ZA201608331A ZA201608331B ZA 201608331 B ZA201608331 B ZA 201608331B ZA 2016/08331 A ZA2016/08331 A ZA 2016/08331A ZA 201608331 A ZA201608331 A ZA 201608331A ZA 201608331 B ZA201608331 B ZA 201608331B
Authority
ZA
South Africa
Prior art keywords
aminoester derivatives
aminoester
derivatives
Prior art date
Application number
ZA2016/08331A
Other languages
English (en)
Inventor
Armani Elisabetta
Amari Gabriele
Capaldi Carmelida
Blackaby Wesley
Linney Ian
Van De Pöel Hervé
Baker-Glenn Charles
Trivedi Naimisha
Original Assignee
Chiesi Farmaceutici S P A An Incorporated Business Forming A Joint Stock Company Of Italian Nat
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chiesi Farmaceutici S P A An Incorporated Business Forming A Joint Stock Company Of Italian Nat filed Critical Chiesi Farmaceutici S P A An Incorporated Business Forming A Joint Stock Company Of Italian Nat
Publication of ZA201608331B publication Critical patent/ZA201608331B/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4436Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a heterocyclic ring having sulfur as a ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/04Drugs for disorders of the respiratory system for throat disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Hydrogenated Pyridines (AREA)
ZA2016/08331A 2014-06-05 2016-12-02 Aminoester derivatives ZA201608331B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP14171266 2014-06-05
PCT/EP2015/062417 WO2015185649A1 (en) 2014-06-05 2015-06-03 Aminoester derivatives

Publications (1)

Publication Number Publication Date
ZA201608331B true ZA201608331B (en) 2018-05-30

Family

ID=50884281

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA2016/08331A ZA201608331B (en) 2014-06-05 2016-12-02 Aminoester derivatives

Country Status (32)

Country Link
US (2) US9763924B2 (enExample)
EP (1) EP3152201B1 (enExample)
JP (1) JP2017516824A (enExample)
KR (1) KR102420323B1 (enExample)
CN (1) CN106459020B (enExample)
AR (1) AR100732A1 (enExample)
AU (1) AU2015270539B2 (enExample)
BR (1) BR112016026725B1 (enExample)
CA (1) CA2953198C (enExample)
CL (1) CL2016003117A1 (enExample)
CY (1) CY1120698T1 (enExample)
DK (1) DK3152201T3 (enExample)
EA (1) EA032761B1 (enExample)
ES (1) ES2688826T3 (enExample)
GE (1) GEP20186922B (enExample)
HR (1) HRP20181967T1 (enExample)
HU (1) HUE042119T2 (enExample)
IL (1) IL249325B (enExample)
LT (1) LT3152201T (enExample)
MA (1) MA39947B1 (enExample)
MX (1) MX377669B (enExample)
PE (1) PE20161557A1 (enExample)
PH (1) PH12016502221A1 (enExample)
PL (1) PL3152201T3 (enExample)
PT (1) PT3152201T (enExample)
RS (1) RS57787B1 (enExample)
SG (1) SG11201610132RA (enExample)
SI (1) SI3152201T1 (enExample)
TN (1) TN2016000546A1 (enExample)
TW (1) TW201625600A (enExample)
WO (1) WO2015185649A1 (enExample)
ZA (1) ZA201608331B (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2016177849A1 (en) 2015-05-07 2016-11-10 Chiesi Farmaceutici S.P.A. Aminoester derivatives
AR104822A1 (es) * 2015-06-01 2017-08-16 Chiesi Farm Spa Derivado de aminoésteres
TW201710254A (zh) * 2015-06-01 2017-03-16 吉斯藥品公司 胺基酯衍生物
CN106866474B (zh) * 2017-02-16 2018-12-28 陕西师范大学 一种手性α-芳基甘氨酸酯衍生物的合成方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2022783A1 (en) * 2007-08-08 2009-02-11 CHIESI FARMACEUTICI S.p.A. "Derivatives of 1-phenyl-2-pyridinyl alkyl alcohols as phosphodiesterase inhibitors"
TW201000476A (en) * 2008-02-06 2010-01-01 Glaxo Group Ltd Dual pharmacophores-PDE4-muscarinic antagonistics
EP2216327A1 (en) * 2009-02-06 2010-08-11 CHIESI FARMACEUTICI S.p.A. Benzoic acid (1-phenyl-2-pyridin-4-yl)ethyl esters as phosphodiesterase inhibitors
EP2928883B1 (en) 2012-12-05 2018-02-14 Chiesi Farmaceutici S.p.A. Phenylethylpyridine derivatives as pde4-inhibitors and muscarinic receptor antagonists
CA2893663A1 (en) 2012-12-05 2014-06-12 Chiesi Farmaceutici S.P.A. Phenylethylpyridine derivatives as pde4-inhibitors
CN104822669A (zh) * 2012-12-05 2015-08-05 奇斯药制品公司 作为pde-4抑制剂的苯基乙基吡啶衍生物
HK1225384A1 (zh) 2013-12-05 2017-09-08 奇斯药制品公司 用於治疗呼吸病的二苯甲基衍生物
EP3077385B1 (en) * 2013-12-05 2017-10-04 Chiesi Farmaceutici S.p.A. Heteroaryl derivatives for the treatment of respiratory diseases

