ZA200500019B - Inhalation medicaments containing a novel anticholinesterase drug in conjunction with corticosteroid and betamimetic drugs - Google Patents
Inhalation medicaments containing a novel anticholinesterase drug in conjunction with corticosteroid and betamimetic drugs Download PDFInfo
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- ZA200500019B ZA200500019B ZA200500019A ZA200500019A ZA200500019B ZA 200500019 B ZA200500019 B ZA 200500019B ZA 200500019 A ZA200500019 A ZA 200500019A ZA 200500019 A ZA200500019 A ZA 200500019A ZA 200500019 B ZA200500019 B ZA 200500019B
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- ZA
- South Africa
- Prior art keywords
- hydroxy
- composition according
- pharmaceutical composition
- methyl
- propellant
- Prior art date
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- 239000003814 drug Substances 0.000 title claims abstract description 7
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- 239000000544 cholinesterase inhibitor Substances 0.000 title 1
- 239000000203 mixture Substances 0.000 claims abstract description 44
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- 150000004677 hydrates Chemical class 0.000 claims abstract description 8
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- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
- A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/46—8-Azabicyclo [3.2.1] octane; Derivatives thereof, e.g. atropine, cocaine
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
Landscapes
- Health & Medical Sciences (AREA)
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- Veterinary Medicine (AREA)
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- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Pulmonology (AREA)
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- Emergency Medicine (AREA)
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- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Steroid Compounds (AREA)
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Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10237739A DE10237739A1 (de) | 2002-08-17 | 2002-08-17 | Inhalative Arzneimittel enthaltend ein neues Anticholinergikum in Kombination mit Corticosteroiden und Betamimetika |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200500019B true ZA200500019B (en) | 2006-07-26 |
Family
ID=30775387
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200500019A ZA200500019B (en) | 2002-08-17 | 2005-01-03 | Inhalation medicaments containing a novel anticholinesterase drug in conjunction with corticosteroid and betamimetic drugs |
Country Status (21)
| Country | Link |
|---|---|
| EP (2) | EP1530471B1 (ko) |
| JP (1) | JP2006501253A (ko) |
| KR (1) | KR101083977B1 (ko) |
| CN (1) | CN1688308A (ko) |
| AT (1) | ATE366574T1 (ko) |
| AU (1) | AU2003255289B2 (ko) |
| BR (1) | BR0313526A (ko) |
| CA (1) | CA2495454C (ko) |
| CO (1) | CO5540380A2 (ko) |
| CY (1) | CY1107742T1 (ko) |
| DE (2) | DE10237739A1 (ko) |
| DK (1) | DK1530471T3 (ko) |
| ES (1) | ES2290549T3 (ko) |
| IL (1) | IL166891A (ko) |
| MX (1) | MXPA05001823A (ko) |
| NZ (1) | NZ538834A (ko) |
| PL (1) | PL212070B1 (ko) |
| PT (1) | PT1530471E (ko) |
| RU (1) | RU2332217C2 (ko) |
| WO (1) | WO2004022058A1 (ko) |
| ZA (1) | ZA200500019B (ko) |
Families Citing this family (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2002012265A1 (en) | 2000-08-05 | 2002-02-14 | Glaxo Group Limited | 6.ALPHA., 9.ALPHA.-DIFLUORO-17.ALPHA.-`(2-FURANYLCARBOXYL) OXY!-11.BETA.-HYDROXY-16.ALPHA.-METHYL-3-OXO-ANDROST-1,4,-DIENE-17-CARBOTHIOIC ACID S-FLUOROMETHYL ESTER AS AN ANTI-INFLAMMATORY AGENT |
