ZA200703700B - New pyridotheinopyrimidine derivatives - Google Patents
New pyridotheinopyrimidine derivatives Download PDFInfo
- Publication number
- ZA200703700B ZA200703700B ZA200703700A ZA200703700A ZA200703700B ZA 200703700 B ZA200703700 B ZA 200703700B ZA 200703700 A ZA200703700 A ZA 200703700A ZA 200703700 A ZA200703700 A ZA 200703700A ZA 200703700 B ZA200703700 B ZA 200703700B
- Authority
- ZA
- South Africa
- Prior art keywords
- dihydro
- pyrano
- thieno
- pyrimidin
- amine
- Prior art date
Links
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- 229960003444 immunosuppressant agent Drugs 0.000 description 1
- 230000002779 inactivation Effects 0.000 description 1
- 125000003453 indazolyl group Chemical group N1N=C(C2=C1C=CC=C2)* 0.000 description 1
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- 125000004594 isoindolinyl group Chemical group C1(NCC2=CC=CC=C12)* 0.000 description 1
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Classifications
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pulmonology (AREA)
- Immunology (AREA)
- Physical Education & Sports Medicine (AREA)
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- Hospice & Palliative Care (AREA)
- Otolaryngology (AREA)
- Ophthalmology & Optometry (AREA)
- Transplantation (AREA)
- Hematology (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ES200402877A ES2259892B1 (es) | 2004-11-30 | 2004-11-30 | Nuevos derivados de piridotienopirimidina. |
Publications (1)
Publication Number | Publication Date |
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ZA200703700B true ZA200703700B (en) | 2008-07-30 |
Family
ID=35064809
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
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ZA200703700A ZA200703700B (en) | 2004-11-30 | 2007-05-08 | New pyridotheinopyrimidine derivatives |
Country Status (19)
Country | Link |
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US (1) | US20080207645A1 (es) |
EP (1) | EP1819712A1 (es) |
JP (1) | JP2008521854A (es) |
KR (1) | KR20070086652A (es) |
CN (1) | CN101068817A (es) |
AR (1) | AR052413A1 (es) |
AU (1) | AU2005311422A1 (es) |
BR (1) | BRPI0518117A (es) |
CA (1) | CA2588808A1 (es) |
ES (1) | ES2259892B1 (es) |
IL (1) | IL183141A0 (es) |
MX (1) | MX2007006172A (es) |
NO (1) | NO20073271L (es) |
PE (1) | PE20061080A1 (es) |
RU (1) | RU2007124493A (es) |
TW (1) | TW200631954A (es) |
UY (1) | UY29240A1 (es) |
WO (1) | WO2006058723A1 (es) |
ZA (1) | ZA200703700B (es) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2281251B1 (es) * | 2005-07-27 | 2008-08-16 | Laboratorios Almirall S.A. | Nuevos derivados de pirido (3',2':4,5) furo (3,2-d) pirimidina. |
WO2012131297A1 (en) | 2011-03-28 | 2012-10-04 | Jonathan Bayldon Baell | Pyrido [3',2' :4,5] thieno [3, 2-d] pyrimidin- 4 - ylamine derivatives and their therapeutical use |
JP2015512862A (ja) | 2011-12-21 | 2015-04-30 | インヴィスタ テクノロジーズ エスアエルエル | 安定なエマルジョンを減じるための抽出溶媒制御 |
CN103242276B (zh) * | 2013-05-07 | 2014-07-16 | 白银安杰利生化科技有限公司 | 2,2-二甲基四氢-2h-吡喃-4-羧酸的合成方法 |
BR112018003417B1 (pt) | 2016-06-22 | 2023-10-24 | Vanderbilt University | Composto modulador alostérico positivo do receptor muscarínico de acetilcolina m4 e composição farmacêutica que o compreende |
