ZA200110453B - Diphosphate salt of a 4"-substituted-9-deoxo-9a-aza-9a-homoerythromycin derivative and its pharmaceutical composition. - Google Patents

Diphosphate salt of a 4"-substituted-9-deoxo-9a-aza-9a-homoerythromycin derivative and its pharmaceutical composition.

Info

Publication number
ZA200110453B
ZA200110453B ZA200110453A ZA200110453A ZA200110453B ZA 200110453 B ZA200110453 B ZA 200110453B ZA 200110453 A ZA200110453 A ZA 200110453A ZA 200110453 A ZA200110453 A ZA 200110453A ZA 200110453 B ZA200110453 B ZA 200110453B
Authority
ZA
South Africa
Prior art keywords
deoxo
aza
substituted
pharmaceutical composition
diphosphate salt
Prior art date
Application number
ZA200110453A
Other languages
English (en)
Inventor
Robert John Rafka
Colman Brendan Ragan
Douglas John Meldrum Allen
Original Assignee
Prizer Products Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Prizer Products Inc filed Critical Prizer Products Inc
Publication of ZA200110453B publication Critical patent/ZA200110453B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Otolaryngology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
ZA200110453A 1999-06-30 2001-12-20 Diphosphate salt of a 4"-substituted-9-deoxo-9a-aza-9a-homoerythromycin derivative and its pharmaceutical composition. ZA200110453B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US14168199P 1999-06-30 1999-06-30

Publications (1)

Publication Number Publication Date
ZA200110453B true ZA200110453B (en) 2003-03-04

Family

ID=22496734

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200110453A ZA200110453B (en) 1999-06-30 2001-12-20 Diphosphate salt of a 4"-substituted-9-deoxo-9a-aza-9a-homoerythromycin derivative and its pharmaceutical composition.

Country Status (42)

Country Link
US (3) US6465437B1 (ru)
EP (1) EP1189913B1 (ru)
JP (1) JP2003503506A (ru)
KR (1) KR100442508B1 (ru)
CN (2) CN101220067A (ru)
AP (1) AP2001002370A0 (ru)
AR (1) AR035551A1 (ru)
AT (1) ATE286906T1 (ru)
AU (1) AU772277B2 (ru)
BG (1) BG65587B1 (ru)
BR (1) BR0012091A (ru)
CA (1) CA2376748C (ru)
CO (1) CO5190679A1 (ru)
CZ (1) CZ20014571A3 (ru)
DE (1) DE60017399T2 (ru)
EA (1) EA004235B1 (ru)
EC (1) ECSP003555A (ru)
EE (1) EE05068B1 (ru)
ES (1) ES2233380T3 (ru)
GT (2) GT200000105AA (ru)
HN (1) HN2000000090A (ru)
HR (1) HRP20010919B1 (ru)
HU (1) HUP0201693A3 (ru)
IL (1) IL146408A0 (ru)
IS (1) IS6159A (ru)
MA (1) MA26745A1 (ru)
MX (1) MXPA02000058A (ru)
MY (1) MY133360A (ru)
NO (1) NO20016221L (ru)
OA (1) OA11965A (ru)
PA (1) PA8496901A1 (ru)
PE (1) PE20010287A1 (ru)
PL (1) PL201891B1 (ru)
PT (1) PT1189913E (ru)
SK (1) SK286243B6 (ru)
TN (1) TNSN00143A1 (ru)
TR (1) TR200103834T2 (ru)
UA (1) UA71013C2 (ru)
UY (1) UY26221A1 (ru)
WO (1) WO2001002414A1 (ru)
YU (1) YU88701A (ru)
ZA (1) ZA200110453B (ru)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6465437B1 (en) * 1999-06-30 2002-10-15 Pfizer Inc. Diphosphate salt of a 4″-substituted-9-deoxo-9A-AZA-9A- homoerythromycin derivative and its pharmaceutical composition
US6791660B1 (en) * 2002-02-12 2004-09-14 Seiko Epson Corporation Method for manufacturing electrooptical device and apparatus for manufacturing the same, electrooptical device and electronic appliances
US20060116336A1 (en) * 2004-03-17 2006-06-01 American Pharmaceutical Partners, Inc. Lyophilized azithromycin formulation
US7468428B2 (en) 2004-03-17 2008-12-23 App Pharmaceuticals, Llc Lyophilized azithromycin formulation
WO2013013834A1 (en) 2011-07-27 2013-01-31 Farma Grs, D.O.O. New crystalline forms of tulathromycin
CN106008622A (zh) * 2016-08-02 2016-10-12 海门慧聚药业有限公司 泰拉霉素新晶型及其制备
CN110885351A (zh) * 2019-12-17 2020-03-17 海门慧聚药业有限公司 泰拉霉素磷酸盐的晶型及其制备方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SI8110592A8 (en) * 1981-03-06 1996-06-30 Pliva Pharm & Chem Works Process for preparing of n-methyl-11-aza-10-deoxo-10-dihydroerythromycine a and derivatives thereof
US4474768A (en) * 1982-07-19 1984-10-02 Pfizer Inc. N-Methyl 11-aza-10-deoxo-10-dihydro-erytromycin A, intermediates therefor
SI9011409A (en) * 1990-07-18 1995-10-31 Pliva Pharm & Chem Works O-methyl azitromycin derivates, methods and intermediates for their preparation and methods for preparation of pharmaceuticals products which comprise them
HN1998000086A (es) * 1997-06-11 1999-03-08 Pfizer Prod Inc Derivados de 9 - desofo - 9 aza - 9a - homoeritromicina a - c - 4 sustituidos.
JP2003512290A (ja) * 1997-09-10 2003-04-02 メルク エンド カムパニー インコーポレーテッド 家畜抗菌剤としての８ａ−アザライド
UA70972C2 (ru) * 1998-11-20 2004-11-15 Пфайзер Продактс Інк. 13-членные азалиды и их применение как антибиотиков
DK1189912T3 (da) * 1999-05-18 2008-06-30 Pfizer Prod Inc Nye krystallinske former af et makrolid antibiotikum
US6465437B1 (en) * 1999-06-30 2002-10-15 Pfizer Inc. Diphosphate salt of a 4″-substituted-9-deoxo-9A-AZA-9A- homoerythromycin derivative and its pharmaceutical composition