| SI1383786T1 (sl) | 2001-04-30 | 2009-02-28 | Glaxo Group Ltd | Protivnetni 17.beta-karbotioatestrski derivati androstana s ciklično estrsko skupino na položaju 17.alfa |
| US7056916B2 (en) | 2002-11-15 | 2006-06-06 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Medicaments for the treatment of chronic obstructive pulmonary disease |
| US7220742B2 (en) | 2004-05-14 | 2007-05-22 | Boehringer Ingelheim International Gmbh | Enantiomerically pure beta agonists, process for the manufacture thereof and use thereof as medicaments |
| US7745621B2 (en) | 2004-05-14 | 2010-06-29 | Boehringer Ingelheim International Gmbh | Long acting bronchodilators for the treatment of respiratory diseases |
| DE102004024453A1 (de) * | 2004-05-14 | 2006-01-05 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Neue langwirksame Bronchodilatoren zur Behandlung von Atemwegserkrankungen |
| US20060034776A1 (en) * | 2004-08-10 | 2006-02-16 | Boehringer Ingelheim International Gmbh | Inhalable medicaments containing a new anticholinergic, corticosteroids, and betamimetics |
| DE102004056579A1 (de) * | 2004-11-23 | 2006-05-24 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Inhalative Arzneimittel enthaltend ein neues Anticholinergikum, Salmeterol und ein Steroid |
| DE102004056578A1 (de) * | 2004-11-23 | 2006-05-24 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Inhalative Arzneimittel enthaltend ein neues Anticholinergikum, Formoterol und ein Steroid |
| CN101119706B (zh) | 2005-02-25 | 2013-04-17 | 奇斯药制品公司 | 用于加压计量吸入器的包含螯合剂的药物气雾制剂 |
| JP2008534611A (ja) * | 2005-03-30 | 2008-08-28 | シェーリング コーポレイション | 抗コリン作用薬、コルチコステロイドおよび長時間作用性βアゴニストを合わせる薬物および方法 |
| WO2006114379A1 (de) * | 2005-04-23 | 2006-11-02 | Boehringer Ingelheim International Gmbh | Arzneimittelkombination für die inhalation enthaltend neben einem anticholinergikum ein betamimetikum und ein steroid |
| CA2619402C (en) | 2005-08-15 | 2015-02-03 | Boehringer Ingelheim International Gmbh | Method for producing betamimetics |
| WO2009052624A1 (en) * | 2007-10-25 | 2009-04-30 | Merck Frosst Canada Ltd. | Combination therapy |
| LT2435025T (lt) | 2009-05-29 | 2016-09-26 | Pearl Therapeutics, Inc. | Veikliosios medžiagos tiekimas per kvėpavimo takus |
| US8815258B2 (en) | 2009-05-29 | 2014-08-26 | Pearl Therapeutics, Inc. | Compositions, methods and systems for respiratory delivery of two or more active agents |
| RU2479304C1 (ru) * | 2012-05-29 | 2013-04-20 | Шолекс Девелопмент Гмбх, | Стабильный раствор фенотерола гидробромида |
| RU2504382C1 (ru) * | 2012-06-13 | 2014-01-20 | Шолекс Девелопмент Гмбх | Ингаляционный препарат для лечения бронхиальной астмы и хронической обструктивной болезни легких и способ его получения |
| ES2693779T3 (es) | 2012-12-21 | 2018-12-13 | Boehringer Ingelheim Vetmedica Gmbh | Ciclesonida para el tratamiento de enfermedades de las vías respiratorias en caballos |
| WO2014096116A1 (en) | 2012-12-21 | 2014-06-26 | Boehringer Ingelheim Vetmedica Gmbh | Pharmaceutical formulation comprising ciclesonide |
| JP6454323B2 (ja) | 2013-03-15 | 2019-01-16 | パール セラピューティクス，インコーポレイテッド | 粒子状結晶性材料のコンディショニングのための方法及びシステム |
| WO2015065220A1 (ru) * | 2013-10-28 | 2015-05-07 | Шолекс Девелопмент Гмбх | Ингаляционный препарат для лечения бронхиальной астмы и хронической обструктивной болезни легких и способ его получения |
| WO2015065223A1 (ru) * | 2013-10-28 | 2015-05-07 | Шолекс Девелопмент Гмбх | Стабильный раствор фенотерола гидробромида |
