ZA200500019B - Inhalation medicaments containing a novel anticholinesterase drug in conjunction with corticosteroid and betamimetic drugs - Google Patents
Inhalation medicaments containing a novel anticholinesterase drug in conjunction with corticosteroid and betamimetic drugs Download PDFInfo
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- ZA200500019B ZA200500019B ZA200500019A ZA200500019A ZA200500019B ZA 200500019 B ZA200500019 B ZA 200500019B ZA 200500019 A ZA200500019 A ZA 200500019A ZA 200500019 A ZA200500019 A ZA 200500019A ZA 200500019 B ZA200500019 B ZA 200500019B
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- ZA
- South Africa
- Prior art keywords
- hydroxy
- composition according
- pharmaceutical composition
- methyl
- propellant
- Prior art date
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- 239000003814 drug Substances 0.000 title claims abstract description 7
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- 239000000544 cholinesterase inhibitor Substances 0.000 title 1
- 239000000203 mixture Substances 0.000 claims abstract description 44
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- 150000004677 hydrates Chemical class 0.000 claims abstract description 8
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- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
- A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/46—8-Azabicyclo [3.2.1] octane; Derivatives thereof, e.g. atropine, cocaine
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10237739A DE10237739A1 (de) | 2002-08-17 | 2002-08-17 | Inhalative Arzneimittel enthaltend ein neues Anticholinergikum in Kombination mit Corticosteroiden und Betamimetika |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200500019B true ZA200500019B (en) | 2006-07-26 |
Family
ID=30775387
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200500019A ZA200500019B (en) | 2002-08-17 | 2005-01-03 | Inhalation medicaments containing a novel anticholinesterase drug in conjunction with corticosteroid and betamimetic drugs |
Country Status (21)
| Country | Link |
|---|---|
| EP (2) | EP1530471B1 (fr) |
| JP (1) | JP2006501253A (fr) |
| KR (1) | KR101083977B1 (fr) |
| CN (1) | CN1688308A (fr) |
| AT (1) | ATE366574T1 (fr) |
| AU (1) | AU2003255289B2 (fr) |
| BR (1) | BR0313526A (fr) |
| CA (1) | CA2495454C (fr) |
| CO (1) | CO5540380A2 (fr) |
| CY (1) | CY1107742T1 (fr) |
| DE (2) | DE10237739A1 (fr) |
| DK (1) | DK1530471T3 (fr) |
| ES (1) | ES2290549T3 (fr) |
| IL (1) | IL166891A (fr) |
| MX (1) | MXPA05001823A (fr) |
| NZ (1) | NZ538834A (fr) |
| PL (1) | PL212070B1 (fr) |
| PT (1) | PT1530471E (fr) |
| RU (1) | RU2332217C2 (fr) |
| WO (1) | WO2004022058A1 (fr) |
| ZA (1) | ZA200500019B (fr) |
Families Citing this family (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1305329B2 (fr) | 2000-08-05 | 2015-03-18 | Glaxo Group Limited | 6.alpha., 9.alpha.-difluoro-17.alpha.-(2-furanylcarboxyle) oxy-11.beta.-hydroxy-16.alpha.-methyle-3-oxo-androst-1,4-diene-17-acide carbothioique s-fluoromethyle ester utilise comme agent anti inflammatoire |
| BR0209271A (pt) | 2001-04-30 | 2004-06-15 | Glaxo Group Ltd | Composto, uso de um composto composição farmacêutica, formulação em aerossol farmacêutica, método para o tratamento de um paciente humano ou animal com uma condição inflamatória e/ou alérgica, e, processo para a preparação de um composto |
