ZA200407461B - Carboxylic acid compounds and drugs containing the compounds as the active ingredient. - Google Patents
Carboxylic acid compounds and drugs containing the compounds as the active ingredient. Download PDFInfo
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- ZA200407461B ZA200407461B ZA200407461A ZA200407461A ZA200407461B ZA 200407461 B ZA200407461 B ZA 200407461B ZA 200407461 A ZA200407461 A ZA 200407461A ZA 200407461 A ZA200407461 A ZA 200407461A ZA 200407461 B ZA200407461 B ZA 200407461B
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- -1 Carboxylic acid compounds Chemical class 0.000 title claims abstract description 59
- 150000001875 compounds Chemical class 0.000 title claims abstract description 41
- 239000003814 drug Substances 0.000 title description 5
- 239000004480 active ingredient Substances 0.000 title description 4
- 229940079593 drug Drugs 0.000 title 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 claims abstract description 33
- 201000010099 disease Diseases 0.000 claims abstract description 21
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- 208000035475 disorder Diseases 0.000 claims abstract description 12
- 208000010668 atopic eczema Diseases 0.000 claims abstract description 11
- 206010012438 Dermatitis atopic Diseases 0.000 claims abstract description 9
- 206010039085 Rhinitis allergic Diseases 0.000 claims abstract description 9
- 208000024780 Urticaria Diseases 0.000 claims abstract description 9
- 201000010105 allergic rhinitis Diseases 0.000 claims abstract description 9
- 201000008937 atopic dermatitis Diseases 0.000 claims abstract description 9
- 206010010744 Conjunctivitis allergic Diseases 0.000 claims abstract description 8
- 206010061218 Inflammation Diseases 0.000 claims abstract description 8
- 208000002205 allergic conjunctivitis Diseases 0.000 claims abstract description 8
- 208000006673 asthma Diseases 0.000 claims abstract description 8
- 208000024998 atopic conjunctivitis Diseases 0.000 claims abstract description 8
- 230000004054 inflammatory process Effects 0.000 claims abstract description 8
- 208000030603 inherited susceptibility to asthma Diseases 0.000 claims abstract description 8
- 206010006482 Bronchospasm Diseases 0.000 claims abstract description 7
- 201000008736 Systemic mastocytosis Diseases 0.000 claims abstract description 7
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Classifications
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
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- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
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- C07D327/00—Heterocyclic compounds containing rings having oxygen and sulfur atoms as the only ring hetero atoms
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Landscapes
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- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Pulmonology (AREA)
- Dermatology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Rheumatology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pain & Pain Management (AREA)
- Ophthalmology & Optometry (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Toxicology (AREA)
- Transplantation (AREA)
- Vascular Medicine (AREA)
- Anesthesiology (AREA)
- Urology & Nephrology (AREA)
- Gastroenterology & Hepatology (AREA)
