ZA200500019B - Inhalation medicaments containing a novel anticholinesterase drug in conjunction with corticosteroid and betamimetic drugs - Google Patents
Inhalation medicaments containing a novel anticholinesterase drug in conjunction with corticosteroid and betamimetic drugs Download PDFInfo
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- ZA200500019B ZA200500019B ZA200500019A ZA200500019A ZA200500019B ZA 200500019 B ZA200500019 B ZA 200500019B ZA 200500019 A ZA200500019 A ZA 200500019A ZA 200500019 A ZA200500019 A ZA 200500019A ZA 200500019 B ZA200500019 B ZA 200500019B
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- ZA
- South Africa
- Prior art keywords
- hydroxy
- composition according
- pharmaceutical composition
- methyl
- propellant
- Prior art date
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- 239000003814 drug Substances 0.000 title claims abstract description 7
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- 239000000544 cholinesterase inhibitor Substances 0.000 title 1
- 239000000203 mixture Substances 0.000 claims abstract description 44
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- 150000004677 hydrates Chemical class 0.000 claims abstract description 8
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- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
- A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/46—8-Azabicyclo [3.2.1] octane; Derivatives thereof, e.g. atropine, cocaine
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
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- A—HUMAN NECESSITIES
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- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
Landscapes
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- Medicinal Chemistry (AREA)
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- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Steroid Compounds (AREA)
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Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10237739A DE10237739A1 (de) | 2002-08-17 | 2002-08-17 | Inhalative Arzneimittel enthaltend ein neues Anticholinergikum in Kombination mit Corticosteroiden und Betamimetika |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200500019B true ZA200500019B (en) | 2006-07-26 |
Family
ID=30775387
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200500019A ZA200500019B (en) | 2002-08-17 | 2005-01-03 | Inhalation medicaments containing a novel anticholinesterase drug in conjunction with corticosteroid and betamimetic drugs |
Country Status (21)
| Country | Link |
|---|---|
| EP (2) | EP1785136A3 (ko) |
| JP (1) | JP2006501253A (ko) |
| KR (1) | KR101083977B1 (ko) |
| CN (1) | CN1688308A (ko) |
| AT (1) | ATE366574T1 (ko) |
| AU (1) | AU2003255289B2 (ko) |
| BR (1) | BR0313526A (ko) |
| CA (1) | CA2495454C (ko) |
| CO (1) | CO5540380A2 (ko) |
| CY (1) | CY1107742T1 (ko) |
| DE (2) | DE10237739A1 (ko) |
| DK (1) | DK1530471T3 (ko) |
| ES (1) | ES2290549T3 (ko) |
| IL (1) | IL166891A (ko) |
| MX (1) | MXPA05001823A (ko) |
| NZ (1) | NZ538834A (ko) |
| PL (1) | PL212070B1 (ko) |
| PT (1) | PT1530471E (ko) |
| RU (1) | RU2332217C2 (ko) |
| WO (1) | WO2004022058A1 (ko) |
| ZA (1) | ZA200500019B (ko) |
Families Citing this family (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU7576001A (en) | 2000-08-05 | 2002-02-18 | Glaxo Group Ltd | 6.alpha., 9.alpha.-difluoro-17.alpha.-`(2-furanylcarboxyl) oxy]-11.beta.-hydroxy-16.alpha.-methyl-3-oxo-androst-1,4,-diene-17-carbothioic acid s-fluoromethyl ester as an anti-inflammatory agent |