Also Published As

Publication number Publication date
OA11965A (en) 2006-04-12
KR20020016875A (ko) 2002-03-06
CZ20014571A3 (cs) 2002-04-17
BR0012091A (pt) 2002-04-02
UA71013C2 (ru) 2004-11-15
EA004235B1 (ru) 2004-02-26
GT200000105AA (es) 2001-12-20
AU4943900A (en) 2001-01-22
EP1189913A1 (en) 2002-03-27
NO20016221D0 (no) 2001-12-19
AU772277B2 (en) 2004-04-22
TR200103834T2 (tr) 2002-05-21
US20030092642A1 (en) 2003-05-15
YU88701A (sh) 2004-09-03
PE20010287A1 (es) 2001-03-05
BG65587B1 (bg) 2009-01-30
SK286243B6 (sk) 2008-06-06
CO5190679A1 (es) 2002-08-29
NO20016221L (no) 2001-12-19
KR100442508B1 (ko) 2004-07-30
EP1189913B1 (en) 2005-01-12
PL201891B1 (pl) 2009-05-29
UY26221A1 (es) 2001-01-31
DE60017399D1 (de) 2005-02-17
BG106123A (en) 2002-05-31
US6465437B1 (en) 2002-10-15
US20040209826A1 (en) 2004-10-21
EA200101178A1 (ru) 2002-06-27
MXPA02000058A (es) 2002-07-02
CA2376748C (en) 2006-03-14
CN101220067A (zh) 2008-07-16
EE200100699A (et) 2003-02-17
US6861412B2 (en) 2005-03-01
US7297682B2 (en) 2007-11-20
PL352900A1 (en) 2003-09-22
HUP0201693A3 (en) 2003-03-28
HN2000000090A (es) 2001-04-20
AP2001002370A0 (en) 2001-12-31
ECSP003555A (es) 2002-01-25
GT200000105A (es) 2001-12-20
WO2001002414A1 (en) 2001-01-11
PA8496901A1 (es) 2002-08-26
IL146408A0 (en) 2002-07-25
AR035551A1 (es) 2004-06-16
CN1358188A (zh) 2002-07-10
DE60017399T2 (de) 2006-03-30
MY133360A (en) 2007-11-30
SK18922001A3 (sk) 2002-04-04
HUP0201693A2 (en) 2002-10-28
PT1189913E (pt) 2005-04-29
HRP20010919A2 (en) 2003-02-28
HRP20010919B1 (en) 2005-06-30
IS6159A (is) 2001-11-13
ATE286906T1 (de) 2005-01-15
EE05068B1 (et) 2008-08-15
ES2233380T3 (es) 2005-06-16
JP2003503506A (ja) 2003-01-28
CA2376748A1 (en) 2001-01-11
MA26745A1 (fr) 2004-12-20
TNSN00143A1 (fr) 2005-11-10

