EA200601587A1 - Новые амидозамещённые гидрокси-6-фенилфенантридины - Google Patents

Новые амидозамещённые гидрокси-6-фенилфенантридины

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Publication number
EA200601587A1
EA200601587A1 EA200601587A EA200601587A EA200601587A1 EA 200601587 A1 EA200601587 A1 EA 200601587A1 EA 200601587 A EA200601587 A EA 200601587A EA 200601587 A EA200601587 A EA 200601587A EA 200601587 A1 EA200601587 A1 EA 200601587A1
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EA
Eurasian Patent Office
Prior art keywords
phenylphenanthridine
substituted hydroxy
new amido
new
amido
Prior art date
Application number
EA200601587A
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English (en)
Other versions
EA012451B1 (ru
Inventor
Томас Майер
Томас Беккерс
Томас Баер
Петра Гиммних
Франк Дулльвебер
Маттиас Феннеманн
Original Assignee
Алтана Фарма Аг
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Publication date
Application filed by Алтана Фарма Аг filed Critical Алтана Фарма Аг
Publication of EA200601587A1 publication Critical patent/EA200601587A1/ru
Publication of EA012451B1 publication Critical patent/EA012451B1/ru

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    • A61K31/4025—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
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Abstract

В заявке описаны соединения формулы I, в которой R1, R2, R3, R4, R5, R6 и R7 имеют значения, указанные в описании, являющиеся новыми эффективными HDAC ингибиторами.
EA200601587A 2004-03-11 2005-03-10 Новые амидозамещённые гидрокси-6-фенилфенантридины EA012451B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP04101003 2004-03-11
PCT/EP2005/051086 WO2005087724A2 (en) 2004-03-11 2005-03-10 Sulphonylpyrroles as hdac inhibitors

Publications (2)

Publication Number Publication Date
EA200601587A1 true EA200601587A1 (ru) 2007-04-27
EA012451B1 EA012451B1 (ru) 2009-10-30

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EA200601587A EA012451B1 (ru) 2004-03-11 2005-03-10 Новые амидозамещённые гидрокси-6-фенилфенантридины

Country Status (26)

Country Link
US (5) US7842820B2 (ru)
EP (2) EP1725528B1 (ru)
JP (1) JP4856623B2 (ru)
KR (1) KR101130556B1 (ru)
CN (1) CN1926103B (ru)
AR (1) AR048427A1 (ru)
AU (1) AU2005221834B2 (ru)
BR (1) BRPI0508464B8 (ru)
CA (1) CA2558552C (ru)
CY (1) CY1114284T1 (ru)
DK (1) DK1725528T3 (ru)
EA (1) EA012451B1 (ru)
ES (1) ES2430371T3 (ru)
HK (1) HK1102583A1 (ru)
HR (1) HRP20130810T1 (ru)
IL (1) IL177168A (ru)
ME (1) ME02122B (ru)
NO (1) NO337457B1 (ru)
NZ (1) NZ549251A (ru)
PL (1) PL1725528T3 (ru)
PT (1) PT1725528E (ru)
RS (1) RS52937B (ru)
SI (1) SI1725528T1 (ru)
TW (1) TWI353977B (ru)
WO (1) WO2005087724A2 (ru)
ZA (1) ZA200606315B (ru)

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