| EP1383786B1 (en) | 2001-04-30 | 2008-10-15 | Glaxo Group Limited | Anti-inflammatory 17.beta.-carbothioate ester derivatives of androstane with a cyclic ester group in position 17.alpha |
| US7056916B2 (en) | 2002-11-15 | 2006-06-06 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Medicaments for the treatment of chronic obstructive pulmonary disease |
| US7220742B2 (en) | 2004-05-14 | 2007-05-22 | Boehringer Ingelheim International Gmbh | Enantiomerically pure beta agonists, process for the manufacture thereof and use thereof as medicaments |
| DE102004024453A1 (de) * | 2004-05-14 | 2006-01-05 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Neue langwirksame Bronchodilatoren zur Behandlung von Atemwegserkrankungen |
| US7745621B2 (en) | 2004-05-14 | 2010-06-29 | Boehringer Ingelheim International Gmbh | Long acting bronchodilators for the treatment of respiratory diseases |
| US20060034776A1 (en) * | 2004-08-10 | 2006-02-16 | Boehringer Ingelheim International Gmbh | Inhalable medicaments containing a new anticholinergic, corticosteroids, and betamimetics |
| DE102004056578A1 (de) * | 2004-11-23 | 2006-05-24 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Inhalative Arzneimittel enthaltend ein neues Anticholinergikum, Formoterol und ein Steroid |
| DE102004056579A1 (de) * | 2004-11-23 | 2006-05-24 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Inhalative Arzneimittel enthaltend ein neues Anticholinergikum, Salmeterol und ein Steroid |
| SG159550A1 (en) | 2005-02-25 | 2010-03-30 | Chiesi Farma Spa | Pharmaceutical aerosol formulations for pressurized metered dose inhalers comprising a sequestering agent |
| CA2603433A1 (en) * | 2005-03-30 | 2006-10-05 | Schering Corporation | Medicaments and methods combining an anticholinergic, a corticosteroid, and a long acting beta agonist |
| WO2006114379A1 (de) * | 2005-04-23 | 2006-11-02 | Boehringer Ingelheim International Gmbh | Arzneimittelkombination für die inhalation enthaltend neben einem anticholinergikum ein betamimetikum und ein steroid |
| ES2530991T3 (es) | 2005-08-15 | 2015-03-09 | Boehringer Ingelheim Int | Procedimiento para la obtención de betamiméticos |
| CA2701956A1 (en) * | 2007-10-25 | 2009-04-30 | Merck Frosst Canada Ltd. | Combination therapy |
| US8815258B2 (en) | 2009-05-29 | 2014-08-26 | Pearl Therapeutics, Inc. | Compositions, methods and systems for respiratory delivery of two or more active agents |
| PL3106149T3 (pl) | 2009-05-29 | 2020-06-01 | Pearl Therapeutics, Inc. | Kompozycje do płucnego dostarczania długo-działających antagonistów muskarynowych i długo-działających agonistów receptora beta-2 adrenergicznego oraz powiązane sposoby i układy |
| RU2479304C1 (ru) * | 2012-05-29 | 2013-04-20 | Шолекс Девелопмент Гмбх, | Стабильный раствор фенотерола гидробромида |
| RU2504382C1 (ru) * | 2012-06-13 | 2014-01-20 | Шолекс Девелопмент Гмбх | Ингаляционный препарат для лечения бронхиальной астмы и хронической обструктивной болезни легких и способ его получения |
| WO2014096115A1 (en) | 2012-12-21 | 2014-06-26 | Boehringer Ingelheim Vetmedica Gmbh | Ciclesonide for the treatment of airway disease in horses |
| LT3473255T (lt) | 2012-12-21 | 2022-03-10 | Boehringer Ingelheim Vetmedica Gmbh | Farmacinė vaisto forma, apimanti ciklezonidą |
| JP6454323B2 (ja) | 2013-03-15 | 2019-01-16 | パール セラピューティクス，インコーポレイテッド | 粒子状結晶性材料のコンディショニングのための方法及びシステム |
| WO2015065223A1 (ru) * | 2013-10-28 | 2015-05-07 | Шолекс Девелопмент Гмбх | Стабильный раствор фенотерола гидробромида |
