ZA200403681B - Piperidine derivatives and their use as modulators of chemokine receptor activity (especially CCR5). - Google Patents
Piperidine derivatives and their use as modulators of chemokine receptor activity (especially CCR5). Download PDFInfo
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- ZA200403681B ZA200403681B ZA200403681A ZA200403681A ZA200403681B ZA 200403681 B ZA200403681 B ZA 200403681B ZA 200403681 A ZA200403681 A ZA 200403681A ZA 200403681 A ZA200403681 A ZA 200403681A ZA 200403681 B ZA200403681 B ZA 200403681B
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- Prior art keywords
- alkyl
- phenyl
- nhc
- compound
- nhs
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- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
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- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A—HUMAN NECESSITIES
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- A61P17/00—Drugs for dermatological disorders
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| SE0103819A SE0103819D0 (sv) | 2001-11-15 | 2001-11-15 | Chemical compounds |
Publications (1)
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| ZA200403681B true ZA200403681B (en) | 2005-08-02 |
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| ZA200403681A ZA200403681B (en) | 2001-11-15 | 2004-05-13 | Piperidine derivatives and their use as modulators of chemokine receptor activity (especially CCR5). |
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| CA2579609A1 (en) | 2003-09-10 | 2005-03-17 | Virochem Pharma Inc. | Spirohydantoin compounds and methods for the modulation of chemokine receptor activity |
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| KR100905260B1 (ko) | 2004-06-09 | 2009-06-30 | 상해 타킷 드러그 주식회사 | 씨씨알5 길항제로서의 화합물 |
| CN1329374C (zh) * | 2004-06-09 | 2007-08-01 | 上海靶点药物有限公司 | 作为ccr5拮抗剂的化合物 |
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| SE0403084D0 (sv) | 2004-12-17 | 2004-12-17 | Astrazeneca Ab | Chemical process |
| JP2009525269A (ja) | 2006-01-30 | 2009-07-09 | ユーロ−セルティーク エス．エイ． | カルシウムチャネルブロッカーとしての環状尿素化合物 |
| GB0625523D0 (en) * | 2006-12-21 | 2007-01-31 | Ge Healthcare Ltd | In vivo imaging agents |
| EP2173715A2 (en) * | 2007-07-13 | 2010-04-14 | Euroscreen S.A. | Use of piperidine derivatives as agonists of chemokine receptor activity |
| CN105579555A (zh) * | 2013-09-25 | 2016-05-11 | 默克专利股份有限公司 | 化合物和介晶介质 |
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| AU744685B2 (en) * | 1997-11-18 | 2002-02-28 | Teijin Pharma Limited | Cyclic amine derivatives and their use as drugs |
| EP1013276A1 (en) * | 1998-12-23 | 2000-06-28 | Pfizer Inc. | Aminoazacycloalkanes as CCR5 modulators |
| SE9902987D0 (sv) * | 1999-08-24 | 1999-08-24 | Astra Pharma Prod | Novel compounds |
| GB0011838D0 (en) * | 2000-05-17 | 2000-07-05 | Astrazeneca Ab | Chemical compounds |
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2002
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Also Published As
| Publication number | Publication date |
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| PL370910A1 (en) | 2005-05-30 |
| RU2004112781A (ru) | 2005-10-10 |
| US20050014788A1 (en) | 2005-01-20 |
| IL161594A0 (en) | 2004-09-27 |
| JP2005513017A (ja) | 2005-05-12 |
| SE0103819D0 (sv) | 2001-11-15 |
| IS7257A (is) | 2004-05-10 |
| CA2464861A1 (en) | 2003-05-22 |
| BR0214141A (pt) | 2004-10-19 |
| EP1448524A1 (en) | 2004-08-25 |
| WO2003042177A8 (en) | 2005-01-06 |
| NO20042156L (no) | 2004-08-11 |
| MXPA04004497A (es) | 2004-08-11 |
| WO2003042177A1 (en) | 2003-05-22 |
| AR037350A1 (es) | 2004-11-03 |
| TW200407140A (en) | 2004-05-16 |
| CN1589261A (zh) | 2005-03-02 |
| HUP0402567A2 (hu) | 2005-03-29 |
| KR20050013526A (ko) | 2005-02-04 |
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