CN1917882A - 非典型抗精神病药物与促肾上腺皮质激素释放因子拮抗剂的治疗剂组合 - Google Patents
非典型抗精神病药物与促肾上腺皮质激素释放因子拮抗剂的治疗剂组合 Download PDFInfo
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- CN1917882A CN1917882A CNA2005800049430A CN200580004943A CN1917882A CN 1917882 A CN1917882 A CN 1917882A CN A2005800049430 A CNA2005800049430 A CN A2005800049430A CN 200580004943 A CN200580004943 A CN 200580004943A CN 1917882 A CN1917882 A CN 1917882A
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- alkyl
- methyl
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
- A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
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- A61K31/4164—1,3-Diazoles
- A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
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- Health & Medical Sciences (AREA)
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- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Psychiatry (AREA)
- Anesthesiology (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US54473104P | 2004-02-13 | 2004-02-13 | |
| US60/544,731 | 2004-02-13 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CN1917882A true CN1917882A (zh) | 2007-02-21 |
Family
ID=34886075
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CNA2005800049430A Pending CN1917882A (zh) | 2004-02-13 | 2005-02-01 | 非典型抗精神病药物与促肾上腺皮质激素释放因子拮抗剂的治疗剂组合 |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US20050209250A1 (enExample) |
| EP (1) | EP1718311A1 (enExample) |
| JP (1) | JP2007522200A (enExample) |
| KR (1) | KR20060110006A (enExample) |
| CN (1) | CN1917882A (enExample) |
| AU (1) | AU2005215257A1 (enExample) |
| BR (1) | BRPI0507609A (enExample) |
| CA (1) | CA2556160A1 (enExample) |
| IL (1) | IL177433A0 (enExample) |
| NO (1) | NO20064054L (enExample) |
| RU (1) | RU2006129307A (enExample) |
| TW (1) | TW200538128A (enExample) |
| WO (1) | WO2005079807A1 (enExample) |
| ZA (1) | ZA200606636B (enExample) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI568448B (zh) * | 2010-01-07 | 2017-02-01 | 阿艾克麥斯製藥愛爾蘭有限公司 | 四級銨鹽前藥 |
Families Citing this family (32)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20050171088A1 (en) * | 2004-01-30 | 2005-08-04 | Astrazeneca Ab | Treatment of psychoses with dibenzothiazepine antipsychotic |
| EP2170399A1 (en) * | 2007-06-05 | 2010-04-07 | Synthon B.V. | Intranasal administration of asenapine and pharmaceutical compositions therefor |
| CN101945869B (zh) * | 2007-12-19 | 2014-06-18 | 癌症研究技术有限公司 | 吡啶并[2,3-b]吡嗪-8-取代化合物及其用途 |
| US20100298397A1 (en) * | 2009-05-19 | 2010-11-25 | Singh Nikhilesh N | Method of treatment of obsessive compulsive disorder with ondansetron |
| EP2445343B1 (en) | 2009-06-25 | 2021-08-04 | Alkermes Pharma Ireland Limited | Prodrugs of nh-acidic compounds |
| HUE033442T2 (en) | 2009-06-25 | 2017-11-28 | Alkermes Pharma Ireland Ltd | Heterocyclic compounds for the treatment of neurological and psychological disorders |
| EP2521545B1 (en) | 2010-01-07 | 2019-11-27 | Alkermes Pharma Ireland Limited | Prodrugs of heteroaromatic compounds |