MA46899A (fr) | 2016-11-07 | 2021-04-14 | Univ Vanderbilt | Modulateurs allostériques positifs du récepteur muscarinique de l'acétylcholine m4 |
MA46722A (fr) | 2016-11-07 | 2019-09-11 | Univ Vanderbilt | Modulateurs allostériques positifs du récepteur muscarinique à l'acétylcholine m4 |
JP7099725B2 (ja) | 2016-11-07 | 2022-07-12 | ヴァンダービルト ユニヴァーシティ | ムスカリン性アセチルコリンレセプターm4のポジティブアロステリック調節因子 |
TW201930311A (zh) | 2017-12-05 | 2019-08-01 | 泛德比爾特大學 | 蕈毒鹼型乙醯膽鹼受體m4之正向別構調節劑 |
US11376254B2 (en) | 2017-12-05 | 2022-07-05 | Vanderbilt University | Positive allosteric modulators of the muscarinic acetylcholine receptor M4 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE19644228A1 (de) * | 1996-10-24 | 1998-04-30 | Merck Patent Gmbh | Thienopyrimidine |
DE19752952A1 (de) * | 1997-11-28 | 1999-06-02 | Merck Patent Gmbh | Thienopyrimidine |
DE19819023A1 (de) * | 1998-04-29 | 1999-11-04 | Merck Patent Gmbh | Thienopyrimidine |
KR20010105399A (ko) * | 1999-03-30 | 2001-11-28 | 쓰끼하시 다미까따 | 티에노피리미딘 화합물 및 그의 염, 및 그들의 제조 방법 |
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2004
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2005
- 2005-11-28 PE PE2005001378A patent/PE20061080A1/es not_active Application Discontinuation
- 2005-11-28 AR ARP050104957A patent/AR052413A1/es unknown
- 2005-11-29 UY UY29240A patent/UY29240A1/es unknown
- 2005-11-30 WO PCT/EP2005/012773 patent/WO2006058723A1/en active Application Filing
- 2005-11-30 CA CA002588808A patent/CA2588808A1/en not_active Abandoned
- 2005-11-30 EP EP05813317A patent/EP1819712A1/en not_active Withdrawn
- 2005-11-30 US US11/791,451 patent/US20080207645A1/en not_active Abandoned
- 2005-11-30 MX MX2007006172A patent/MX2007006172A/es not_active Application Discontinuation
- 2005-11-30 TW TW094142174A patent/TW200631954A/zh unknown
- 2005-11-30 AU AU2005311422A patent/AU2005311422A1/en not_active Abandoned
- 2005-11-30 RU RU2007124493/04A patent/RU2007124493A/ru not_active Application Discontinuation
- 2005-11-30 CN CNA2005800409703A patent/CN101068817A/zh active Pending
- 2005-11-30 BR BRPI0518117-8A patent/BRPI0518117A/pt not_active IP Right Cessation
- 2005-11-30 KR KR1020077014496A patent/KR20070086652A/ko not_active Application Discontinuation
- 2005-11-30 JP JP2007543766A patent/JP2008521854A/ja active Pending
-
2007
- 2007-05-08 ZA ZA200703700A patent/ZA200703700B/en unknown
- 2007-05-10 IL IL183141A patent/IL183141A0/en unknown
- 2007-06-26 NO NO20073271A patent/NO20073271L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
CN101068817A (zh) | 2007-11-07 |
PE20061080A1 (es) | 2006-11-10 |
ES2259892A1 (es) | 2006-10-16 |
MX2007006172A (es) | 2007-07-13 |
NO20073271L (no) | 2007-06-26 |
RU2007124493A (ru) | 2009-01-10 |
KR20070086652A (ko) | 2007-08-27 |
WO2006058723A8 (en) | 2007-07-12 |
WO2006058723A1 (en) | 2006-06-08 |
AR052413A1 (es) | 2007-03-21 |
TW200631954A (en) | 2006-09-16 |
ES2259892B1 (es) | 2007-11-01 |
IL183141A0 (en) | 2007-09-20 |
UY29240A1 (es) | 2006-02-24 |
US20080207645A1 (en) | 2008-08-28 |
EP1819712A1 (en) | 2007-08-22 |
CA2588808A1 (en) | 2006-06-08 |
JP2008521854A (ja) | 2008-06-26 |
BRPI0518117A (pt) | 2008-11-04 |
AU2005311422A1 (en) | 2006-06-08 |
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