| WO2015065220A1 (ru) * | 2013-10-28 | 2015-05-07 | Шолекс Девелопмент Гмбх | Ингаляционный препарат для лечения бронхиальной астмы и хронической обструктивной болезни легких и способ его получения |
| PL3157522T3 (pl) * | 2014-06-18 | 2020-03-31 | Boehringer Ingelheim Vetmedica Gmbh | Antagonisty muskarynowi i ich kombinacje do leczenia choroby dróg oddechowych u koni |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0003935D0 (en) * | 2000-02-08 | 2000-04-12 | King S College London | Formulation for dry powder inhaler |
| DE10050994A1 (de) * | 2000-10-14 | 2002-04-18 | Boehringer Ingelheim Pharma | Neue als Arneimittel einsetzbare Anticholinergika sowie Verfahren zu deren Herstellung |
| DE10130371A1 (de) * | 2001-06-23 | 2003-01-02 | Boehringer Ingelheim Pharma | Neue Arzneimittelkompositionen auf der Basis von Anticholinergika, Corticosteroiden und Betamimetika |
-
2002
- 2002-08-17 DE DE10237739A patent/DE10237739A1/de not_active Withdrawn
-
2003
- 2003-07-25 CA CA2495454A patent/CA2495454C/en not_active Expired - Fee Related
- 2003-07-25 RU RU2005107475/15A patent/RU2332217C2/ru not_active IP Right Cessation
- 2003-07-25 NZ NZ538834A patent/NZ538834A/en not_active IP Right Cessation
- 2003-07-25 WO PCT/EP2003/008222 patent/WO2004022058A1/de active IP Right Grant
- 2003-07-25 PL PL375233A patent/PL212070B1/pl not_active IP Right Cessation
- 2003-07-25 EP EP07103257A patent/EP1785136A3/de not_active Withdrawn
- 2003-07-25 EP EP03793643A patent/EP1530471B1/de not_active Expired - Lifetime
- 2003-07-25 AU AU2003255289A patent/AU2003255289B2/en not_active Ceased
- 2003-07-25 MX MXPA05001823A patent/MXPA05001823A/es active IP Right Grant
- 2003-07-25 KR KR1020057002691A patent/KR101083977B1/ko not_active IP Right Cessation
- 2003-07-25 PT PT03793643T patent/PT1530471E/pt unknown
- 2003-07-25 CN CNA038237989A patent/CN1688308A/zh active Pending
- 2003-07-25 ES ES03793643T patent/ES2290549T3/es not_active Expired - Lifetime
- 2003-07-25 DE DE50307659T patent/DE50307659D1/de not_active Expired - Lifetime
- 2003-07-25 JP JP2004533275A patent/JP2006501253A/ja active Pending
- 2003-07-25 AT AT03793643T patent/ATE366574T1/de active
- 2003-07-25 DK DK03793643T patent/DK1530471T3/da active
- 2003-07-25 BR BR0313526-8A patent/BR0313526A/pt not_active Expired - Fee Related
-
2005
- 2005-01-03 ZA ZA200500019A patent/ZA200500019B/en unknown
- 2005-02-15 IL IL166891A patent/IL166891A/en not_active IP Right Cessation
- 2005-03-15 CO CO05024193A patent/CO5540380A2/es not_active Application Discontinuation
-
2007
- 2007-09-19 CY CY20071101217T patent/CY1107742T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| DK1530471T3 (da) | 2007-10-22 |
| EP1785136A2 (de) | 2007-05-16 |
| PL212070B1 (pl) | 2012-08-31 |
| PL375233A1 (en) | 2005-11-28 |
| CO5540380A2 (es) | 2005-07-29 |
| EP1530471B1 (de) | 2007-07-11 |
| AU2003255289B2 (en) | 2009-08-20 |
| IL166891A (en) | 2010-04-15 |
| RU2005107475A (ru) | 2006-04-10 |
| EP1785136A3 (de) | 2009-04-22 |
| MXPA05001823A (es) | 2005-04-19 |
| BR0313526A (pt) | 2005-06-28 |
| CY1107742T1 (el) | 2013-04-18 |
| ES2290549T3 (es) | 2008-02-16 |
| EP1530471A1 (de) | 2005-05-18 |
| KR20050051644A (ko) | 2005-06-01 |
| CA2495454A1 (en) | 2004-03-18 |
| KR101083977B1 (ko) | 2011-11-22 |
| PT1530471E (pt) | 2007-07-26 |
| NZ538834A (en) | 2007-10-26 |
| WO2004022058A1 (de) | 2004-03-18 |
| DE50307659D1 (de) | 2007-08-23 |
| CN1688308A (zh) | 2005-10-26 |
| ATE366574T1 (de) | 2007-08-15 |
| AU2003255289A1 (en) | 2004-03-29 |
| CA2495454C (en) | 2011-09-06 |
| RU2332217C2 (ru) | 2008-08-27 |
| JP2006501253A (ja) | 2006-01-12 |
| DE10237739A1 (de) | 2004-02-26 |
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