| US7056916B2 (en) | 2002-11-15 | 2006-06-06 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Medicaments for the treatment of chronic obstructive pulmonary disease |
| US7220742B2 (en) | 2004-05-14 | 2007-05-22 | Boehringer Ingelheim International Gmbh | Enantiomerically pure beta agonists, process for the manufacture thereof and use thereof as medicaments |
| DE102004024453A1 (de) * | 2004-05-14 | 2006-01-05 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Neue langwirksame Bronchodilatoren zur Behandlung von Atemwegserkrankungen |
| US7745621B2 (en) | 2004-05-14 | 2010-06-29 | Boehringer Ingelheim International Gmbh | Long acting bronchodilators for the treatment of respiratory diseases |
| US20060034776A1 (en) * | 2004-08-10 | 2006-02-16 | Boehringer Ingelheim International Gmbh | Inhalable medicaments containing a new anticholinergic, corticosteroids, and betamimetics |
| DE102004056578A1 (de) * | 2004-11-23 | 2006-05-24 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Inhalative Arzneimittel enthaltend ein neues Anticholinergikum, Formoterol und ein Steroid |
| DE102004056579A1 (de) * | 2004-11-23 | 2006-05-24 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Inhalative Arzneimittel enthaltend ein neues Anticholinergikum, Salmeterol und ein Steroid |
| JP5259193B2 (ja) | 2005-02-25 | 2013-08-07 | チエシイ・ファルマセウテイシイ・エス・ペー・アー | 加圧下にある用量計量型吸入器用の金属イオン封鎖剤を含む薬用エーロゾル配合物 |
| EP2484382A1 (fr) * | 2005-03-30 | 2012-08-08 | Schering Corporation | Médicament à base d'un inhibiteur de la phosphodiestérase IV sous une forme adaptée à l'inhalation |
| JP2008538758A (ja) * | 2005-04-23 | 2008-11-06 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 抗コリン作用薬に加えてベータ受容体刺激薬及びステロイドを含有する吸入用の医薬組成物 |
| JP5270343B2 (ja) | 2005-08-15 | 2013-08-21 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | ベータミメティックスの製造方法 |
| WO2009052624A1 (fr) * | 2007-10-25 | 2009-04-30 | Merck Frosst Canada Ltd. | Polythérapie |
| US9463161B2 (en) | 2009-05-29 | 2016-10-11 | Pearl Therapeutics, Inc. | Compositions for pulmonary delivery of long-acting muscarinic antagonists and associated methods and systems |
| US8815258B2 (en) | 2009-05-29 | 2014-08-26 | Pearl Therapeutics, Inc. | Compositions, methods and systems for respiratory delivery of two or more active agents |
| RU2479304C1 (ru) * | 2012-05-29 | 2013-04-20 | Шолекс Девелопмент Гмбх, | Стабильный раствор фенотерола гидробромида |
| RU2504382C1 (ru) * | 2012-06-13 | 2014-01-20 | Шолекс Девелопмент Гмбх | Ингаляционный препарат для лечения бронхиальной астмы и хронической обструктивной болезни легких и способ его получения |
| DK2934544T3 (en) | 2012-12-21 | 2019-03-04 | Boehringer Ingelheim Vetmedica Gmbh | PHARMACEUTICAL FORMULA INCLUDING CICLESONID |
| CA2888428C (fr) | 2012-12-21 | 2021-07-13 | Boehringer Ingelheim Vetmedica Gmbh | Ciclesonide pour le traitement d'une maladie des voies respiratoires chez les chevaux |
| JP6454323B2 (ja) | 2013-03-15 | 2019-01-16 | パール セラピューティクス，インコーポレイテッド | 粒子状結晶性材料のコンディショニングのための方法及びシステム |
| WO2015065220A1 (fr) * | 2013-10-28 | 2015-05-07 | Шолекс Девелопмент Гмбх | Préparation inhalable pour le traitement de l'asthme bronchial et de maladies à obstruction chronique des poumons, et procédé de production |
| WO2015065223A1 (fr) * | 2013-10-28 | 2015-05-07 | Шолекс Девелопмент Гмбх | Solution stable de fénotérol bromhydrate |
