ZA200901633B - Certain substituted amides, method of making, and method of use thereof - Google Patents
Certain substituted amides, method of making, and method of use thereofInfo
- Publication number
- ZA200901633B ZA200901633B ZA200901633A ZA200901633A ZA200901633B ZA 200901633 B ZA200901633 B ZA 200901633B ZA 200901633 A ZA200901633 A ZA 200901633A ZA 200901633 A ZA200901633 A ZA 200901633A ZA 200901633 B ZA200901633 B ZA 200901633B
- Authority
- ZA
- South Africa
- Prior art keywords
- making
- substituted amides
- certain substituted
- amides
- certain
- Prior art date
Links
- 150000001408 amides Chemical class 0.000 title 1
- 238000004519 manufacturing process Methods 0.000 title 1
- 238000000034 method Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/63—One oxygen atom
- C07D213/64—One oxygen atom attached in position 2 or 6
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Immunology (AREA)
- Pulmonology (AREA)
- Oncology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Epidemiology (AREA)
- Hematology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pyridine Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Steroid Compounds (AREA)
- Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
- Medicinal Preparation (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US84395906P | 2006-09-11 | 2006-09-11 |
Publications (1)
Publication Number | Publication Date |
---|---|
ZA200901633B true ZA200901633B (en) | 2009-12-30 |
Family
ID=38951317
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ZA200901633A ZA200901633B (en) | 2006-09-11 | 2009-03-06 | Certain substituted amides, method of making, and method of use thereof |
Country Status (23)
Country | Link |
---|---|
US (1) | US8058446B2 (xx) |
EP (1) | EP2081923B1 (xx) |
JP (1) | JP5295961B2 (xx) |
KR (1) | KR101442585B1 (xx) |
CN (1) | CN101679361A (xx) |
AR (1) | AR063706A1 (xx) |
AU (1) | AU2007296559B2 (xx) |
BR (1) | BRPI0716918A2 (xx) |
CA (2) | CA2941688A1 (xx) |
CL (1) | CL2007002640A1 (xx) |
CO (1) | CO6160313A2 (xx) |
CR (1) | CR10710A (xx) |
EC (1) | ECSP099239A (xx) |
ES (1) | ES2576478T3 (xx) |
IL (1) | IL197230A0 (xx) |
MA (1) | MA30782B1 (xx) |
MX (1) | MX2009002649A (xx) |
NO (1) | NO20091424L (xx) |
PE (1) | PE20080839A1 (xx) |
RU (1) | RU2009113693A (xx) |
TW (1) | TW200829579A (xx) |
WO (1) | WO2008033854A1 (xx) |
ZA (1) | ZA200901633B (xx) |
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US7838523B2 (en) * | 2006-09-11 | 2010-11-23 | Cgi Pharmaceuticals, Inc. | Certain substituted amides, method of making, and method of use thereof |
CL2008002793A1 (es) * | 2007-09-20 | 2009-09-04 | Cgi Pharmaceuticals Inc | Compuestos derivados de amidas sustituidas, inhibidores de la actividad de btk; composicion farmaceutica que los comprende; utiles en el tratamiento del cancer, trastornos oseos, enfermedades autoinmunes, entre otras |
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MX2010012848A (es) | 2008-06-03 | 2011-03-01 | Intermune Inc | Compuestos y metodos para tratar trastornos inflamatorios y fibroticos. |
UA103327C2 (xx) | 2008-06-24 | 2013-10-10 | Ф. Хоффманн-Ля Рош Аг | Заміщені піридин-2-они й піридазин-3-они$замещенные пиридин-2-оны и пиридазин-3-оны |
WO2010000633A1 (en) * | 2008-07-02 | 2010-01-07 | F. Hoffmann-La Roche Ag | Novel phenylpyrazinones as kinase inhibitors |
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KR102613433B1 (ko) | 2017-10-11 | 2023-12-13 | 주식회사 대웅제약 | 신규한 페닐피리딘 유도체 및 이를 포함하는 약학 조성물 |