Similar Documents

Publication Publication Date Title
HUP0103406A3 (en) 1h-imidazopyridine derivatives and pharmaceutical compositions thereof
HUS1200028I1 (hu) 4"-Szubsztituált-9-dezoxo-9a-aza-9a-homoeritromicin-származékok és ezeket tartalmazó gyógyszerek
HUP0102990A3 (en) Tetrahydroimidazo-naphtyridine derivatives and pharmaceutical compositions thereof
HUP0100178A3 (en) Tetrahydro-naphtiridinyl-imidazolydinyl-carboxylic acid derivatives and pharmaceutical compositions thereof
IL149757A0 (en) Aminothiazole derivatives and pharmaceutical compositions containing the same
AU2319100A (en) Amide derivatives and drug compositions
HUP0001243A3 (en) Nicotinamide derivatives and pharmaceutical compositions containing them
HUP0103256A3 (en) Thiobenzimidazole derivatives and pharmaceutical compositions containing the compounds
HUP0200588A2 (hu) Diarilszármazékok és azokat tartalmazó gyógyszerkészítmények és alkalmazásuk
HUP0001494A3 (en) 3-phenoxy-, 3-dibenzo[a,d]cycloheptenyloxy-, 3-dibenz[b,f][1,4]oxazepinyloxy-1-amino-2-propanol derivatives and pharmaceutical compositions containing them
HUP0101381A3 (en) Benzofurylpyrone derivatives and pharmaceutical compositions containing them
HUP0103203A3 (en) Azaadamantane derivatives and pharmaceutical compositions thereof
IL147214A0 (en) 1-methylcarbapenem derivatives and pharmaceutical compositions containing the same
HUP9800147A3 (en) Isoxasol-and crotonoil-amide derivatives and pharmaceutical and diagnostical compositions containing them
HUP0105204A3 (en) Substituted phenethylamine derivatives and pharmaceutical compositions containing them
HUP0105075A3 (en) 3,3-biarylpiperidine and 2,2-biarylmorpholine derivatives, their use and pharmaceutical compositions containing them
HUP9801256A3 (en) 5'-deoxy-cytidine derivatives, preparation and use thereof and pharmaceutical compositions
IL148807A0 (en) Tetrahydrothiopyran derivatives and pharmaceutical compositions containing the same
IL139775A0 (en) A substituted triazolo-pyridazine derivative and pharmaceutical compositions made therefrom
HUP0002331A3 (en) 20-aralkyl-5alpha-pregnane derivatives and pharmaceutical compositions thereof
HUP9602196A2 (en) Sulfonyl- and sulfinyl-benzoyl-guanidine derivatives and pharmaceutical compositions thereof
HUP0102025A3 (en) Derivatives of 1,3,4-oxadiazolone, pharmaceutical compositions containing them and their use
HUP0001940A3 (en) Benzisothiazole derivatives, their use and pharmaceutical compositions containing them
HUP0003189A3 (en) Pharmaceutical composition comprising fexofenadine and its derivatives
ZA200110453B (en) Diphosphate salt of a 4"-substituted-9-deoxo-9a-aza-9a-homoerythromycin derivative and its pharmaceutical composition.