ZA200606636B - Therapeutic combinations of atypical antipsychotic with corticotropin releasing factor antagonists - Google Patents

Therapeutic combinations of atypical antipsychotic with corticotropin releasing factor antagonists Download PDF

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Publication number
ZA200606636B
ZA200606636B ZA200606636A ZA200606636A ZA200606636B ZA 200606636 B ZA200606636 B ZA 200606636B ZA 200606636 A ZA200606636 A ZA 200606636A ZA 200606636 A ZA200606636 A ZA 200606636A ZA 200606636 B ZA200606636 B ZA 200606636B
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ZA
South Africa
Prior art keywords
alkyl
methyl
ethyl
dimethyl
phenyl
Prior art date
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ZA200606636A
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English (en)
Inventor
Romano Steven Joseph
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Pfizer Prod Inc
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Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of ZA200606636B publication Critical patent/ZA200606636B/en

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
    • A—HUMAN NECESSITIES
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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    • A—HUMAN NECESSITIES
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    • A61K31/47—Quinolines; Isoquinolines
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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    • A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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    • A61P25/24—Antidepressants

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  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
ZA200606636A 2004-02-13 2006-08-10 Therapeutic combinations of atypical antipsychotic with corticotropin releasing factor antagonists ZA200606636B (en)

Applications Claiming Priority (1)

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US54473104P 2004-02-13 2004-02-13

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ZA200606636B true ZA200606636B (en) 2008-01-30

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ZA200606636A ZA200606636B (en) 2004-02-13 2006-08-10 Therapeutic combinations of atypical antipsychotic with corticotropin releasing factor antagonists

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US (1) US20050209250A1 (enExample)
EP (1) EP1718311A1 (enExample)
JP (1) JP2007522200A (enExample)
KR (1) KR20060110006A (enExample)
CN (1) CN1917882A (enExample)
AU (1) AU2005215257A1 (enExample)
BR (1) BRPI0507609A (enExample)
CA (1) CA2556160A1 (enExample)
IL (1) IL177433A0 (enExample)
NO (1) NO20064054L (enExample)
RU (1) RU2006129307A (enExample)
TW (1) TW200538128A (enExample)
WO (1) WO2005079807A1 (enExample)
ZA (1) ZA200606636B (enExample)

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IL177433A0 (en) 2006-12-10
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TW200538128A (en) 2005-12-01
AU2005215257A1 (en) 2005-09-01
JP2007522200A (ja) 2007-08-09
US20050209250A1 (en) 2005-09-22
CN1917882A (zh) 2007-02-21
WO2005079807A1 (en) 2005-09-01
KR20060110006A (ko) 2006-10-23

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