ZA200710817B - Benzamide derivatives and uses related thereto - Google Patents
Benzamide derivatives and uses related theretoInfo
- Publication number
- ZA200710817B ZA200710817B ZA200710817A ZA200710817A ZA200710817B ZA 200710817 B ZA200710817 B ZA 200710817B ZA 200710817 A ZA200710817 A ZA 200710817A ZA 200710817 A ZA200710817 A ZA 200710817A ZA 200710817 B ZA200710817 B ZA 200710817B
- Authority
- ZA
- South Africa
- Prior art keywords
- benzamide derivatives
- uses related
- benzamide
- derivatives
- Prior art date
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- C07C233/66—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by halogen atoms or by nitro or nitroso groups
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- C07D277/22—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D277/28—Radicals substituted by nitrogen atoms
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- C07C235/54—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton with carbon atoms of carboxamide groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring
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- C07C255/44—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring the carbon skeleton being further substituted by singly-bound nitrogen atoms, not being further bound to other hetero atoms at least one of the singly-bound nitrogen atoms being acylated
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- C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
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US7605289B2 (en) | 2005-06-17 | 2009-10-20 | Amgen, Inc. | Benzamide derivatives and uses related thereto |
PE20110235A1 (es) | 2006-05-04 | 2011-04-14 | Boehringer Ingelheim Int | Combinaciones farmaceuticas que comprenden linagliptina y metmorfina |
CA2654699A1 (en) * | 2006-06-08 | 2007-12-21 | Amgen Inc. | Benzamide derivatives and uses related thereto |
TW200808695A (en) * | 2006-06-08 | 2008-02-16 | Amgen Inc | Benzamide derivatives and uses related thereto |
EP2025674A1 (de) | 2007-08-15 | 2009-02-18 | sanofi-aventis | Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
WO2009036297A1 (en) * | 2007-09-14 | 2009-03-19 | The Trustees Of The University Of Pennsylvania | Novel compounds for treatment of malignant tumors |
JP5609150B2 (ja) * | 2009-02-27 | 2014-10-22 | アステラス製薬株式会社 | ピペリジン誘導体 |
ES2350077B1 (es) | 2009-06-04 | 2011-11-04 | Laboratorios Salvat, S.A. | Compuestos inhibidores de 11beta-hidroxiesteroide deshidrogenasa de tipo 1. |
JP2011098893A (ja) * | 2009-11-04 | 2011-05-19 | Sumitomo Chemical Co Ltd | テストステロンの生合成を抑制するための化合物の使用およびその化合物 |
WO2011107494A1 (de) | 2010-03-03 | 2011-09-09 | Sanofi | Neue aromatische glykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung |
EP2582709B1 (de) | 2010-06-18 | 2018-01-24 | Sanofi | Azolopyridin-3-on-derivate als inhibitoren von lipasen und phospholipasen |
US8530413B2 (en) | 2010-06-21 | 2013-09-10 | Sanofi | Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments |
TW201215387A (en) | 2010-07-05 | 2012-04-16 | Sanofi Aventis | Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament |
TW201215388A (en) | 2010-07-05 | 2012-04-16 | Sanofi Sa | (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments |
TW201221505A (en) | 2010-07-05 | 2012-06-01 | Sanofi Sa | Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament |
EP2766349B1 (de) | 2011-03-08 | 2016-06-01 | Sanofi | Mit carbozyklen oder heterozyklen substituierte oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung |
EP2683700B1 (de) | 2011-03-08 | 2015-02-18 | Sanofi | Tetrasubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung |
US8828994B2 (en) | 2011-03-08 | 2014-09-09 | Sanofi | Di- and tri-substituted oxathiazine derivatives, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof |
US8710050B2 (en) | 2011-03-08 | 2014-04-29 | Sanofi | Di and tri- substituted oxathiazine derivatives, method for the production, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof |
US8828995B2 (en) | 2011-03-08 | 2014-09-09 | Sanofi | Branched oxathiazine derivatives, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof |
WO2013037390A1 (en) | 2011-09-12 | 2013-03-21 | Sanofi | 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
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CN103917524B (zh) | 2011-10-18 | 2016-05-04 | 安斯泰来制药有限公司 | 双环杂环化合物 |
MX2018011177A (es) * | 2016-04-04 | 2018-11-21 | Res Triangle Inst | Agonistas de receptor de neuropéptido s (npsr). |
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PE20070137A1 (es) | 2007-04-11 |
AU2006259349B2 (en) | 2011-10-27 |
CR9667A (es) | 2008-02-11 |
AU2006259349A1 (en) | 2006-12-28 |
BRPI0612993A2 (pt) | 2010-12-14 |
EP1904435B1 (en) | 2013-01-02 |
GT200600260A (es) | 2008-01-03 |
UY29609A1 (es) | 2007-01-31 |
WO2006138508A3 (en) | 2007-02-01 |
KR20080032039A (ko) | 2008-04-14 |
US7605289B2 (en) | 2009-10-20 |
US20100069447A1 (en) | 2010-03-18 |
EP1904435A2 (en) | 2008-04-02 |
CA2611687A1 (en) | 2006-12-28 |
WO2006138508B1 (en) | 2008-06-05 |
WO2006138508A2 (en) | 2006-12-28 |
CA2611687C (en) | 2014-08-19 |
AR059942A1 (es) | 2008-05-14 |
EA200800081A1 (ru) | 2008-06-30 |
US8637576B2 (en) | 2014-01-28 |
CN101198584A (zh) | 2008-06-11 |
ES2400691T3 (es) | 2013-04-11 |
JP2008546709A (ja) | 2008-12-25 |
IL187776A0 (en) | 2008-08-07 |
NO20076134L (no) | 2008-02-29 |
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