ZA200304557B - Tetrahydro-(benzo or thieno)-azepine-pyrazine and triazine derivatives as mGluR 1 antagonists. - Google Patents
Tetrahydro-(benzo or thieno)-azepine-pyrazine and triazine derivatives as mGluR 1 antagonists. Download PDFInfo
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- ZA200304557B ZA200304557B ZA200304557A ZA200304557A ZA200304557B ZA 200304557 B ZA200304557 B ZA 200304557B ZA 200304557 A ZA200304557 A ZA 200304557A ZA 200304557 A ZA200304557 A ZA 200304557A ZA 200304557 B ZA200304557 B ZA 200304557B
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Classifications
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- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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- Health & Medical Sciences (AREA)
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- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP00128329 | 2000-12-22 |
Publications (1)
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| ZA200304557B true ZA200304557B (en) | 2004-09-13 |
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| US7678363B2 (en) | 2005-08-26 | 2010-03-16 | Braincells Inc | Methods of treating psychiatric conditions comprising administration of muscarinic agents in combination with SSRIs |
| EP2258359A3 (en) | 2005-08-26 | 2011-04-06 | Braincells, Inc. | Neurogenesis by muscarinic receptor modulation with sabcomelin |
| WO2007047978A2 (en) | 2005-10-21 | 2007-04-26 | Braincells, Inc. | Modulation of neurogenesis by pde inhibition |
| AU2006308889A1 (en) | 2005-10-31 | 2007-05-10 | Braincells, Inc. | GABA receptor mediated modulation of neurogenesis |
| MX2008009178A (es) * | 2006-01-19 | 2008-12-05 | Athersys Inc | Tiofenil y pirrolil acepinas como ligandos del receptor de serotonina 5-ht2c y sus usos. |
| US20100216734A1 (en) | 2006-03-08 | 2010-08-26 | Braincells, Inc. | Modulation of neurogenesis by nootropic agents |
| WO2007134077A2 (en) | 2006-05-09 | 2007-11-22 | Braincells, Inc. | 5 ht receptor mediated neurogenesis |
| CA2651813A1 (en) | 2006-05-09 | 2007-11-22 | Braincells, Inc. | Neurogenesis by modulating angiotensin |
| CA2662491A1 (en) | 2006-09-08 | 2008-03-13 | Braincells, Inc. | Combinations containing a 4-acylaminopyridine derivative |
| US20100184806A1 (en) | 2006-09-19 | 2010-07-22 | Braincells, Inc. | Modulation of neurogenesis by ppar agents |
| WO2010099217A1 (en) | 2009-02-25 | 2010-09-02 | Braincells, Inc. | Modulation of neurogenesis using d-cycloserine combinations |
| KR101100864B1 (ko) * | 2009-06-12 | 2012-01-02 | 양준호 | 자동차 광택기용 광택패드 |
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| DE3136654A1 (de) | 1981-09-16 | 1983-03-31 | Zahnradfabrik Friedrichshafen Ag, 7990 Friedrichshafen | Linearverschieblicher arbeitsarm, insbesondere fuer handhabungsgeraete |
| EP1059090A4 (en) * | 1998-03-03 | 2002-02-27 | Yamanouchi Pharma Co Ltd | DRUGS AGAINST BLEEDING OF THE BRAIN |
| PT1117403E (pt) * | 1998-10-02 | 2004-04-30 | Sibia Neurosciences Inc | Antagonistas de mglurs para o tratamento da dor e ansiedade |
| GB9823847D0 (en) * | 1998-11-02 | 1998-12-23 | Lilly Co Eli | Pharmaceutical compounds |
| EP1074549B1 (en) * | 1999-08-06 | 2003-11-19 | F. Hoffmann-La Roche Ag | Tetrahydro-benzo(d)azepines and their use as antagonists at metabotropic glutamate receptors |
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- 2001-12-11 JP JP2002552562A patent/JP4077319B2/ja not_active Expired - Fee Related
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2003
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Also Published As
| Publication number | Publication date |
|---|---|
| CN1487831A (zh) | 2004-04-07 |
| ATE297734T1 (de) | 2005-07-15 |
| DE60111568D1 (de) | 2005-07-21 |
| MXPA03005515A (es) | 2003-09-25 |
| AU2002216095B2 (en) | 2005-12-01 |
| KR100545906B1 (ko) | 2006-01-26 |
| PT1345609E (pt) | 2005-08-31 |
| CN1260226C (zh) | 2006-06-21 |
| EP1345609B1 (en) | 2005-06-15 |
| WO2002051418A1 (en) | 2002-07-04 |
| ES2243400T3 (es) | 2005-12-01 |
| CA2432077A1 (en) | 2002-07-04 |
| DK1345609T3 (da) | 2005-10-03 |
| CA2432077C (en) | 2011-01-18 |
| EP1345609A1 (en) | 2003-09-24 |
| BR0116378A (pt) | 2003-10-28 |
| KR20030062444A (ko) | 2003-07-25 |
| JP2004517850A (ja) | 2004-06-17 |
| DE60111568T2 (de) | 2006-05-11 |
| JP4077319B2 (ja) | 2008-04-16 |
| AR032379A1 (es) | 2003-11-05 |
| US6586422B2 (en) | 2003-07-01 |
| US20020123488A1 (en) | 2002-09-05 |
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