ZA200802163B - 5-(phenylisoxazolylethoxy)-triazol-3-YL substituted pyridine compounds for the treatment of neurological, psychiatric or pain disorders - Google Patents

5-(phenylisoxazolylethoxy)-triazol-3-YL substituted pyridine compounds for the treatment of neurological, psychiatric or pain disorders

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Publication number
ZA200802163B
ZA200802163B ZA200802163A ZA200802163A ZA200802163B ZA 200802163 B ZA200802163 B ZA 200802163B ZA 200802163 A ZA200802163 A ZA 200802163A ZA 200802163 A ZA200802163 A ZA 200802163A ZA 200802163 B ZA200802163 B ZA 200802163B
Authority
ZA
South Africa
Prior art keywords
phenylisoxazolylethoxy
psychiatric
triazol
neurological
treatment
Prior art date
Application number
ZA200802163A
Other languages
English (en)
Inventor
Minidis Alexander
Wensbo David
Slassi Abdelmalik
Isaac Methvin
Ericsson Caroline
Profir Veronica
Bergstrom Per-Olov
Edwards Louise
Arora Jalaj
Xin Tao
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of ZA200802163B publication Critical patent/ZA200802163B/xx

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
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  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
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  • Diabetes (AREA)
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  • Pulmonology (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Obesity (AREA)
  • Emergency Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Psychology (AREA)
  • Cardiology (AREA)
  • Virology (AREA)
  • Rheumatology (AREA)
  • Oncology (AREA)
  • Reproductive Health (AREA)
  • Molecular Biology (AREA)
  • Addiction (AREA)
  • Tropical Medicine & Parasitology (AREA)
ZA200802163A 2005-09-29 2008-03-07 5-(phenylisoxazolylethoxy)-triazol-3-YL substituted pyridine compounds for the treatment of neurological, psychiatric or pain disorders ZA200802163B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US72152705P 2005-09-29 2005-09-29

Publications (1)

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ZA200802163B true ZA200802163B (en) 2009-09-30

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ZA200802163A ZA200802163B (en) 2005-09-29 2008-03-07 5-(phenylisoxazolylethoxy)-triazol-3-YL substituted pyridine compounds for the treatment of neurological, psychiatric or pain disorders

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Country Link
US (4) US20080227824A1 (enExample)
EP (1) EP1934209A1 (enExample)
JP (2) JP2009510064A (enExample)
KR (1) KR20080050421A (enExample)
CN (1) CN101273037A (enExample)
AR (1) AR058807A1 (enExample)
AU (1) AU2006297462A1 (enExample)
BR (1) BRPI0616228A2 (enExample)
CA (1) CA2623009A1 (enExample)
EC (1) ECSP088283A (enExample)
IL (1) IL189990A0 (enExample)
NO (1) NO20081434L (enExample)
RU (1) RU2008108219A (enExample)
TW (1) TW200800976A (enExample)
UA (1) UA92503C2 (enExample)
UY (1) UY29796A1 (enExample)
WO (1) WO2007040982A1 (enExample)
ZA (1) ZA200802163B (enExample)

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US8080568B1 (en) * 2010-06-29 2011-12-20 Ewha University - Industry Collaboration Foundation 2-pyridyl substituted imidazoles as therapeutic ALK5 and/or ALK4 inhibitors
UA112418C2 (uk) * 2010-09-07 2016-09-12 Астеллас Фарма Інк. Терапевтичний болезаспокійливий засіб
CN103429583A (zh) 2010-12-08 2013-12-04 奥斯陆大学医院公司 作为wnt信号通路抑制剂的三唑衍生物
MX2013010698A (es) 2011-03-18 2014-02-17 Novartis Ag Combinaciones de activadores del receptor de acetil-colina nicotinico alfa-7 y antagonistas del receptor de glutamato metabotropico 5 (mglur5) para usarse en la discinesia inducida por dopamina en la enfermedad de parkinson.
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KR102027368B1 (ko) * 2018-05-29 2019-10-01 서울대학교산학협력단 통증의 강도를 측정하는 방법
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US7585881B2 (en) * 2004-02-18 2009-09-08 Astrazeneca Ab Additional heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists
JP5084269B2 (ja) 2004-02-18 2012-11-28 アストラゼネカ アクチボラグ テトラゾール化合物及び代謝共役型グルタミン酸受容体アンタゴニストとしてのそれらの使用
EA200601266A1 (ru) 2004-02-18 2007-02-27 Астразенека Аб Соединения триазола и их применение в качестве антагонистов метаботропного рецептора глутамата
JP2007523181A (ja) 2004-02-18 2007-08-16 アストラゼネカ アクチボラグ ポリヘテロ環式化合物、および、代謝型グルタミン酸受容体アンタゴニストとしてのそれらの使用
BRPI0507495A (pt) 2004-02-18 2007-07-10 Astrazeneca Ab composto, composição farmacêutica, uso do composto método para o tratamento de distúrbios mediados por mglur5, e, método para inibir a ativação de receptores de mglur5
KR20070026382A (ko) 2004-02-18 2007-03-08 아스트라제네카 아베 아세틸린성 피페라진 화합물 및 대사성 글루타메이트수용체 길항제로서 이들의 용도
UY29796A1 (es) * 2005-09-29 2007-04-30 Astrazeneca Ab Nuevos compuestos para el tratamiento de trastornos neurológicos, psiquiátricos o del dolor

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ECSP088283A (es) 2008-04-28
NO20081434L (no) 2008-05-19
TW200800976A (en) 2008-01-01
US20070270468A1 (en) 2007-11-22
AU2006297462A1 (en) 2007-04-12
US20070129408A1 (en) 2007-06-07
IL189990A0 (en) 2008-08-07
JP2009510064A (ja) 2009-03-12
US20070270469A1 (en) 2007-11-22
AR058807A1 (es) 2008-02-27
CA2623009A1 (en) 2007-04-12
BRPI0616228A2 (pt) 2011-06-14
US7476684B2 (en) 2009-01-13
UA92503C2 (ru) 2010-11-10
EP1934209A1 (en) 2008-06-25
JP2010013476A (ja) 2010-01-21
UY29796A1 (es) 2007-04-30
WO2007040982A1 (en) 2007-04-12
CN101273037A (zh) 2008-09-24
US20080227824A1 (en) 2008-09-18
RU2008108219A (ru) 2009-11-10

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