| WO2011084849A1 (en) * | 2010-01-07 | 2011-07-14 | Alkermes, Inc. | Diaryldiazepine prodrugs for the treatment of neurological and psychological disorders |
| JP5848761B2 (ja) | 2010-06-24 | 2016-01-27 | アルカーメス ファーマ アイルランド リミテッド | Nh酸性化合物のプロドラッグ:エステル、カルボネート、カルバメートおよびホスホネートの誘導体 |
| US20120302616A1 (en) * | 2010-12-03 | 2012-11-29 | Nikhilesh Singh | Method of treatment of obsessive compulsive disorder with ondansetron |
| EP3156056B1 (en) | 2011-03-18 | 2023-12-06 | Alkermes Pharma Ireland Limited | Pharmaceutical compositions comprising sorbitan esters |
| JP5952912B2 (ja) | 2011-12-15 | 2016-07-13 | アルカーメス ファーマ アイルランド リミテッド | 二級アミン化合物のプロドラッグ |
| AU2013235523B9 (en) | 2012-03-19 | 2018-01-04 | Alkermes Pharma Ireland Limited | Pharmaceutical compositions comprising glycerol esters |
| AU2013235526B2 (en) | 2012-03-19 | 2017-11-30 | Alkermes Pharma Ireland Limited | Pharmaceutical compositions comprising benzyl alcohol |
| CA2867121C (en) | 2012-03-19 | 2021-05-25 | Alkermes Pharma Ireland Limited | Pharmaceutical compositions comprising fatty acid esters |
| ES2792149T3 (es) | 2012-09-19 | 2020-11-10 | Alkermes Pharma Ireland Ltd | Composiciones farmacéuticas que tienen estabilidad de almacenamiento mejorada |
| JP6440625B2 (ja) | 2012-11-14 | 2018-12-19 | ザ・ジョンズ・ホプキンス・ユニバーシティー | 精神分裂病を処置するための方法および組成物 |
| CN106102740A (zh) | 2014-01-21 | 2016-11-09 | 纽罗克里生物科学有限公司 | 治疗先天性肾上腺增生的crf1受体拮抗剂 |
| AU2015231278B2 (en) | 2014-03-20 | 2020-01-23 | Alkermes Pharma Ireland Limited | Aripiprazole formulations having increased injection speeds |
| US11077108B2 (en) * | 2016-09-07 | 2021-08-03 | The Regents Of The University Of California | Allosteric corticotropin-releasing factor receptor 1 (CRFR1) antagonists that decrease p-tau and improve cognition |
| EP3338768B1 (en) | 2016-12-20 | 2019-10-30 | LTS Lohmann Therapie-Systeme AG | Transdermal therapeutic system containing asenapine |
| KR102614709B1 (ko) | 2016-12-20 | 2023-12-18 | 에르테에스 로만 테라피-시스테메 아게 | 아세나핀 및 폴리실록산 또는 폴리이소부틸렌을 함유하는 경피흡수 치료 시스템 |
| US11033512B2 (en) | 2017-06-26 | 2021-06-15 | Lts Lohmann Therapie-Systeme Ag | Transdermal therapeutic system containing asenapine and silicone acrylic hybrid polymer |
| WO2019032720A1 (en) | 2017-08-09 | 2019-02-14 | Sanford Burnham Prebys Medical Discovery Institute | APELIN RECEPTOR AGONISTS AND METHODS OF USE |
| WO2019036503A1 (en) | 2017-08-14 | 2019-02-21 | Spruce Biosciences, Inc. | CORTICOTROPIN RELEASE FACTOR RECEPTOR ANTAGONISTS |
| CA3092335A1 (en) | 2018-03-05 | 2019-09-12 | Alkermes Pharma Ireland Limited | Aripiprazole dosing strategy |
| US12329862B2 (en) | 2018-06-20 | 2025-06-17 | Lts Lohmann Therapie-Systeme Ag | Transdermal therapeutic system containing asenapine |
| AU2019291060B2 (en) | 2018-06-20 | 2024-09-05 | Lts Lohmann Therapie-Systeme Ag | Transdermal therapeutic system containing asenapine |
| EP3984523B1 (en) | 2018-12-07 | 2025-09-03 | Neurocrine Biosciences, Inc. | Crf1 receptor antagonist, pharmaceutical formulations and solid forms thereof for the treatment of congenital adrenal hyperplasia |