- Otolaryngology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2002076456 | 2002-03-19 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200407461B true ZA200407461B (en) | 2005-07-01 |
Family
ID=28035445
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200407461A ZA200407461B (en) | 2002-03-19 | 2004-09-16 | Carboxylic acid compounds and drugs containing the compounds as the active ingredient. |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US7351705B2 (pl) |
| EP (1) | EP1486491B1 (pl) |
| JP (2) | JP4547913B2 (pl) |
| KR (1) | KR20040095302A (pl) |
| CN (1) | CN100378083C (pl) |
| AT (1) | ATE516277T1 (pl) |
| AU (1) | AU2003221325A1 (pl) |
| BR (1) | BR0308518A (pl) |
| CA (1) | CA2479352A1 (pl) |
| ES (1) | ES2365985T3 (pl) |
| IL (1) | IL164094A0 (pl) |
| MX (1) | MXPA04009095A (pl) |
| NO (1) | NO20043894L (pl) |
| NZ (1) | NZ535309A (pl) |
| PL (1) | PL372466A1 (pl) |
| RU (1) | RU2329256C2 (pl) |
| WO (1) | WO2003078409A1 (pl) |
| ZA (1) | ZA200407461B (pl) |
Families Citing this family (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2003297398B2 (en) | 2002-12-20 | 2009-09-24 | Amgen Inc. | Asthma and allergic inflammation modulators |
| AR041089A1 (es) * | 2003-05-15 | 2005-05-04 | Merck & Co Inc | Procedimiento y composiciones farmaceutiicas para tratar aterosclerosis, dislipidemias y afecciones relacionadas |
| WO2005028455A1 (ja) * | 2003-09-17 | 2005-03-31 | Ono Pharmaceutical Co., Ltd. | カルボン酸化合物およびそれらを有効成分として含有する医薬組成物 |
| TWI258478B (en) | 2003-10-31 | 2006-07-21 | Arena Pharm Inc | Tetrazole derivatives and methods of treatment of metabolic-related disorders thereof |
| US20070244107A1 (en) * | 2004-08-25 | 2007-10-18 | Waters M Gerard | Method of Treating Atherosclerosis, Dyslipidemias and Related Conditions |
| JP2008518957A (ja) * | 2004-11-04 | 2008-06-05 | メルク エンド カムパニー インコーポレーテッド | ナイアシン受容体作動薬、そのような化合物を含んでいる組成物及び治療方法 |
| WO2006052798A2 (en) * | 2004-11-08 | 2006-05-18 | Merck & Co., Inc. | Method of treating pathological blushing |
| EP1824812A4 (en) * | 2004-11-23 | 2009-10-28 | Merck & Co Inc | AGONISTS OF THE NIACIN RECEPTOR, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND TREATMENT PROCEDURES |
| PE20060949A1 (es) | 2004-12-23 | 2006-10-11 | Arena Pharm Inc | Derivados fusionados de pirazol como agonistas del receptor de niacina |
| JPWO2006068162A1 (ja) * | 2004-12-24 | 2008-06-12 | 塩野義製薬株式会社 | 慢性閉塞性肺疾患の治療剤 |
| AU2006214018A1 (en) * | 2005-02-17 | 2006-08-24 | Merck Sharp & Dohme Corp. | Method of treating atherosclerosis, dyslipidemias and related conditions |
| AU2006296004B2 (en) * | 2005-09-27 | 2011-11-17 | Shionogi & Co., Ltd. | Sulfonamide derivative having PGD2 receptor antagonistic activity |
| HUE030850T2 (en) | 2006-06-16 | 2017-06-28 | Univ Pennsylvania | Prostaglandin D2 receptor antagonists for the treatment of hair loss |
| US20100260841A1 (en) * | 2007-02-08 | 2010-10-14 | Paolini John F | Method of Treating Atherosclerosis, Dyslipidemias and Related Conditions |
| TWI410410B (zh) * | 2007-08-10 | 2013-10-01 | Ono Pharmaceutical Co | Phenylacetic acid compounds |
| GB0721611D0 (en) * | 2007-11-02 | 2007-12-12 | Glaxo Group Ltd | Novel compounds |
| ES2471919T3 (es) | 2007-12-19 | 2014-06-27 | Amgen, Inc | Derivados de ácido fenilac�tico como moduladores de inflamación |
| WO2010030360A1 (en) * | 2008-09-11 | 2010-03-18 | Arena Pharmaceuticals, Inc. | 3H-IMIDAZO[4,5-b]PYRIDIN-5-OL DERIVATIVES USEFUL IN THE TREATMENT OF GPR81 RECEPTOR DISORDERS |
