ZA200802946B - Preparation and use of tetrahydropyrrolo [3,2-c] pyridin-4-one derivatives for treatment of obesity, psychiatric and neurological disorders - Google Patents
Preparation and use of tetrahydropyrrolo [3,2-c] pyridin-4-one derivatives for treatment of obesity, psychiatric and neurological disordersInfo
- Publication number
- ZA200802946B ZA200802946B ZA200802946A ZA200802946A ZA200802946B ZA 200802946 B ZA200802946 B ZA 200802946B ZA 200802946 A ZA200802946 A ZA 200802946A ZA 200802946 A ZA200802946 A ZA 200802946A ZA 200802946 B ZA200802946 B ZA 200802946B
- Authority
- ZA
- South Africa
- Prior art keywords
- tetrahydropyrrolo
- psychiatric
- pyridin
- obesity
- derivatives
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
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US72415605P | 2005-10-06 | 2005-10-06 |
Publications (1)
Publication Number | Publication Date |
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ZA200802946B true ZA200802946B (en) | 2009-03-25 |
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Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
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ZA200802946A ZA200802946B (en) | 2005-10-06 | 2008-04-03 | Preparation and use of tetrahydropyrrolo [3,2-c] pyridin-4-one derivatives for treatment of obesity, psychiatric and neurological disorders |
Country Status (21)
Country | Link |
---|---|
US (2) | US7875626B2 (fr) |
EP (1) | EP1937679B1 (fr) |
JP (1) | JP4277062B2 (fr) |
KR (1) | KR20080058456A (fr) |
CN (1) | CN101277957A (fr) |
AR (1) | AR056560A1 (fr) |
AT (1) | ATE440099T1 (fr) |
AU (1) | AU2006298530B2 (fr) |
BR (1) | BRPI0616653A2 (fr) |
CA (1) | CA2624495A1 (fr) |
DE (1) | DE602006008641D1 (fr) |
EC (1) | ECSP088413A (fr) |
ES (1) | ES2329616T3 (fr) |
HK (1) | HK1122808A1 (fr) |
IL (1) | IL190025A0 (fr) |
NO (1) | NO20081523L (fr) |
RU (1) | RU2415856C2 (fr) |
TW (1) | TW200730525A (fr) |
UY (1) | UY29838A1 (fr) |
WO (1) | WO2007039740A2 (fr) |
ZA (1) | ZA200802946B (fr) |
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KR101273643B1 (ko) * | 2010-10-12 | 2013-06-11 | 한국화학연구원 | 5,6-디하이드로-피롤로[3,4-b]피리딘-7-온 유도체 또는 이의 약학적으로 허용 가능한 염, 이의 제조방법 및 이를 유효성분으로 포함하는 약학적 조성물 |
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FR2692575B1 (fr) | 1992-06-23 | 1995-06-30 | Sanofi Elf | Nouveaux derives du pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant. |
FR2714057B1 (fr) | 1993-12-17 | 1996-03-08 | Sanofi Elf | Nouveaux dérivés du 3-pyrazolecarboxamide, procédé pour leur préparation et compositions pharmaceutiques les contenant. |
FR2758723B1 (fr) | 1997-01-28 | 1999-04-23 | Sanofi Sa | Utilisation des antagonistes des recepteurs aux cannabinoides centraux pour la preparation de medicaments |
US6858616B2 (en) | 1998-12-23 | 2005-02-22 | Bristol-Myers Squibb Pharma Company | Nitrogen containing heterobicycles as factor Xa inhibitors |
DK1268435T3 (da) | 2000-03-23 | 2007-03-12 | Solvay Pharm Bv | 4,5-dihydro-1H-pyrazolderivater med CB1-antagonistisk aktivitet |
CA2461142A1 (fr) | 2001-09-24 | 2003-04-03 | Bayer Pharmaceuticals Corporation | Preparation et utilisation de derives de la 1,5,6,7-tetrahydropyrrolo[3,2-c]pyridine pour le traitement de l'obesite |
