ZA200403681B - Piperidine derivatives and their use as modulators of chemokine receptor activity (especially CCR5). - Google Patents
Piperidine derivatives and their use as modulators of chemokine receptor activity (especially CCR5). Download PDFInfo
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- ZA200403681B ZA200403681B ZA200403681A ZA200403681A ZA200403681B ZA 200403681 B ZA200403681 B ZA 200403681B ZA 200403681 A ZA200403681 A ZA 200403681A ZA 200403681 A ZA200403681 A ZA 200403681A ZA 200403681 B ZA200403681 B ZA 200403681B
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- Prior art keywords
- alkyl
- phenyl
- nhc
- compound
- nhs
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- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
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- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A—HUMAN NECESSITIES
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- A61P17/00—Drugs for dermatological disorders
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- C—CHEMISTRY; METALLURGY
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/56—Nitrogen atoms
- C07D211/58—Nitrogen atoms attached in position 4
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- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
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Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
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| SE0103819A SE0103819D0 (sv) | 2001-11-15 | 2001-11-15 | Chemical compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200403681B true ZA200403681B (en) | 2005-08-02 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| ZA200403681A ZA200403681B (en) | 2001-11-15 | 2004-05-13 | Piperidine derivatives and their use as modulators of chemokine receptor activity (especially CCR5). |
Country Status (19)
| Country | Link |
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| US (1) | US20050014788A1 (pt) |
| EP (1) | EP1448524A1 (pt) |
| JP (1) | JP2005513017A (pt) |
| KR (1) | KR20050013526A (pt) |
| CN (1) | CN1589261A (pt) |
| AR (1) | AR037350A1 (pt) |
| BR (1) | BR0214141A (pt) |
| CA (1) | CA2464861A1 (pt) |
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| SE (1) | SE0103819D0 (pt) |
| TW (1) | TW200407140A (pt) |
| WO (1) | WO2003042177A1 (pt) |
| ZA (1) | ZA200403681B (pt) |
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| SE0202483D0 (sv) * | 2002-08-21 | 2002-08-21 | Astrazeneca Ab | Chemical compounds |
| SE0301369D0 (sv) * | 2003-05-09 | 2003-05-09 | Astrazeneca Ab | Chemical compounds |
| SE0302090D0 (sv) * | 2003-07-16 | 2003-07-16 | Astrazeneca Ab | Chemical compounds |
| EP1654229B1 (en) * | 2003-07-31 | 2007-05-09 | AstraZeneca AB | Piperidine derivatives as ccr5 receptor modulators |
| EP1786816A4 (en) | 2003-09-10 | 2009-11-04 | Virochem Pharma Inc | SPIROHYDANTOIN COMPOUNDS AND METHODS FOR MODULATING CHEMOKINE RECEPTOR ACTIVITY |
| SE0303396D0 (sv) * | 2003-12-16 | 2003-12-16 | Astrazeneca Ab | Chemical compounds |
| CN1329374C (zh) * | 2004-06-09 | 2007-08-01 | 上海靶点药物有限公司 | 作为ccr5拮抗剂的化合物 |
| KR100905260B1 (ko) | 2004-06-09 | 2009-06-30 | 상해 타킷 드러그 주식회사 | 씨씨알5 길항제로서의 화합물 |
| SE0401656D0 (sv) * | 2004-06-24 | 2004-06-24 | Astrazeneca Ab | Chemical compounds |
| SE0403084D0 (sv) | 2004-12-17 | 2004-12-17 | Astrazeneca Ab | Chemical process |
| WO2007085357A1 (en) | 2006-01-30 | 2007-08-02 | Euro-Celtique S.A. | Cyclourea compounds as calcium channel blockers |
| GB0625523D0 (en) * | 2006-12-21 | 2007-01-31 | Ge Healthcare Ltd | In vivo imaging agents |
| EP2173715A2 (en) * | 2007-07-13 | 2010-04-14 | Euroscreen S.A. | Use of piperidine derivatives as agonists of chemokine receptor activity |
| US10343982B2 (en) * | 2013-09-25 | 2019-07-09 | Merck Patent Gmbh | Compounds and mesogenic media |
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| HUP0004200A3 (en) * | 1997-11-18 | 2001-04-28 | Dupont Pharmaceuticals Res Lab | Cyclic amine derivatives and their use as drugs |
| EP1013276A1 (en) * | 1998-12-23 | 2000-06-28 | Pfizer Inc. | Aminoazacycloalkanes as CCR5 modulators |
| SE9902987D0 (sv) * | 1999-08-24 | 1999-08-24 | Astra Pharma Prod | Novel compounds |
| GB0011838D0 (en) * | 2000-05-17 | 2000-07-05 | Astrazeneca Ab | Chemical compounds |
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2001
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2002
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- 2002-11-12 MX MXPA04004497A patent/MXPA04004497A/es unknown
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- 2002-11-12 IL IL16159402A patent/IL161594A0/xx unknown
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- 2002-11-12 HU HU0402567A patent/HUP0402567A2/hu unknown
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- 2002-11-12 CN CNA028227409A patent/CN1589261A/zh active Pending
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2004
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Also Published As
| Publication number | Publication date |
|---|---|
| KR20050013526A (ko) | 2005-02-04 |
| RU2004112781A (ru) | 2005-10-10 |
| IL161594A0 (en) | 2004-09-27 |
| WO2003042177A8 (en) | 2005-01-06 |
| JP2005513017A (ja) | 2005-05-12 |
| SE0103819D0 (sv) | 2001-11-15 |
| AR037350A1 (es) | 2004-11-03 |
| PL370910A1 (en) | 2005-05-30 |
| BR0214141A (pt) | 2004-10-19 |
| WO2003042177A1 (en) | 2003-05-22 |
| MXPA04004497A (es) | 2004-08-11 |
| HUP0402567A2 (hu) | 2005-03-29 |
| CN1589261A (zh) | 2005-03-02 |
| IS7257A (is) | 2004-05-10 |
| TW200407140A (en) | 2004-05-16 |
| NO20042156L (no) | 2004-08-11 |
| US20050014788A1 (en) | 2005-01-20 |
| EP1448524A1 (en) | 2004-08-25 |
| CA2464861A1 (en) | 2003-05-22 |
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