| ES2759247T3 (es) | 2014-06-18 | 2020-05-08 | Boehringer Ingelheim Vetmedica Gmbh | Antagonistas muscarínicos y combinaciones de estos para el tratamiento de enfermedades de las vías respiratorias en caballos |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0003935D0 (en) * | 2000-02-08 | 2000-04-12 | King S College London | Formulation for dry powder inhaler |
| DE10050994A1 (de) * | 2000-10-14 | 2002-04-18 | Boehringer Ingelheim Pharma | Neue als Arneimittel einsetzbare Anticholinergika sowie Verfahren zu deren Herstellung |
| DE10130371A1 (de) * | 2001-06-23 | 2003-01-02 | Boehringer Ingelheim Pharma | Neue Arzneimittelkompositionen auf der Basis von Anticholinergika, Corticosteroiden und Betamimetika |
-
2002
- 2002-08-17 DE DE10237739A patent/DE10237739A1/de not_active Withdrawn
-
2003
- 2003-07-25 DE DE50307659T patent/DE50307659D1/de not_active Expired - Lifetime
- 2003-07-25 AT AT03793643T patent/ATE366574T1/de active
- 2003-07-25 CN CNA038237989A patent/CN1688308A/zh active Pending
- 2003-07-25 EP EP03793643A patent/EP1530471B1/fr not_active Expired - Lifetime
- 2003-07-25 WO PCT/EP2003/008222 patent/WO2004022058A1/fr active IP Right Grant
- 2003-07-25 KR KR1020057002691A patent/KR101083977B1/ko not_active IP Right Cessation
- 2003-07-25 ES ES03793643T patent/ES2290549T3/es not_active Expired - Lifetime
- 2003-07-25 CA CA2495454A patent/CA2495454C/fr not_active Expired - Fee Related
- 2003-07-25 RU RU2005107475/15A patent/RU2332217C2/ru not_active IP Right Cessation
- 2003-07-25 NZ NZ538834A patent/NZ538834A/en not_active IP Right Cessation
- 2003-07-25 JP JP2004533275A patent/JP2006501253A/ja active Pending
- 2003-07-25 PL PL375233A patent/PL212070B1/pl not_active IP Right Cessation
- 2003-07-25 PT PT03793643T patent/PT1530471E/pt unknown
- 2003-07-25 MX MXPA05001823A patent/MXPA05001823A/es active IP Right Grant
- 2003-07-25 AU AU2003255289A patent/AU2003255289B2/en not_active Ceased
- 2003-07-25 DK DK03793643T patent/DK1530471T3/da active
- 2003-07-25 BR BR0313526-8A patent/BR0313526A/pt not_active Expired - Fee Related
- 2003-07-25 EP EP07103257A patent/EP1785136A3/fr not_active Withdrawn
-
2005
- 2005-01-03 ZA ZA200500019A patent/ZA200500019B/en unknown
- 2005-02-15 IL IL166891A patent/IL166891A/en not_active IP Right Cessation
- 2005-03-15 CO CO05024193A patent/CO5540380A2/es not_active Application Discontinuation
-
2007
- 2007-09-19 CY CY20071101217T patent/CY1107742T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| RU2005107475A (ru) | 2006-04-10 |
| JP2006501253A (ja) | 2006-01-12 |
| CO5540380A2 (es) | 2005-07-29 |
| DE50307659D1 (de) | 2007-08-23 |
| EP1530471B1 (fr) | 2007-07-11 |
| PT1530471E (pt) | 2007-07-26 |
| AU2003255289B2 (en) | 2009-08-20 |
| MXPA05001823A (es) | 2005-04-19 |
| BR0313526A (pt) | 2005-06-28 |
| EP1785136A2 (fr) | 2007-05-16 |
| RU2332217C2 (ru) | 2008-08-27 |
| KR101083977B1 (ko) | 2011-11-22 |
| EP1530471A1 (fr) | 2005-05-18 |
| DE10237739A1 (de) | 2004-02-26 |
| ATE366574T1 (de) | 2007-08-15 |
| NZ538834A (en) | 2007-10-26 |
| DK1530471T3 (da) | 2007-10-22 |
| CY1107742T1 (el) | 2013-04-18 |
| ES2290549T3 (es) | 2008-02-16 |
| WO2004022058A1 (fr) | 2004-03-18 |
| KR20050051644A (ko) | 2005-06-01 |
| CN1688308A (zh) | 2005-10-26 |
| IL166891A (en) | 2010-04-15 |
| EP1785136A3 (fr) | 2009-04-22 |
| AU2003255289A1 (en) | 2004-03-29 |
| PL212070B1 (pl) | 2012-08-31 |
| CA2495454A1 (fr) | 2004-03-18 |
| CA2495454C (fr) | 2011-09-06 |
| PL375233A1 (en) | 2005-11-28 |
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