GB0403780D0 (en) | 2004-02-20 | 2004-03-24 | Astrazeneca Ab | Therapeutic agents |
BRPI0507786A (pt) | 2004-02-20 | 2007-07-17 | Astrazeneca Ab | composto e sais farmaceuticamente aceitáveis do mesmo, formulação farmacêutica, uso de um composto, método de tratar uma doença, e, processo para a preparação de compostos |
AU2005229459B9 (en) | 2004-04-03 | 2009-01-22 | Astrazeneca Ab | Therapeutic agents |
AR056560A1 (es) * | 2005-10-06 | 2007-10-10 | Astrazeneca Ab | Pirrolopiridinonas como moduladores cb1 |
-
2006
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- 2006-10-04 UY UY29838A patent/UY29838A1/es unknown
- 2006-10-05 KR KR1020087010582A patent/KR20080058456A/ko not_active Application Discontinuation
- 2006-10-05 CN CNA2006800365273A patent/CN101277957A/zh active Pending
- 2006-10-05 ES ES06794647T patent/ES2329616T3/es active Active
- 2006-10-05 AU AU2006298530A patent/AU2006298530B2/en not_active Ceased
- 2006-10-05 US US11/915,643 patent/US7875626B2/en not_active Expired - Fee Related
- 2006-10-05 AT AT06794647T patent/ATE440099T1/de not_active IP Right Cessation
- 2006-10-05 CA CA002624495A patent/CA2624495A1/fr not_active Abandoned
- 2006-10-05 DE DE602006008641T patent/DE602006008641D1/de active Active
- 2006-10-05 RU RU2008109185/04A patent/RU2415856C2/ru not_active IP Right Cessation
- 2006-10-05 BR BRPI0616653-9A patent/BRPI0616653A2/pt not_active IP Right Cessation
- 2006-10-05 EP EP06794647A patent/EP1937679B1/fr active Active
- 2006-10-05 JP JP2008526558A patent/JP4277062B2/ja not_active Expired - Fee Related
- 2006-10-05 TW TW095137255A patent/TW200730525A/zh unknown
- 2006-10-05 WO PCT/GB2006/003695 patent/WO2007039740A2/fr active Application Filing
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2007
- 2007-04-03 US US11/730,640 patent/US7576095B2/en not_active Expired - Fee Related
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2008
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- 2008-03-28 NO NO20081523A patent/NO20081523L/no not_active Application Discontinuation
- 2008-04-03 ZA ZA200802946A patent/ZA200802946B/xx unknown
- 2008-04-30 EC EC2008008413A patent/ECSP088413A/es unknown
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Also Published As
Publication number | Publication date |
---|---|
ECSP088413A (es) | 2008-05-30 |
RU2008109185A (ru) | 2009-11-20 |
EP1937679A2 (fr) | 2008-07-02 |
DE602006008641D1 (de) | 2009-10-01 |
WO2007039740A3 (fr) | 2007-05-31 |
US7576095B2 (en) | 2009-08-18 |
US20080312269A1 (en) | 2008-12-18 |
AU2006298530B2 (en) | 2009-10-29 |
RU2415856C2 (ru) | 2011-04-10 |
AR056560A1 (es) | 2007-10-10 |
CA2624495A1 (fr) | 2007-04-12 |
CN101277957A (zh) | 2008-10-01 |
US7875626B2 (en) | 2011-01-25 |
KR20080058456A (ko) | 2008-06-25 |
HK1122808A1 (en) | 2009-05-29 |
AU2006298530A1 (en) | 2007-04-12 |
JP4277062B2 (ja) | 2009-06-10 |
ES2329616T3 (es) | 2009-11-27 |
NO20081523L (no) | 2008-07-02 |
TW200730525A (en) | 2007-08-16 |
EP1937679B1 (fr) | 2009-08-19 |
JP2009504722A (ja) | 2009-02-05 |
UY29838A1 (es) | 2007-05-31 |
WO2007039740A2 (fr) | 2007-04-12 |
IL190025A0 (en) | 2008-08-07 |
US20080009513A1 (en) | 2008-01-10 |
BRPI0616653A2 (pt) | 2011-06-28 |
ATE440099T1 (de) | 2009-09-15 |
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