| TWI508960B (zh) * | 2009-10-08 | 2015-11-21 | Sanofi Aventis | 作為ｐｇｄｓ抑制劑之苯基二唑衍生物 |
| MX2021003131A (es) | 2018-09-20 | 2021-05-14 | Ono Pharmaceutical Co | Antagonista de prostanoide tipo d (dp). |
| EP3960730A4 (en) | 2019-04-26 | 2023-02-08 | Nissan Chemical Corporation | PROCESS FOR PREPARING AN ARYLSULPHONIC ACID ESTER COMPOUND |
| JP7047954B2 (ja) * | 2020-03-19 | 2022-04-05 | 小野薬品工業株式会社 | フェニル酢酸化合物を含有する医薬組成物 |
| JP7088411B2 (ja) * | 2020-03-19 | 2022-06-21 | 小野薬品工業株式会社 | フェニル酢酸化合物の結晶 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0218728A1 (en) * | 1985-04-03 | 1987-04-22 | Yamanouchi Pharmaceutical Co. Ltd. | Phenylene derivatives |
| PL191760B1 (pl) | 1996-12-13 | 2006-06-30 | Shionogi & Co | Związki, pochodne benzotiofenokarboksyamidu, związki pośrednie, kompozycja farmaceutyczna zawierająca te pochodne oraz lek do leczenia blokady nosa |
| BR0109050A (pt) * | 2000-03-09 | 2004-04-27 | Ono Pharmaceutical Co | Derivados de indol, processo para prepapação e uso dos mesmos |
-
2003
- 2003-03-06 PL PL03372466A patent/PL372466A1/pl not_active Application Discontinuation
- 2003-03-06 JP JP2003576415A patent/JP4547913B2/ja not_active Expired - Fee Related
- 2003-03-06 BR BR0308518-0A patent/BR0308518A/pt not_active IP Right Cessation
- 2003-03-06 IL IL16409403A patent/IL164094A0/xx unknown
- 2003-03-06 AT AT03710260T patent/ATE516277T1/de not_active IP Right Cessation
- 2003-03-06 RU RU2004130837/04A patent/RU2329256C2/ru not_active IP Right Cessation
- 2003-03-06 KR KR10-2004-7014688A patent/KR20040095302A/ko not_active Application Discontinuation
- 2003-03-06 MX MXPA04009095A patent/MXPA04009095A/es active IP Right Grant
- 2003-03-06 AU AU2003221325A patent/AU2003221325A1/en not_active Abandoned
- 2003-03-06 CN CNB03811495XA patent/CN100378083C/zh not_active Expired - Fee Related
- 2003-03-06 NZ NZ535309A patent/NZ535309A/en unknown
- 2003-03-06 ES ES03710260T patent/ES2365985T3/es not_active Expired - Lifetime
- 2003-03-06 CA CA002479352A patent/CA2479352A1/en not_active Abandoned
- 2003-03-06 WO PCT/JP2003/002635 patent/WO2003078409A1/ja active Application Filing
- 2003-03-06 US US10/507,885 patent/US7351705B2/en not_active Expired - Fee Related
- 2003-03-06 EP EP03710260A patent/EP1486491B1/en not_active Expired - Lifetime
-
2004
- 2004-09-16 ZA ZA200407461A patent/ZA200407461B/en unknown
- 2004-09-17 NO NO20043894A patent/NO20043894L/no not_active Application Discontinuation
-
2010
- 2010-04-30 JP JP2010105565A patent/JP5168315B2/ja not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| NZ535309A (en) | 2006-05-26 |
| EP1486491A1 (en) | 2004-12-15 |
| ES2365985T3 (es) | 2011-10-14 |
| CN1656085A (zh) | 2005-08-17 |
| NO20043894L (no) | 2004-12-17 |
| AU2003221325A1 (en) | 2003-09-29 |
| JP5168315B2 (ja) | 2013-03-21 |
| PL372466A1 (pl) | 2005-07-25 |
| RU2004130837A (ru) | 2005-05-27 |
| EP1486491B1 (en) | 2011-07-13 |
| CN100378083C (zh) | 2008-04-02 |
| US7351705B2 (en) | 2008-04-01 |
| IL164094A0 (en) | 2005-12-18 |
| EP1486491A4 (en) | 2006-02-15 |
| MXPA04009095A (es) | 2004-12-06 |
| JPWO2003078409A1 (ja) | 2005-07-14 |
| CA2479352A1 (en) | 2003-09-25 |
| RU2329256C2 (ru) | 2008-07-20 |
| JP4547913B2 (ja) | 2010-09-22 |
| JP2010189431A (ja) | 2010-09-02 |
| WO2003078409A1 (fr) | 2003-09-25 |
| KR20040095302A (ko) | 2004-11-12 |
| US20050222216A1 (en) | 2005-10-06 |
| BR0308518A (pt) | 2005-02-22 |
| ATE516277T1 (de) | 2011-07-15 |
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