ZA200404226B - Citric acid salt of a therapeutic compound and pharmaceutical compositions thereof. - Google Patents
Citric acid salt of a therapeutic compound and pharmaceutical compositions thereof. Download PDFInfo
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- ZA200404226B ZA200404226B ZA200404226A ZA200404226A ZA200404226B ZA 200404226 B ZA200404226 B ZA 200404226B ZA 200404226 A ZA200404226 A ZA 200404226A ZA 200404226 A ZA200404226 A ZA 200404226A ZA 200404226 B ZA200404226 B ZA 200404226B
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- 229960001790 sodium citrate Drugs 0.000 description 1
- 235000011083 sodium citrates Nutrition 0.000 description 1
- 235000019333 sodium laurylsulphate Nutrition 0.000 description 1
- 239000008247 solid mixture Substances 0.000 description 1
- 239000007790 solid phase Substances 0.000 description 1
- 239000007921 spray Substances 0.000 description 1
- 238000000547 structure data Methods 0.000 description 1
- 238000010254 subcutaneous injection Methods 0.000 description 1
- 239000007929 subcutaneous injection Substances 0.000 description 1
- 239000005720 sucrose Substances 0.000 description 1
- 239000000829 suppository Substances 0.000 description 1
- 239000000375 suspending agent Substances 0.000 description 1
- 239000003765 sweetening agent Substances 0.000 description 1
- 235000020357 syrup Nutrition 0.000 description 1
- 239000006188 syrup Substances 0.000 description 1
- 239000000454 talc Substances 0.000 description 1
- 229910052623 talc Inorganic materials 0.000 description 1
- 235000012222 talc Nutrition 0.000 description 1
- HBDDRESWUAFAHY-UHFFFAOYSA-N thiomorpholin-3-one Chemical compound O=C1CSCCN1 HBDDRESWUAFAHY-UHFFFAOYSA-N 0.000 description 1
- 230000000699 topical effect Effects 0.000 description 1
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 description 1
- 238000002424 x-ray crystallography Methods 0.000 description 1
Classifications
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
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- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
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- C07D417/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing aromatic rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D279/10—1,4-Thiazines; Hydrogenated 1,4-thiazines
- C07D279/12—1,4-Thiazines; Hydrogenated 1,4-thiazines not condensed with other rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Psychiatry (AREA)
- Addiction (AREA)
- Endocrinology (AREA)
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- Epidemiology (AREA)
- Psychology (AREA)
- Reproductive Health (AREA)
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- Obesity (AREA)
- Child & Adolescent Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US33834301P | 2001-12-07 | 2001-12-07 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200404226B true ZA200404226B (en) | 2005-08-29 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| ZA200404226A ZA200404226B (en) | 2001-12-07 | 2004-05-28 | Citric acid salt of a therapeutic compound and pharmaceutical compositions thereof. |
Country Status (29)
| Country | Link |
|---|---|
| US (1) | US6825193B2 (de) |
| EP (1) | EP1451166B1 (de) |
| JP (1) | JP4165882B2 (de) |
| KR (1) | KR100572430B1 (de) |
| CN (1) | CN100358878C (de) |
| AR (1) | AR037711A1 (de) |
| AT (1) | ATE301647T1 (de) |
| AU (1) | AU2002347504B2 (de) |
| BR (1) | BR0214780A (de) |
| CA (1) | CA2469225C (de) |
| DE (1) | DE60205504T2 (de) |
| DK (1) | DK1451166T3 (de) |
| ES (1) | ES2243774T3 (de) |
| GT (1) | GT200200260A (de) |
| HK (1) | HK1071133A1 (de) |
| HN (1) | HN2002000354A (de) |
| IL (1) | IL162096A0 (de) |
| MX (1) | MXPA04005418A (de) |
| NO (1) | NO327100B1 (de) |
| NZ (1) | NZ532993A (de) |
| PA (1) | PA8560101A1 (de) |
| PE (1) | PE20030663A1 (de) |
| PL (1) | PL370307A1 (de) |
| PT (1) | PT1451166E (de) |
| RU (1) | RU2270834C2 (de) |
| TW (1) | TWI233356B (de) |
| UY (1) | UY27570A1 (de) |
| WO (1) | WO2003048141A1 (de) |
| ZA (1) | ZA200404226B (de) |
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| EP1746091A1 (de) * | 2001-08-30 | 2007-01-24 | Pfizer Products Inc. | Verfahren zur Herstellung von 2-substituiertem 2-[-(4-Methylpiperazin-1-yl)-benzyliden]-thiomorpholin-3-on citrat |
| US20050171095A1 (en) * | 2004-01-06 | 2005-08-04 | Pfizer Inc | Combination of CRF antagonists and 5-HT1B receptor antagonists |
| MXPA06013163A (es) * | 2004-05-11 | 2007-02-13 | Pfizer Prod Inc | Combinacion de antipsicoticos atipicos y antagonistas del receptor 5-ht1b. |
| WO2005113526A2 (en) * | 2004-05-21 | 2005-12-01 | Pfizer Products Inc. | Metabolites of 4-(3,4-dichloro-phenyl)-2-[2-(4-methyl-piperazin-1-yl)-benzylidene]-thiomorpholin-3-one |
| EP1791541A2 (de) * | 2004-09-10 | 2007-06-06 | Pfizer Products Inc. | Verfahren zur behandlung von stimmungsstörungen unter verwendung benzisoxazole enthaltender diazabicyclischer verbindungen |
| US20100189788A1 (en) | 2009-01-23 | 2010-07-29 | Teva Pharmaceutical Industries, Ltd. | Delayed release rasagiline base formulation |
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| US6423708B1 (en) * | 1996-09-30 | 2002-07-23 | Pfizer Inc | Aralkyl and aralkylidene heterocyclic lactams and imides |
| UA56185C2 (uk) * | 1996-09-30 | 2003-05-15 | Пфайзер Інк. | Аралкіл- та аралкіліденгетероциклічні лактами та іміди, фармацевтична композиція та спосіб лікування |
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