| WO2021062246A1 (en) | 2019-09-27 | 2021-04-01 | Neurocrine Biosciences, Inc. | Crf receptor antagonists and methods of use |
| EP4175572A4 (en) | 2020-08-12 | 2024-03-27 | Spruce Biosciences, Inc. | Methods and compositions for treating polycystic ovary syndrome |
| US20250276066A1 (en) * | 2021-02-10 | 2025-09-04 | Gero Pte. Ltd. | Methods, compositions and compounds for treating age-related diseases and conditions |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL7605526A (nl) * | 1976-05-24 | 1977-11-28 | Akzo Nv | Nieuwe tetracyclische derivaten. |
| TW574214B (en) * | 1994-06-08 | 2004-02-01 | Pfizer | Corticotropin releasing factor antagonists |
| TW477787B (en) * | 1996-08-27 | 2002-03-01 | Pfizer | Pyrido six-membered nitrogen-containing cyclic ring derivatives having corticotropin releasing factor antagonist activity and pharmaceutical composition containing same |
| IL127497A (en) * | 1997-12-18 | 2002-07-25 | Pfizer Prod Inc | Medicinal products containing piperazinyl-heterocyclic compounds for the treatment of psychiatric disorders |
| EP1040831A3 (en) * | 1999-04-02 | 2003-05-02 | Pfizer Products Inc. | Use of corticotropin releasing factor (CRF) antagonists to prevent sudden death |
| US6432989B1 (en) * | 1999-08-27 | 2002-08-13 | Pfizer Inc | Use of CRF antagonists to treat circadian rhythm disorders |
-
2005
- 2005-02-01 WO PCT/IB2005/000251 patent/WO2005079807A1/en not_active Ceased
- 2005-02-01 RU RU2006129307/15A patent/RU2006129307A/ru not_active Application Discontinuation
- 2005-02-01 KR KR1020067018643A patent/KR20060110006A/ko not_active Ceased
- 2005-02-01 AU AU2005215257A patent/AU2005215257A1/en not_active Abandoned
- 2005-02-01 CA CA002556160A patent/CA2556160A1/en not_active Abandoned
- 2005-02-01 BR BRPI0507609-9A patent/BRPI0507609A/pt not_active IP Right Cessation
- 2005-02-01 JP JP2006552710A patent/JP2007522200A/ja active Pending
- 2005-02-01 CN CNA2005800049430A patent/CN1917882A/zh active Pending
- 2005-02-01 EP EP05702400A patent/EP1718311A1/en not_active Withdrawn
- 2005-02-05 TW TW094103864A patent/TW200538128A/zh unknown
- 2005-02-14 US US11/058,329 patent/US20050209250A1/en not_active Abandoned
-
2006
- 2006-08-10 ZA ZA200606636A patent/ZA200606636B/en unknown
- 2006-08-10 IL IL177433A patent/IL177433A0/en unknown
- 2006-09-08 NO NO20064054A patent/NO20064054L/no not_active Application Discontinuation
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI568448B (zh) * | 2010-01-07 | 2017-02-01 | 阿艾克麥斯製藥愛爾蘭有限公司 | 四級銨鹽前藥 |
Also Published As
| Publication number | Publication date |
|---|---|
| CA2556160A1 (en) | 2005-09-01 |
| BRPI0507609A (pt) | 2007-07-03 |
| EP1718311A1 (en) | 2006-11-08 |
| NO20064054L (no) | 2006-11-10 |
| ZA200606636B (en) | 2008-01-30 |
| IL177433A0 (en) | 2006-12-10 |
| RU2006129307A (ru) | 2008-02-20 |
| TW200538128A (en) | 2005-12-01 |
| AU2005215257A1 (en) | 2005-09-01 |
| JP2007522200A (ja) | 2007-08-09 |
| US20050209250A1 (en) | 2005-09-22 |
| WO2005079807A1 (en) | 2005-09-01 |
| KR20060110006A (ko) | 2006-10-23 |
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