ZA200305659B - Sulfamidothienopyrimidines and the use of the same as phosphodiesterase V inhibitors. - Google Patents
Sulfamidothienopyrimidines and the use of the same as phosphodiesterase V inhibitors. Download PDFInfo
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- ZA200305659B ZA200305659B ZA200305659A ZA200305659A ZA200305659B ZA 200305659 B ZA200305659 B ZA 200305659B ZA 200305659 A ZA200305659 A ZA 200305659A ZA 200305659 A ZA200305659 A ZA 200305659A ZA 200305659 B ZA200305659 B ZA 200305659B
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Classifications
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
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- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pulmonology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Urology & Nephrology (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Immunology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Ophthalmology & Optometry (AREA)
- Physical Education & Sports Medicine (AREA)
- Hospice & Palliative Care (AREA)
- Vascular Medicine (AREA)
- Gynecology & Obstetrics (AREA)
- Gastroenterology & Hepatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10064994A DE10064994A1 (de) | 2000-12-23 | 2000-12-23 | Sulfamidothienopyrimidine |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200305659B true ZA200305659B (en) | 2004-08-27 |
Family
ID=7668967
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200305659A ZA200305659B (en) | 2000-12-23 | 2003-07-22 | Sulfamidothienopyrimidines and the use of the same as phosphodiesterase V inhibitors. |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US7019013B2 (fr) |
| EP (1) | EP1353927B1 (fr) |
| JP (1) | JP4550361B2 (fr) |
| KR (1) | KR20030062438A (fr) |
| CN (1) | CN1483035A (fr) |
| AR (1) | AR035524A1 (fr) |
| AT (1) | ATE302781T1 (fr) |
| BR (1) | BR0115996A (fr) |
| CA (1) | CA2432582C (fr) |
| CZ (1) | CZ20031815A3 (fr) |
| DE (2) | DE10064994A1 (fr) |
| ES (1) | ES2247007T3 (fr) |
| HU (1) | HUP0302515A3 (fr) |
| MX (1) | MXPA03005714A (fr) |
| PL (1) | PL361733A1 (fr) |
| RU (1) | RU2003122189A (fr) |
| SK (1) | SK8432003A3 (fr) |
| WO (1) | WO2002051848A2 (fr) |
| ZA (1) | ZA200305659B (fr) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN101100472A (zh) * | 2001-04-30 | 2008-01-09 | 美国拜尔公司 | 4-氨基-5,6-取代的噻吩并[2,3-d]嘧啶化合物及其应用 |
| EP1847543A1 (fr) | 2006-04-19 | 2007-10-24 | Boehringer Ingelheim Pharma GmbH & Co. KG | Dihydrothienopyrimidines pour le traitement de maladies inflammatoires |
| BRPI0608387A2 (pt) * | 2006-04-19 | 2009-12-29 | Boehringer Ingelheim Int | compostos para o tratamento de doenças inflamatórias |
| US8080549B2 (en) * | 2007-01-12 | 2011-12-20 | Concert Pharmaceuticals, Inc. | Endothelin receptor antagonists |
| US8071596B2 (en) | 2007-01-12 | 2011-12-06 | Concert Pharmaceuticals, Inc. | Endothelin receptor antagonists |
| CN101641099A (zh) | 2007-01-24 | 2010-02-03 | 葛兰素集团有限公司 | 包含3,5-二氨基-6-(2,3-二氯苯基)-1,2,4-三嗪或r(-)-2,4-二氨基-5-(2,3-二氯苯基)-6-氟甲基嘧啶和nk1的药物组合物 |
| JP5150728B2 (ja) * | 2007-10-19 | 2013-02-27 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 置換ピペリジノ−ジヒドロチエノピリミジン |
| WO2009050236A1 (fr) | 2007-10-19 | 2009-04-23 | Boehringer Ingelheim International Gmbh | Nouveaux dérivés de pipérazino-dihydrothiénopyrimidine |
| CN101827853A (zh) | 2007-10-19 | 2010-09-08 | 贝林格尔.英格海姆国际有限公司 | 杂环取代的哌嗪子基-二氢噻吩并嘧啶 |
| WO2012012712A2 (fr) | 2010-07-23 | 2012-01-26 | President And Fellows Of Harvard College | Composés renforçant l'activité protéasome tricyclique |