| HUE051527T2 (hu) * | 2014-06-18 | 2021-03-01 | Boehringer Ingelheim Vetmedica Gmbh | Muszkarin-antagonisták és kombinációik légúti betegség lovakban történõ kezelésére |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0003935D0 (en) * | 2000-02-08 | 2000-04-12 | King S College London | Formulation for dry powder inhaler |
| DE10050994A1 (de) * | 2000-10-14 | 2002-04-18 | Boehringer Ingelheim Pharma | Neue als Arneimittel einsetzbare Anticholinergika sowie Verfahren zu deren Herstellung |
| DE10130371A1 (de) * | 2001-06-23 | 2003-01-02 | Boehringer Ingelheim Pharma | Neue Arzneimittelkompositionen auf der Basis von Anticholinergika, Corticosteroiden und Betamimetika |
-
2002
- 2002-08-17 DE DE10237739A patent/DE10237739A1/de not_active Withdrawn
-
2003
- 2003-07-25 PL PL375233A patent/PL212070B1/pl not_active IP Right Cessation
- 2003-07-25 AT AT03793643T patent/ATE366574T1/de active
- 2003-07-25 DE DE50307659T patent/DE50307659D1/de not_active Expired - Lifetime
- 2003-07-25 BR BR0313526-8A patent/BR0313526A/pt not_active Expired - Fee Related
- 2003-07-25 AU AU2003255289A patent/AU2003255289B2/en not_active Ceased
- 2003-07-25 CA CA2495454A patent/CA2495454C/en not_active Expired - Fee Related
- 2003-07-25 EP EP03793643A patent/EP1530471B1/de not_active Expired - Lifetime
- 2003-07-25 PT PT03793643T patent/PT1530471E/pt unknown
- 2003-07-25 CN CNA038237989A patent/CN1688308A/zh active Pending
- 2003-07-25 WO PCT/EP2003/008222 patent/WO2004022058A1/de active IP Right Grant
- 2003-07-25 MX MXPA05001823A patent/MXPA05001823A/es active IP Right Grant
- 2003-07-25 KR KR1020057002691A patent/KR101083977B1/ko not_active IP Right Cessation
- 2003-07-25 RU RU2005107475/15A patent/RU2332217C2/ru not_active IP Right Cessation
- 2003-07-25 NZ NZ538834A patent/NZ538834A/en not_active IP Right Cessation
- 2003-07-25 EP EP07103257A patent/EP1785136A3/de not_active Withdrawn
- 2003-07-25 DK DK03793643T patent/DK1530471T3/da active
- 2003-07-25 JP JP2004533275A patent/JP2006501253A/ja active Pending
- 2003-07-25 ES ES03793643T patent/ES2290549T3/es not_active Expired - Lifetime
-
2005
- 2005-01-03 ZA ZA200500019A patent/ZA200500019B/en unknown
- 2005-02-15 IL IL166891A patent/IL166891A/en not_active IP Right Cessation
- 2005-03-15 CO CO05024193A patent/CO5540380A2/es not_active Application Discontinuation
-
2007
- 2007-09-19 CY CY20071101217T patent/CY1107742T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| MXPA05001823A (es) | 2005-04-19 |
| NZ538834A (en) | 2007-10-26 |
| KR20050051644A (ko) | 2005-06-01 |
| ATE366574T1 (de) | 2007-08-15 |
| DE50307659D1 (de) | 2007-08-23 |
| RU2005107475A (ru) | 2006-04-10 |
| DK1530471T3 (da) | 2007-10-22 |
| CY1107742T1 (el) | 2013-04-18 |
| CA2495454C (en) | 2011-09-06 |
| EP1785136A3 (de) | 2009-04-22 |
| PL212070B1 (pl) | 2012-08-31 |
| CA2495454A1 (en) | 2004-03-18 |
| EP1530471A1 (de) | 2005-05-18 |
| IL166891A (en) | 2010-04-15 |
| PT1530471E (pt) | 2007-07-26 |
| WO2004022058A1 (de) | 2004-03-18 |
| CO5540380A2 (es) | 2005-07-29 |
| KR101083977B1 (ko) | 2011-11-22 |
| ES2290549T3 (es) | 2008-02-16 |
| PL375233A1 (en) | 2005-11-28 |
| CN1688308A (zh) | 2005-10-26 |
| EP1530471B1 (de) | 2007-07-11 |
| EP1785136A2 (de) | 2007-05-16 |
| BR0313526A (pt) | 2005-06-28 |
| JP2006501253A (ja) | 2006-01-12 |
| AU2003255289B2 (en) | 2009-08-20 |
| DE10237739A1 (de) | 2004-02-26 |
| AU2003255289A1 (en) | 2004-03-29 |
| RU2332217C2 (ru) | 2008-08-27 |
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