ZA200606315B - Novel amido-substituted hydroxy-6-phenylphenanthridines - Google Patents

Novel amido-substituted hydroxy-6-phenylphenanthridines

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Publication number
ZA200606315B
ZA200606315B ZA200606315A ZA200606315A ZA200606315B ZA 200606315 B ZA200606315 B ZA 200606315B ZA 200606315 A ZA200606315 A ZA 200606315A ZA 200606315 A ZA200606315 A ZA 200606315A ZA 200606315 B ZA200606315 B ZA 200606315B
Authority
ZA
South Africa
Prior art keywords
phenylphenanthridines
substituted hydroxy
novel amido
amido
novel
Prior art date
Application number
ZA200606315A
Other languages
English (en)
Inventor
Maier Thomas
Beckers Thomas
Baer Thomas
Gimmnich Petra
Dullweber Frank
Vennemann Matthias
Original Assignee
Altana Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Altana Pharma Ag filed Critical Altana Pharma Ag
Publication of ZA200606315B publication Critical patent/ZA200606315B/xx

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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4025Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
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    • C07D207/46Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with hetero atoms directly attached to the ring nitrogen atom
    • C07D207/48Sulfur atoms
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    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07DHETEROCYCLIC COMPOUNDS
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    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

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ZA200606315A 2004-03-11 2006-07-31 Novel amido-substituted hydroxy-6-phenylphenanthridines ZA200606315B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP04101003 2004-03-11

Publications (1)

Publication Number Publication Date
ZA200606315B true ZA200606315B (en) 2008-02-27

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US (5) US7842820B2 (ru)
EP (2) EP1725528B1 (ru)
JP (1) JP4856623B2 (ru)
KR (1) KR101130556B1 (ru)
CN (1) CN1926103B (ru)
AR (1) AR048427A1 (ru)
AU (1) AU2005221834B2 (ru)
BR (1) BRPI0508464B8 (ru)
CA (1) CA2558552C (ru)
CY (1) CY1114284T1 (ru)
DK (1) DK1725528T3 (ru)
EA (1) EA012451B1 (ru)
ES (1) ES2430371T3 (ru)
HK (1) HK1102583A1 (ru)
HR (1) HRP20130810T1 (ru)
IL (1) IL177168A (ru)
ME (1) ME02122B (ru)
NO (1) NO337457B1 (ru)
NZ (1) NZ549251A (ru)
PL (1) PL1725528T3 (ru)
PT (1) PT1725528E (ru)
RS (1) RS52937B (ru)
SI (1) SI1725528T1 (ru)
TW (1) TWI353977B (ru)
WO (1) WO2005087724A2 (ru)
ZA (1) ZA200606315B (ru)

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EP1868994B1 (en) 2005-04-07 2011-05-25 4Sc Ag Sulfonylpyrroles as histone deacetylase inhibitors
EP1928872B1 (en) 2005-09-21 2012-03-14 4Sc Ag Novel sulphonylpyrroles as inhibitors of hdac
CN101287706A (zh) * 2005-09-21 2008-10-15 尼科梅德有限责任公司 作为组蛋白脱乙酰基酶抑制剂的磺酰基吡咯盐酸盐
EP2060565A1 (en) * 2007-11-16 2009-05-20 4Sc Ag Novel bifunctional compounds which inhibit protein kinases and histone deacetylases
EP2100882A1 (en) * 2008-03-12 2009-09-16 4Sc Ag (E) -N -(2-Amino-phenyl) -3-{1-[4-(1-methyl-1H-pyrazol-4-yl)- benzenesulfonyl]-1H-pyrrol-3-yl} -acrylamide salts

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