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PE20081370A1 (es) * | 2006-09-11 | 2008-11-28 | Cgi Pharmaceuticals Inc | Determinadas amidas sustituidas, metodo de elaboracion y metodo de uso de las mismas |
US20100160292A1 (en) * | 2006-09-11 | 2010-06-24 | Cgi Pharmaceuticals, Inc | Kinase Inhibitors, and Methods of Using and Identifying Kinase Inhibitors |
CL2008002793A1 (es) * | 2007-09-20 | 2009-09-04 | Cgi Pharmaceuticals Inc | Compuestos derivados de amidas sustituidas, inhibidores de la actividad de btk; composicion farmaceutica que los comprende; utiles en el tratamiento del cancer, trastornos oseos, enfermedades autoinmunes, entre otras |
-
2007
- 2007-09-10 AR ARP070103988A patent/AR063706A1/es unknown
- 2007-09-10 PE PE2007001211A patent/PE20080839A1/es not_active Application Discontinuation
- 2007-09-11 KR KR1020097007477A patent/KR101442585B1/ko active IP Right Grant
- 2007-09-11 ES ES07842263.1T patent/ES2576478T3/es active Active
- 2007-09-11 US US11/853,485 patent/US8058446B2/en active Active
- 2007-09-11 RU RU2009113693/04A patent/RU2009113693A/ru not_active Application Discontinuation
- 2007-09-11 TW TW096133884A patent/TW200829579A/zh unknown
- 2007-09-11 AU AU2007296559A patent/AU2007296559B2/en not_active Ceased
- 2007-09-11 BR BRPI0716918-3A patent/BRPI0716918A2/pt not_active Application Discontinuation
- 2007-09-11 JP JP2009527625A patent/JP5295961B2/ja active Active
- 2007-09-11 CN CN200780041849A patent/CN101679361A/zh active Pending
- 2007-09-11 WO PCT/US2007/078181 patent/WO2008033854A1/en active Application Filing
- 2007-09-11 CL CL200702640A patent/CL2007002640A1/es unknown
- 2007-09-11 CA CA2941688A patent/CA2941688A1/en not_active Abandoned
- 2007-09-11 MX MX2009002649A patent/MX2009002649A/es not_active Application Discontinuation
- 2007-09-11 EP EP07842263.1A patent/EP2081923B1/en active Active
- 2007-09-11 CA CA2661654A patent/CA2661654C/en not_active Expired - Fee Related
-
2009
- 2009-02-24 IL IL197230A patent/IL197230A0/en unknown
- 2009-03-06 ZA ZA200901633A patent/ZA200901633B/xx unknown
- 2009-03-31 CO CO09033014A patent/CO6160313A2/es unknown
- 2009-04-03 CR CR10710A patent/CR10710A/es not_active Application Discontinuation
- 2009-04-06 MA MA31766A patent/MA30782B1/fr unknown
- 2009-04-07 EC EC2009009239A patent/ECSP099239A/es unknown
- 2009-04-07 NO NO20091424A patent/NO20091424L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
EP2081923B1 (en) | 2016-03-16 |
US20080139557A1 (en) | 2008-06-12 |
CL2007002640A1 (es) | 2008-06-20 |
MX2009002649A (es) | 2009-03-26 |
JP2010504287A (ja) | 2010-02-12 |
PE20080839A1 (es) | 2008-08-23 |
ECSP099239A (es) | 2009-07-31 |
IL197230A0 (en) | 2009-12-24 |
CO6160313A2 (es) | 2010-05-20 |
AU2007296559B2 (en) | 2013-01-17 |
AU2007296559A1 (en) | 2008-03-20 |
CR10710A (es) | 2009-07-14 |
NO20091424L (no) | 2009-06-10 |
KR20090074762A (ko) | 2009-07-07 |
ES2576478T3 (es) | 2016-07-07 |
AR063706A1 (es) | 2009-02-11 |
US8058446B2 (en) | 2011-11-15 |
WO2008033854A1 (en) | 2008-03-20 |
TW200829579A (en) | 2008-07-16 |
CA2661654C (en) | 2016-10-11 |
BRPI0716918A2 (pt) | 2013-11-05 |
CA2941688A1 (en) | 2008-03-20 |
KR101442585B1 (ko) | 2014-10-02 |
CA2661654A1 (en) | 2008-03-20 |
CN101679361A (zh) | 2010-03-24 |
MA30782B1 (fr) | 2009-10-01 |
EP2081923A1 (en) | 2009-07-29 |
JP5295961B2 (ja) | 2013-09-18 |
RU2009113693A (ru) | 2010-10-20 |
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