| US20130059866A1 (en) | 2011-08-24 | 2013-03-07 | Boehringer Ingelheim International Gmbh | Novel piperidino-dihydrothienopyrimidine sulfoxides and their use for treating copd and asthma |
| US9802954B2 (en) | 2011-08-24 | 2017-10-31 | Boehringer Ingelheim International Gmbh | Piperidino-dihydrothienopyrimidine sulfoxides and their use for treating COPD and asthma |
| WO2013112706A1 (fr) | 2012-01-25 | 2013-08-01 | Proteostasis Therapeutics, Inc. | Composés permettant de moduler l'activité de protéasome |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19644228A1 (de) * | 1996-10-24 | 1998-04-30 | Merck Patent Gmbh | Thienopyrimidine |
| DE19752952A1 (de) * | 1997-11-28 | 1999-06-02 | Merck Patent Gmbh | Thienopyrimidine |
| DE19819023A1 (de) * | 1998-04-29 | 1999-11-04 | Merck Patent Gmbh | Thienopyrimidine |
| US6482948B1 (en) | 1999-03-30 | 2002-11-19 | Nippon Soda Co., Ltd. | Thienopyrimidine compounds and salts thereof and process for the preparation of the same |
-
2000
- 2000-12-23 DE DE10064994A patent/DE10064994A1/de not_active Withdrawn
-
2001
- 2001-12-03 US US10/451,183 patent/US7019013B2/en not_active Expired - Fee Related
- 2001-12-03 CA CA2432582A patent/CA2432582C/fr not_active Expired - Fee Related
- 2001-12-03 MX MXPA03005714A patent/MXPA03005714A/es not_active Application Discontinuation
- 2001-12-03 JP JP2002552942A patent/JP4550361B2/ja not_active Expired - Fee Related
- 2001-12-03 SK SK843-2003A patent/SK8432003A3/sk unknown
- 2001-12-03 CN CNA018212190A patent/CN1483035A/zh active Pending
- 2001-12-03 PL PL01361733A patent/PL361733A1/xx unknown
- 2001-12-03 CZ CZ20031815A patent/CZ20031815A3/cs unknown
- 2001-12-03 DE DE50107230T patent/DE50107230D1/de not_active Expired - Lifetime
- 2001-12-03 RU RU2003122189/04A patent/RU2003122189A/ru not_active Application Discontinuation
- 2001-12-03 KR KR10-2003-7008265A patent/KR20030062438A/ko not_active Application Discontinuation
- 2001-12-03 HU HU0302515A patent/HUP0302515A3/hu unknown
- 2001-12-03 EP EP01271992A patent/EP1353927B1/fr not_active Expired - Lifetime
- 2001-12-03 BR BR0115996-8A patent/BR0115996A/pt not_active Application Discontinuation
- 2001-12-03 ES ES01271992T patent/ES2247007T3/es not_active Expired - Lifetime
- 2001-12-03 AT AT01271992T patent/ATE302781T1/de not_active IP Right Cessation
- 2001-12-03 WO PCT/EP2001/014102 patent/WO2002051848A2/fr active IP Right Grant
- 2001-12-19 AR ARP010105889A patent/AR035524A1/es not_active Application Discontinuation
-
2003
- 2003-07-22 ZA ZA200305659A patent/ZA200305659B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| DE10064994A1 (de) | 2002-07-04 |
| DE50107230D1 (de) | 2005-09-29 |
| EP1353927A2 (fr) | 2003-10-22 |
| WO2002051848A3 (fr) | 2002-10-24 |
| KR20030062438A (ko) | 2003-07-25 |
| ATE302781T1 (de) | 2005-09-15 |
| JP4550361B2 (ja) | 2010-09-22 |
| RU2003122189A (ru) | 2004-12-27 |
| SK8432003A3 (en) | 2003-10-07 |
| CN1483035A (zh) | 2004-03-17 |
| US20040063943A1 (en) | 2004-04-01 |
| EP1353927B1 (fr) | 2005-08-24 |
| HUP0302515A2 (hu) | 2003-11-28 |
| CA2432582C (fr) | 2011-01-25 |
| JP2004516329A (ja) | 2004-06-03 |
| MXPA03005714A (es) | 2003-10-06 |
| US7019013B2 (en) | 2006-03-28 |
| CZ20031815A3 (cs) | 2003-10-15 |
| AR035524A1 (es) | 2004-06-02 |
| PL361733A1 (en) | 2004-10-04 |
| CA2432582A1 (fr) | 2002-07-04 |
| BR0115996A (pt) | 2004-01-06 |
| ES2247007T3 (es) | 2006-03-01 |
| WO2002051848A2 (fr) | 2002-07-04 |
| HUP0302515A3 (en) | 2005-06-28 |
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