Also Published As

Publication number Publication date
AR100732A1 (es) 2016-10-26
MA39947A (fr) 2017-04-12
WO2015185649A9 (en) 2017-01-05
CN106459020A (zh) 2017-02-22
KR102420323B1 (ko) 2022-07-13
US20170340616A1 (en) 2017-11-30
CY1120698T1 (el) 2019-12-11
AU2015270539B2 (en) 2018-11-08
TW201625600A (zh) 2016-07-16
BR112016026725A2 (pt) 2017-08-15
RS57787B1 (sr) 2018-12-31
CA2953198C (en) 2023-06-13
PH12016502221A1 (en) 2017-02-06
HRP20181967T1 (hr) 2019-02-08
IL249325A0 (en) 2017-02-28
SI3152201T1 (sl) 2018-10-30
US10117860B2 (en) 2018-11-06
CL2016003117A1 (es) 2017-06-23
PL3152201T3 (pl) 2019-02-28
KR20170015294A (ko) 2017-02-08
PE20161557A1 (es) 2017-02-07
EA201692227A1 (ru) 2017-05-31
EA032761B1 (ru) 2019-07-31
MA39947B1 (fr) 2018-10-31
PT3152201T (pt) 2018-10-26
TN2016000546A1 (en) 2018-04-04
CA2953198A1 (en) 2015-12-10
MX2016015958A (es) 2017-04-10
JP2017516824A (ja) 2017-06-22
BR112016026725A8 (pt) 2021-06-29
WO2015185649A1 (en) 2015-12-10
EP3152201B1 (en) 2018-08-29
HUE042119T2 (hu) 2019-06-28
DK3152201T3 (en) 2018-11-19
US20150352091A1 (en) 2015-12-10
MX377669B (es) 2025-03-11
AU2015270539A1 (en) 2016-12-22
IL249325B (en) 2018-12-31
BR112016026725B1 (pt) 2024-02-27
LT3152201T (lt) 2018-10-10
EP3152201A1 (en) 2017-04-12
US9763924B2 (en) 2017-09-19
ES2688826T3 (es) 2018-11-07
CN106459020B (zh) 2019-06-18
GEP20186922B (en) 2018-11-12
SG11201610132RA (en) 2017-01-27

Similar Documents

Publication Publication Date Title
GB201413050D0 (en) None
GB201516266D0 (en) None
GB201516146D0 (en) None
ZA201704602B (en) Dihydroindolizinone derivative
SG11201609205WA (en) Heterocyclyl-butanamide derivatives
PL3418273T3 (pl) Pochodne flawaglin
HUE050450T2 (hu) Fluoralkil-fluorén-származékok
IL248773A0 (en) History of naphthyridinedione
IL248629A0 (en) Substances containing diheteroaryl conjugated to cycloalkyl and their uses
HUE044703T2 (hu) Új CYP-eikozanoid származékok
ZA201608331B (en) Aminoester derivatives
IL248772A0 (en) A consequence of cyclohexyl pyridine
PL3119744T3 (pl) Pochodne 2-cyjano-3-cyklopropylo-3-hydroksy-N-arylo-tioakryloamidu
GB201409138D0 (en) None
GB201400327D0 (en) None provided