ZA200603280B - Method of inhibiting remnant lipoprotein production - Google Patents

Method of inhibiting remnant lipoprotein production

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Publication number
ZA200603280B
ZA200603280B ZA200603280A ZA200603280A ZA200603280B ZA 200603280 B ZA200603280 B ZA 200603280B ZA 200603280 A ZA200603280 A ZA 200603280A ZA 200603280 A ZA200603280 A ZA 200603280A ZA 200603280 B ZA200603280 B ZA 200603280B
Authority
ZA
South Africa
Prior art keywords
remnant lipoprotein
lipoprotein production
inhibiting remnant
inhibiting
production
Prior art date
Application number
ZA200603280A
Other languages
English (en)
Inventor
Hiroshi Okamoto
Noboru Furukawa
Tomohiko Sasase
Original Assignee
Japan Tobacco Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Japan Tobacco Inc filed Critical Japan Tobacco Inc
Publication of ZA200603280B publication Critical patent/ZA200603280B/xx

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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/255Esters, e.g. nitroglycerine, selenocyanates of sulfoxy acids or sulfur analogues thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • AHUMAN NECESSITIES
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/16Amides, e.g. hydroxamic acids
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    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • AHUMAN NECESSITIES
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
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    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/196Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
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    • A61K31/4402Non condensed pyridines; Hydrogenated derivatives thereof only substituted in position 2, e.g. pheniramine, bisacodyl
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    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
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    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Emergency Medicine (AREA)
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  • Hematology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Obesity (AREA)
  • Vascular Medicine (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Steroid Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
ZA200603280A 2003-09-26 2006-04-25 Method of inhibiting remnant lipoprotein production ZA200603280B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2003373453 2003-09-26

Publications (1)

Publication Number Publication Date
ZA200603280B true ZA200603280B (en) 2010-05-26

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Application Number Title Priority Date Filing Date
ZA200806375A ZA200806375B (en) 2003-09-26 2006-04-25 Method of inhibiting remnant lipoprotein production
ZA200603280A ZA200603280B (en) 2003-09-26 2006-04-25 Method of inhibiting remnant lipoprotein production

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Application Number Title Priority Date Filing Date
ZA200806375A ZA200806375B (en) 2003-09-26 2006-04-25 Method of inhibiting remnant lipoprotein production

Country Status (17)

Country Link
US (3) US20070054839A1 (de)
EP (3) EP2319509A1 (de)
JP (2) JP4536061B2 (de)
KR (2) KR20070087197A (de)
CN (3) CN1886124A (de)
AU (1) AU2004275637C1 (de)
BR (1) BRPI0414822A (de)
CA (1) CA2554982A1 (de)
CO (1) CO5690566A2 (de)
IL (2) IL174310A (de)
MX (1) MXPA06003357A (de)
NO (1) NO20061818L (de)
NZ (2) NZ546732A (de)
RU (1) RU2330682C2 (de)
SG (1) SG146695A1 (de)
WO (1) WO2005030185A2 (de)
ZA (2) ZA200806375B (de)

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JP6140168B2 (ja) 2011-09-27 2017-05-31 ドクター レディズ ラボラトリーズ リミテッド アテローム性動脈硬化症の処置のために有用なコレステリルエステル転送タンパク質(cetp)インヒビターとしての5−ベンジルアミノメチル−6−アミノピラゾロ[3,4−b]ピリジン誘導体
WO2014017569A1 (ja) * 2012-07-26 2014-01-30 興和株式会社 血中ldlを低下させるための医薬
PT2978859T (pt) 2013-03-27 2018-10-04 Hoffmann La Roche Marcadores genéticos para previsão da capacidade de resposta à terapêutica
WO2014165827A1 (en) 2013-04-05 2014-10-09 Salk Institute For Biological Studies Ppar agonists
RU2703192C2 (ru) 2014-07-30 2019-10-15 Ф. Хоффманн-Ля Рош Аг Генетические маркеры для прогнозирования ответа на терапию поднимающими уровень hdl или имитирующими hdl агентами
CN113004205B (zh) 2015-10-07 2024-07-02 米托布里奇公司 Ppar激动剂、化合物、药物组合物及其使用方法
ES2861503T3 (es) 2016-04-13 2021-10-06 Mitobridge Inc Agonistas de PPAR, compuestos, composiciones farmacéuticas y métodos de uso de los mismos

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IL193771A (en) 2013-09-30
EP1670446A2 (de) 2006-06-21
AU2004275637B2 (en) 2008-07-17
JP5214638B2 (ja) 2013-06-19
KR20060080214A (ko) 2006-07-07
US20110189210A1 (en) 2011-08-04
CN103330703A (zh) 2013-10-02
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JP4536061B2 (ja) 2010-09-01
WO2005030185A2 (en) 2005-04-07
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WO2005030185A3 (en) 2005-08-11
CN1886124A (zh) 2006-12-27
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